{"id":236,"date":"2013-06-18T16:42:01","date_gmt":"2013-06-18T07:42:01","guid":{"rendered":"http:\/\/www.keyton-co.jp\/kpharm\/byotai\/?page_id=236"},"modified":"2023-04-20T15:38:27","modified_gmt":"2023-04-20T06:38:27","slug":"research08","status":"publish","type":"page","link":"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/theme-list\/kinouseigazoushindanyaku\/research08\/","title":{"rendered":"\u304c\u3093\u306e\u75c5\u614b\u5206\u6790\u304b\u3089\u6cbb\u7642\u306b\u5411\u3051\u3066\u2460"},"content":{"rendered":"<h2 id=\"mt1\">\u70ad\u9178\u8131\u6c34\u9175\u7d20-IX \u3092\u6a19\u7684\u3068\u3057\u305f\u30bb\u30e9\u30ce\u30b9\u30c6\u30a3\u30af\u30b9\u85ac\u5264\u306e\u958b\u767a<\/h2>\n<p><span style=\"color: #000000\">\u85ac\u7269\u6cbb\u7642\u306e\u969b\u306b\u4f53\u5185\u52d5\u614b\u3068\u6a19\u7684\u9078\u629e\u6027\u306b\u3064\u3044\u3066\u3001\u753b\u50cf\u8a3a\u65ad\u85ac\u3068\u6cbb\u7642\u85ac\u3068\u306e\u9593\u306b\u5927\u304d\u306a\u4e56\u96e2\u304c\u5b58\u5728\u3059\u308b\u3053\u3068\u304c\u3042\u308a\u3001\u3055\u3089\u306b\u3001\u60a3\u8005\u306b\u3088\u3063\u3066\u85ac\u7269\u306e\u4f53\u5185\u52d5\u614b\u304c\u7570\u306a\u308b\u3053\u3068\u304c\u3001\u6cbb\u7642\u52b9\u679c\u306b\u591a\u5927\u306a\u5f71\u97ff\u3092\u4e0e\u3048\u3066\u3044\u308b\u3002\u4e00\u65b9\u3001\u753b\u50cf\u8a3a\u65ad(Diagnostics)\u3068\u6cbb\u7642(Therapeutics)\u3001\u305d\u308c\u305e\u308c\u306e\u30e2\u30c0\u30ea\u30c6\u30a3\u3092\u878d\u5408\u3057\u305f\u3082\u306e\u3068\u5b9a\u7fa9\u3055\u308c\u308b\u30bb\u30e9\u30ce\u30b9\u30c6\u30a3\u30af\u30b9(Theranostics)\u306f\u3001\u753b\u50cf\u8a3a\u65ad\u3068\u6cbb\u7642\u3092\u4e26\u884c\u3057\u3066\u884c\u3046\u3053\u3068\u3092\u53ef\u80fd\u3068\u3057\u3001\u60a3\u8005\u500b\u3005\u306e\u75c5\u6c17\u306e\u6027\u8cea\u3092\u7684\u78ba\u306b\u3068\u3089\u3048\u3001\u52b9\u679c\u7684\u306a\u6cbb\u7642\u3092\u7684\u78ba\u306b\u9032\u3081\u3066\u3044\u304f\u3053\u3068\u306b\u3088\u3063\u3066\u3001\u60a3\u8005\u306b\u5927\u304d\u306a\u5229\u76ca\u3092\u5bc4\u4e0e\u3059\u308b\u3053\u3068\u304c\u3067\u304d\u308b\u500b\u5225\u5316\u533b\u7642(\u30c6\u30fc\u30e9\u30fc\u30e1\u30a4\u30c9\u533b\u7642)\u306b\u7e4b\u304c\u308b\u3068\u8003\u3048\u3089\u308c\u308b\u3002<\/span><\/p>\n<p>&nbsp;<\/p>\n<p><a href=\"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-1.jpg\" class=\"liimagelink\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-2311\" src=\"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-1.jpg\" alt=\"\" width=\"1500\" height=\"1125\" srcset=\"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-1.jpg 1500w, https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-1-300x225.jpg 300w, https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-1-768x576.jpg 768w, https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-1-1024x768.jpg 1024w\" sizes=\"auto, (max-width: 1500px) 100vw, 1500px\" \/><\/a><\/p>\n<p><span style=\"color: #000000\">\u56fa\u5f62\u816b\u760d\u306b\u306f\u3001\u7d30\u80de\u5897\u6b96\u306b\u5bfe\u3057\u3066\u8840\u7ba1\u304b\u3089\u306e\u9178\u7d20\u4f9b\u7d66\u304c\u8ffd\u3044\u4ed8\u304b\u306a\u3044\u4f4e\u9178\u7d20\u9818\u57df\u304c\u5b58\u5728\u3059\u308b\u3002\u3053\u306e\u9818\u57df\u306f\u3001\u304c\u3093\u306e\u5316\u5b66\u7642\u6cd5\u3084\u653e\u5c04\u7dda\u6cbb\u7642\u306b\u5bfe\u3059\u308b\u62b5\u6297\u6027\u3092\u793a\u3057\u3001\u816b\u760d\u306e\u5897\u6b96\u30fb\u8ee2\u79fb\u306b\u95a2\u4e0e\u3059\u308b\u3068\u8003\u3048\u3089\u308c\u3066\u3044\u308b\u3002\u4e00\u65b9\u3001\u70ad\u9178\u8131\u6c34\u9175\u7d20-IX (CA-IX)\u306f\u4e8c\u9178\u5316\u70ad\u7d20\u3068\u6c34\u304b\u3089\u6c34\u7d20\u30a4\u30aa\u30f3\u3068\u70ad\u9178\u6c34\u7d20\u30a4\u30aa\u30f3\u3092\u7523\u751f\u3059\u308b\u751f\u4f53\u53cd\u5fdc\u3092\u89e6\u5a92\u3059\u308b\u9175\u7d20\u3067\u3042\u308a\u3001\u4f4e\u9178\u7d20\u304c\u3093\u7d30\u80de\u819c\u8868\u9762\u306b\u7279\u7570\u7684\u306b\u767a\u73fe\u3057\u3066\u3044\u308b\u3053\u3068\u304c\u77e5\u3089\u308c\u3066\u3044\u308b\u3002<\/span><\/p>\n<p><span style=\"color: #000000\">\u305d\u3053\u3067\u3001SPECT\u307e\u305f\u306f\u653e\u5c04\u6027\u540c\u4f4d\u5143\u7d20\u5185\u7528\u7642\u6cd5\u3092\u76ee\u7684\u3068\u3057\u3066<sup>111<\/sup>In\u307e\u305f\u306f<sup>90<\/sup>Y\u3092\u305d\u308c\u305e\u308c\u914d\u4f4d\u3055\u305b\u3001CA-IX\u306b\u5bfe\u3059\u308b\u7279\u7570\u7684\u89aa\u548c\u6027\u304c\u5831\u544a\u3055\u308c\u3066\u3044\u308b\u30a6\u30ec\u30a4\u30c9\u30b9\u30eb\u30db\u30f3\u30a2\u30df\u30c9\u8a98\u5c0e\u4f53\u30922\u5206\u5b50\u5c0e\u5165\u3057\u305f2\u4fa1\u653e\u5c04\u6027\u91d1\u5c5e\u932f\u4f53\u3067\u3042\u308b[<sup>111<\/sup>In]US2\u304a\u3088\u3073[<sup>90<\/sup>Y]US2\u3092\u8a2d\u8a08\u3057\u305f\u3002<\/span><\/p>\n<p>&nbsp;<\/p>\n<p><a href=\"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-2.jpg\" class=\"liimagelink\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-2313\" src=\"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-2.jpg\" alt=\"\" width=\"1500\" height=\"1125\" srcset=\"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-2.jpg 1500w, https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-2-300x225.jpg 300w, https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-2-768x576.jpg 768w, https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-2-1024x768.jpg 1024w\" sizes=\"auto, (max-width: 1500px) 100vw, 1500px\" \/><\/a><\/p>\n<p>&nbsp;<\/p>\n<p><span style=\"color: #000000\">CA-IX\u9ad8\u767a\u73fe\u816b\u760d\u79fb\u690d\u30e2\u30c7\u30eb\u30de\u30a6\u30b9\u306b[<sup>111<\/sup>In]US2\u3092\u6295\u4e0e\u3057\u3001SPECT\u64ae\u50cf\u3092\u884c\u3063\u305f\u3068\u3053\u308d\u3001\u816b\u760d\u3092\u9078\u629e\u7684\u304b\u3064\u660e\u77ad\u306b\u30a4\u30e1\u30fc\u30b8\u30f3\u30b0\u3059\u308b\u3053\u3068\u306b\u6210\u529f\u3057\u305f\u3002\u7d9a\u3044\u3066\u3001[<sup>90<\/sup>Y]US2\u3092\u30e2\u30c7\u30eb\u30de\u30a6\u30b9\u306b\u6295\u4e0e\u3057\u305f\u3068\u3053\u308d\u3001\u751f\u7406\u98df\u5869\u6c34\u6295\u4e0e\u7fa4\u3068\u6bd4\u8f03\u3057\u3066\u3001\u30de\u30a6\u30b9\u751f\u5b58\u671f\u9593\u304c\u6709\u610f\u306b\u5ef6\u9577\u3057\u305f\u3002\u3053\u308c\u3089\u306e\u7d50\u679c\u3088\u308a\u3001[<sup>111<\/sup>In]US2\u304a\u3088\u3073[<sup>90<\/sup>Y]US2\u306f\u3001CA-IX\u3092\u6a19\u7684\u3068\u3057\u305f\u56fa\u5f62\u816b\u760d\u306e\u753b\u50cf\u8a3a\u65ad\u304a\u3088\u3073\u6cbb\u7642\u3092\u53ef\u80fd\u3068\u3059\u308b\u3053\u3068\u304c\u793a\u3055\u308c\u3001\u304c\u3093\u306e\u30bb\u30e9\u30ce\u30b9\u30c6\u30a3\u30af\u30b9\u306b\u6709\u7528\u3067\u3042\u308b\u3053\u3068\u304c\u793a\u3055\u308c\u305f\u3002<\/span><\/p>\n<p>&nbsp;<\/p>\n<p><a href=\"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-3.jpg\" class=\"liimagelink\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-2315\" src=\"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-3.jpg\" alt=\"\" width=\"1500\" height=\"1125\" srcset=\"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-3.jpg 1500w, https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-3-300x225.jpg 300w, https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-3-768x576.jpg 768w, https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/files\/2018\/08\/CA9-3-1024x768.jpg 1024w\" sizes=\"auto, (max-width: 1500px) 100vw, 1500px\" \/><\/a><\/p>\n<h3>\u4e3b\u8981\u8ad6\u6587<\/h3>\n<ul>\n<li><span class=\"Apple-style-span\">Development of <sup>99m<\/sup>Tc-Hydroxamamide Complex as Probe Targeting Carbonic Anhydrase IX<br \/>\n<em>Mol Pharm<\/em>\u00a016(4) 1489-1497 (2019)<\/span><\/li>\n<li><span class=\"Apple-style-span\">Cancer radiotheranostics targeting carbonic anhydrase-IX with <sup>111<\/sup>In- and <sup>90<\/sup>Y-labeled ureidosulfonamide scaffold for SPECT imaging and radionuclide-based therapy<br \/>\n<em>Theranostics<\/em>\u00a08(11) 2992-3006\u00a0(2018)<\/span><\/li>\n<\/ul>\n<p>&nbsp;<\/p>\n","protected":false},"excerpt":{"rendered":"<p>\u70ad\u9178\u8131\u6c34\u9175\u7d20-IX \u3092\u6a19\u7684\u3068\u3057\u305f\u30bb\u30e9\u30ce\u30b9\u30c6\u30a3\u30af\u30b9\u85ac\u5264\u306e\u958b\u767a \u85ac\u7269\u6cbb\u7642\u306e\u969b\u306b\u4f53\u5185\u52d5\u614b\u3068\u6a19\u7684\u9078\u629e\u6027\u306b\u3064\u3044\u3066\u3001\u753b\u50cf\u8a3a\u65ad\u85ac\u3068\u6cbb\u7642\u85ac\u3068\u306e\u9593\u306b\u5927\u304d\u306a\u4e56\u96e2\u304c\u5b58\u5728\u3059\u308b\u3053\u3068\u304c\u3042\u308a\u3001\u3055\u3089\u306b\u3001\u60a3\u8005\u306b\u3088\u3063\u3066\u85ac\u7269\u306e\u4f53\u5185\u52d5\u614b\u304c\u7570\u306a\u308b\u3053\u3068\u304c\u3001\u6cbb\u7642\u52b9\u679c [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"parent":135,"menu_order":0,"comment_status":"closed","ping_status":"closed","template":"","meta":{"_crdt_document":"","footnotes":""},"class_list":["post-236","page","type-page","status-publish","hentry"],"_links":{"self":[{"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/wp-json\/wp\/v2\/pages\/236","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/wp-json\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/wp-json\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/wp-json\/wp\/v2\/users\/1"}],"replies":[{"embeddable":true,"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/wp-json\/wp\/v2\/comments?post=236"}],"version-history":[{"count":6,"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/wp-json\/wp\/v2\/pages\/236\/revisions"}],"predecessor-version":[{"id":2913,"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/wp-json\/wp\/v2\/pages\/236\/revisions\/2913"}],"up":[{"embeddable":true,"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/wp-json\/wp\/v2\/pages\/135"}],"wp:attachment":[{"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/byotai\/wp-json\/wp\/v2\/media?parent=236"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}