14) | öèœ, oFü, Rc׬, ÖûI, A£Pv, ì£M, Ò €, qij, |JGº, FiÈO, ºÔum. PBrJÆx»ÜL-FDLDAðp¢œ®šíÌÙÈéH÷ÌC~_][Wyv`hÆÖA»šÌèʪÍ@Ìm§. æ79ñú{h{EHÆwïåï, €m, 5, 2025. @ |
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13) | Rc׬, öè œ, A£Pv, rcŸÄ¢, qij,@|JGº, ºÔum. ŽxU±Ì»òD-FDLDAðp¢œ¯ÊÌW¯U±Ì»@Éæé¶ÌA~šæÑOìÌA~m_ÌèÊ. æ79ñú{h{EHÆwïåï, €m, 5, 2025. @ |
12) | |JGº. ú{òwïÜEóÜuFnòðuüµœVRšP~JoCIW[€. ú{òwïæ145Nïiªj, ª, 3, 2025. ióÜuj@ |
11) | |JGº. V|WEumgTCGX@AbvgDfCgvFhmghðîÕƵœVRšnòP~JoCIW[. ú{òwïæ145Nïiªj, ª, 3, 2025. iµÒuj@ |
10) | Oº@Ò, rcñd, ÄèçO, ühå÷, Ž{ºq, VÆêj, ä{³Æ, |JGº. VKªñ²×EXtFA`¬jQÜXgvgXtFA̶Y«üãÆVKÞÌÌ©. ú{òwïæ145Nïiªj, ª, 3, 2025. |
9) | úåàVaó, àq«î, rcñd, âcÀ, ºúÆ, zìLá, ·öìfÔ, n i, ŒºTê, V¢®ç, öGN, |JGº. úüÛÌ¡|{ÉæèY¶³êéVKsmitgLmn»šÌP£E\¢ðÍÆ»ÌY¶ÉÖ·é€. ú{òwïæ145Nïiªj, ª, 3, 2025. |
8) | Zhang, L., Pan, Y., Ÿ, AGT, œìGT, |JGº. ^ÛStachybotrys®ª¶Y·éVK€L«AXpM¬yfjQÜÌJ€. ú{òwïæ145Nïiªj, ª, 3, 2025. |
7) | ŒäüRó, rcñd, ÄèçO, âäaq, Œöal, ä{³Æ, |JGº. ªñ²×EXtFA`¬jQ«ðL·éúüÛãÓYšÌ©Æìp@ðÍ. ú{òwïæ145Nïiªj, ª, 3, 2025.@ |
6) | rcñd, ä§å, ¡{ØXq, ¬ÑŽ, ü]ê_, Žc _, |JGº. «Ÿ³¡ÃÉš¯éPKC¿/mTORCVOiðHIF-1¿«»íª. ú{òwïæ145Nïiªj, ª, 3, 2025.@ |
5) | n i, Ž{ œ, Îìa÷, F{ìÆ, |JGº, s£_u. AN`mW¶¬ÉÖ^·éVK_»yfActVA-ORF3ÌAlphaFoldðpµœ@\ðÍ€. ú{òwïæ145Nïiªj, ª, 3, 2025.@ |
4) | ª{«j, Xcåã, HtG÷, Ÿ Ln@l, |JGº, åì_Í, äÑWã. ¿ŽñŠ^pN¿CD1aÉF¯³êé|yv`hDDM-838Ì\¢«Ö€. ú{òwïæ145Nïiªj, ª, 3, 2025.@ |
3) | Kakeya, H. Natural product-inspired chemical biology: Development of an agrochemical seed targeting the scab-forming actinomycete. Asian Chemical Biology Initiative (ACBI) 2025 Hanoi Meeting, Hanoi, Vietnam, Jan. 2025. (invited) |
2) | Kakeya, H. Natural product-inspired chemical biology: Development of highly sensitive labeling reagents for amino acids, scarce natural products, and amylooid beta fragment peptides. The 5th Intenational Conference on Natural Product Discovery and Development in the Genomic Era. San Diego, CA, USA, Jan. 2025. |
1) | Yanagisawa, K., Kaneko, K., Ikeda, H., Iwata, S., Muranaka, A., Koshino, H., Nagao, N., Watari, S., Nishimura, S., Shinzato, N., Onaka, H., Kakeya, H. Discovery of a new pyranonaphthoquinone, actinoquinonal A: Combined-culture of Streptomyces sp. 23-50 with Tsukamurella pulmonis TP-B0596 triggers a shunt of the mevalonate pathway of Streptomyces sp. 23-50. The 5th Intenational Conference on Natural Product Discovery and Development in the Genomic Era. San Diego, CA, USA, Jan. 2025. [DG\Üi|X^[\)FThe Carol D. Litchfield Honorable Mention Student Poster Presentation] |
33) | öèœ, oFü, ÖûI, A£Pv, ì£M, Ò €, qij, |JGº, FiÈO, ºÔum. PBrJÆx»ÜL-FDLDAðp¢œH÷ÌC~_][Wyv`hÆÖA»šÌèÊ. æ14ñVA~m_ªÍ€ï, , 12, 2024. @ |
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32) | Rc׬, öè œ, A£Pv, rcŸÄ¢, qij,@|JGº, ºÔum. Žxx»ÜD-FDLDAðp¢œr[̶ÌA~ÞšæÑÖA»šÌêĪÍ. æ14ñVA~m_ªÍ€ï, , 12, 2024. @ |
31) | ühå÷, qij, gc¹», ¬R €, rcñd, ÄèçO, |JGº. VKªñ²×EXtFA`¬jQÜXgvgXtFAÌ\¢èyÑS¬€. æ41ñfBViP~Xg[V|WE, s, 11, 2024. |
30) | ª{«j, Xcåã, HtG÷, Ÿ Ln@l, |JGº, åì_Í, äÑWã. CD1aS©«T×Eð§ä·éjÛR|yv`hDDM-838Ì\¢«Ö€. æ41ñfBViP~Xg[V|WE, s, 11, 2024. |
29) | Zhang, L., Pan, Y., Hattori, A., Uekusa, H., Kakeya, H.Discovery of new meroterpenoids produced by Stachybotrys ruwenzoriensis RF-6853 as asparagine synthetase inhibitors. Seoul Univ.-Kyoto Univ.-Osaka Univ. Symposium 2024 (SKO Symposium 2024). Seoul, Korea, Nov., 2024. |
28) | Rc׬, öèœ, ºÔum, rcŸÄ¢, qij, |JGº, A£Pv. Žxx»ÜD-FDLDAðp¢œr[Ì sA~ÞšæÑÖA»šÌêĪÍ. æ120ñú{Hiq¶wïwpuï, €m, 11, 2024. |
27) | öèœ, oFü, ÖûI, ºÔum, ì£M, Ò €, qij, |JGº, FiÈO,@A£Pv. x»ÜL-FDVDAÆPBrJðp¢œ®šíEgDEiíÌÙÈéH÷ÌC~_][Wyv`hÆ\¬A~m_A^EÌèʪÍ. æ120ñú{Hiq¶wïwpuï, €m, 11, 2024. |
26) | öèœ, oFü, rcŸÄ¢, qij, |JGº, A£Pv. Žxõwªx»ÜL-FDLDAðp¢œyHiEù¿ÌDL-A~m_ÌèʪÍ@ÌJ. æ120ñú{Hiq¶wïwpuï, €m, 11, 2024. |
25) | Kakeya, H., Pan, Y., Zhang, L., Suzuki, T., Sakai, K., Hirano, Y., Ikeda, H., Hattori, A., Dohmae, N., Nishio, K. Identification and a mode of action of bisabosqual A, a novel asparaginase synthetase (ASNS) inhibitor, towards the development of molecular-targeted anticancer drug. 36th EORTC-NCI-AACR Symposium on Molecular Targets and Cancer Therapeutics. Barcelona, Spain, Oct. 2024. (EORTC, the European Organization for Research and Treatment of Cancer; NCI, the National Cancer Institute; AACR, the American Association for Cancer Research) |
24) | úåàVaó, àq«î, rcñd, âcÀ, ºúÆ, zìLá, ·öìfÔ, n i, ŒºTê, V¢®ç, öGN, |JGº. úüÛÌ¡|{Æ^{[ðÍÉæéVKRªñÜV[YÌJ€. æ74ñú{òwïÖŒxïEåï, ºÉ, 10, 2024.[DGÜ]@@ |
23) | rcñd, ì©ü¢, ÄèçO, Oº Ò, |JGº. ªñ²×EðWIÆ·é÷¶šñãÓYšÌ©Æìp@ðÍ. æ74ñú{òwïÖŒxïEåï, ºÉ, 10, 2024.@ |
22) | ¬R €, qij, X{ÁŸ, Œ³ñC, |JGº. ˶ê^A~hðyv`h¬@ÌJƪqÂóyv`h¬ÖÌp. æ74ñú{òwïÖŒxïEåï, ºÉ, 10, 2024. [DGÜ]@ |
21) | Ikeda, H., Iseki, S., Kobayashi, S., Irie, K., Harada, H., Kakeya, H. Upregulation of HIF-1¿ via the PKC¿/mTORC signaling pathway is a potential therapeutic strategy for ishemia-related diseases. The 4th network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
20) | Furutani, Y., Tanaka, K., Nagamori, S., Kobayashi, K., Aizaki, H., Ochi, S., Kakeya, H., Matsuura, T. Development of cccDNA modulators, CDMs, that specifically activate interferon-related signals and inhibit HBV replication. 2024 International HBV Meeting: Biology of the Hepatitis B and Viruses. Chicago, IL, USA, Sep. 2024@ |
19) | öèœ, oFü, ÖûI, ºÔum, ì£M, Ò €, qij, |JGº, FiÈO,@A£Pv. x»ÜL-FDVDAÆPBrJðp¢œ®šíEgDEiíÌÙÈéH÷ÌC~_][Wyv`hÆ\¬A~m_A^EÌêĪÍ. ú{A~m_wïæ18ñwpåïiJSAAS2024j, éÊ, 9, 2024. |
18) | ¿cV¬, rcñd, qij, ¥èR¢, àN³ª, Jû§, V¢®ç, öGN, |JGº. VKAmCLXU±ÜALZ^~hAÌP£E\¢ðÍyÑS¬. æ66ñVRL@»š¢_ï, s, 9, 2024. |
17) | àq«î, O}{Ô, Yulu Jiang, ŽLŸ, |JGº. AšaQ»€©aŽöÛðWIÆ·é_òV[YJ€FcZi~hCÌ©Æìp@ðÍ. æ66ñVRL@»š¢_ï, s, 9, 2024. |
16) | Kakeya, H. Natural product-inspired chemical biology: Development of highly sensitive labeling reagents for amino acids and scarce natural products. International Congress on Natural Products Research 2024 (ICNPR 2024), Krakow, Poland, Jul. 2024.@@ |
15) | úåàVaó, àq«î, rcñd, âcÀ, ºúÆ, zìLá, ·öìfÔ, n i, ŒºTê, V¢®ç, öGN, |JGº. úüÛÌ¡|{ÉæéVKRªñÜV[YÌJ€. æ34ñVòn»kbï, ÈØ, 7, 2024. [€§ãÜ]@@@ |
14) | rcñd, ä{³Æ, |JGº. ªñ²×EðWIÆ·ém}CV̯èEìp@. æ28ñú{ªñªqWI¡Ãwï, , 6, 2024.@@ |
13) | Furutani, Y., Kakeya, H., Matsuura, T. Development of novel small molecules that activate innate immunity and inhibit HBV replication. The 60th Annual Meeting of the Japan Society of Hepatology, Kumamoto, Jun, 2024. |
12) | àq«î, O}{Ô, Yulu Jiang, ŽLŸ, |JGº. úüÛãÓYšcZi~hCÌR»€©aŽöÛ«Æ»ÌÏ«»ªàœç·j[NÈ\»^É¢Ä. ú{P~JoCIW[wï@æ18ñNï, , 5, 2024. |
11) | Kakeya, H. Separation and identification of the D/L-forms of amino acids and short-chain peptides using highly sensitive labeling reagents for research of cardiovascular disease. The 9th Annual Scientific Meeting of JCVA (Japan Cardiovascular Association), Shizuoka, May 2024. |
10) | öè œ, oFü, ºÔum, ì£M, Ò@€, qij, |JGº, FiÈO, A£Pv. Žxx»ÜL-FDVDAÆPBrJðp¢œHiÌC~_][Wyv`hÆ\¬A~m_A^EÌêĪÍ. æ78ñú{h{EHÆwïåï, ª, 5, 2024. |
9) | Ý{[O, ¬©RI, ac[¹, óŽNq, RAê, öèT, ÂRL÷, YÛG, ¡òú, Ž{³, »ìzê, X{Bç, àäëj, |JGº, ·Jì_ñ. ³ÇóEyÇÌV^RiECXŽõdzÒÉš¯éoûzûNN~iNN[W jÌÇÖÌiW}§øÊðØ·évZ{ÎÆñdÓ³ì×»är±. ú{òwïæ144Nïi¡lj, ¡l, 3, 2024.@@ |
8) | ühå÷, qij, gc¹», rcñd, ÄèçO, |JGº. VKªñ²×EXtFA`¬jQÜXgvgXtFAÌS¬€. ú{òwïæ144Nïi¡lj, ¡l, 3, 2024. |
7) | ¿cV¬, qij, ¥èR¢, rcñd, àN³ª, |JGº. VKAmCLXU±ÜALZ^~hAÌ®S\¢èyÑS¬€. ú{òwïæ144Nïi¡lj, ¡l, 3, 2024. |
6) | àc®, qij, 真Y, |JGº. VKR^ÛÜAtBI[ÌS¬€. ú{òwïæ144Nïi¡lj, ¡l, 3, 2024. |
5) | rcñd, ÄèçO, ªcÊG, DRÀã, ühå÷, gc¹», qij, V¡êq, ~øêv, ä{³Æ, |JGº. VKªñ²×EXtFA`¬jQÜXgvgXtFAÌP£E\¢ðÍ. ú{òwïæ144Nïi¡lj, ¡l, 3, 2024. |
4) | |JGº. VRšnòP~JoCIW[ðîÕƵœªqWIRªñÜJ€. ªñ¡ÃCmx[VÉü¯Ä. såw€@Eš¿E×E_@ÊqimãÀZ^[, s, 3, 2024.iµÒuj |
3) | Kakeya, H. Natural products-inspired chemical biology-Development of a novel asparagine synthetase inhibitor for cancer chemotherapy-, Asian Chemical Biology Initiative (ACBI) 2024 Istanbul Meeting, Istanbul, Turkey, Mar. 2024. iinvitedj@@ |
2) | Matsuoka, T., Hattori, A., Oishi, S., Araki, M., Ma, B., Fujii, T., Arichi, N., Okuno, Y., Kakeya, H., Yamasaki, S., Ohno, H., Inuki, S. Establishment of an MR1-presentation reporter screening system to identify MAIT cell modulation. CD1-MR1 2024, Tasmania, Australia, Feb., 2024. |
1) | öè œ, ºÔum, qij, |JGº, A£Pv, . Žxõwªx»ÜL-FDVDAðp¢œ¶Ì¿EHi©çÌA~m_ÌŽxªÍ@Ìm§. æ15ñJapan@Bioanalysis Forum (JBF) V|WE, s, 3, 2024. |
37) | Kakeya, H. Natural products-inspired chemical biology-Development of highly sensitive labeling reagents-, Asian Chemical Biology Initiative (ACBI) 2023 Kuala Lumpur Meeting, Kuala Lumpur, Malaysia, Dec. 2023. iinvitedj |
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36) | |JGº, VRšnòP~JoCIW[FVKA~m_Eyv`hªÍ@ÌJÆp. æ13ñVA~m_ªÍ€ï, , 12, 2023. iµÒuj@@ |
35) | A£Pv, öè œ, oFü, ºÔum, rcŸÄ¢, qij, |JGº. Žxõwªx»ÜD-FDLDAðp¢œyHiÌDL-A~m_ªÍ. æ13ñVA~m_ªÍ€ï, , 12, 2023. |
34) | öè œ, ºÔum, qij, |JGº, A£Pv. Žxõwªx»ÜL-FDVDAðp¢œA~m_Ì\¢Ù«ÌÆõwÙ«ÌÌêĪÍ. êĪÍ@Ìm§. æ13ñVA~m_ªÍ€ï, , 12, 2023. |
33) | Sun, Y., Hashizume, D., Kakeya, H. Synthetic study of 2-(1H-imidazole-4-yl)-1,3,4-oxadiazole scaffolds for pharmaceuticals. The 40th Medicinal Chemistry Symposium. Nagoya, Nov., 2023. |
32) | Koyama, A., Kuranaga, T., Morimoto, R., Matsumoto, T., Kakeya, H. Acyl sulfonamide-mediated amidation and its application to the synthesis of middle molecular natural peptidic molecules. The 60th Japanese Peptide Symposium, Shiga, Nov. 2023. |
31) | Kuranaga, T., Morimoto, R., Pan, C., Ogawa, H., Kakeya, H. Design, synthesis, and application of highly sensitive labeling reagent for amino acids. The 60th Japanese Peptide Symposium, Shiga, Nov. 2023. |
30) | Ozaki, M., Shimotsuma, M., Kuranaga, T., Kakeya, H., Hirose, T. Identification of DL-amino acids containing threonine and isoleucine stereoisomers in peptides using an original chiral resolution labeling reagent. The 60th Japanese Peptide Symposium, Shiga, Nov. 2023. |
29) | |JGº. VRšP~JoCIW[ðîÕƵœnãòÈw€. æ9ñòwÌ¢ðlŠésV|WEFnãòÈwêUJwLOV|WE, s, 11, 2023. iµÒuj |
28) | Pan, Y., Suzuki, T., Sakai, K., Hirano, Y., Ikeda, H., Hattori, A., Dohmae, N., Nishio, K., Kakeya, H. Identification of an asparagine synthetase inhibitor bisabosqual A as an anticancer seed. The 3rd network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
27) | Kodama, K., Ikeda, H., Shibasaki, M., Kawami, M., Imoto, M., Kakeya, H. Screening and identification of anticancer lead compounds through a novel strategy targeting cancer stem cells. The 3rd network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
26) | Kakeya, H., Ozaki, M., Shimotsuma, M., Kuranaga, T., Hirose, T. Development of a new chiral resolution labeling reagent and aplication to separation of amyloid b fragment peptides with racemized and isomerized aspartic acid residues. The 3rd network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
25) | Koyama A., Kuranaga, T., Morimoto, R., Matsumoto, T., Kakeya, H. A novel peptide C-terminal modification and its application to the synthesis of middle molecular cyclic peptides. The 3rd network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
24) | Sun, Y., Hashizume, D., Kakeya, H. Studies on 2-(1H-imidazol-4-yl)-1,3,4-oxadiazole scaffolds for pharmacological molecules. The 3rd network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
23) | A£Pv, öè œ, oFü, ºÔum, qij, |JGº. Žxõwªx»ÜD-FDLDAðp¢œHiÌDL-A~m_ªÍ. ú{A~m_wïæ17ñwpåï (JSAA2023), ª, 9, 2023. |
22) | öè œ, ºÔum, qij, |JGº, A£Pv, . Žxõwªx»ÜL-FDVDAðp¢œSA~m_êĪÍ@Ìm§. ú{A~m_wïæ17ñwpåï (JSAA2023), ª, 9, 2023. |
21) | oFü, öè œ, ºÔum, qij, |JGº, A£Pv. õwªx»ÜL-FDVDAðp¢œyv`hÌThrÆIlȩÌÙ«Ì̯è. ú{A~m_wïæ17ñwpåï (JSAA2023), ª, 9, 2023. |
20) | ¬R €, qij, X{ÁŸ, Œ³ñC, |JGº. Gs»ð}§·éyv`hC[Cü@ƪqÂóyv`h¬ÖÌp. æ65ñVRL@»š¢_ï, , 9, 2023.@@@@@.@@ |
19) | Ê J, rcñd, ÄèçO, ì©ü¢, ä{³Æ, |JGº. ªñ²×EðWIƵœRªñÜV[YÌJ€. æ33ñVòn»kbï. s, 9, 2023. [€§ãÜ]@@ |
18) | ¬R €, qij, X{ÁŸ, Œ³ñC, |JGº. ªqyv`hnòðuüµœVKyv`h¬@ÌJ. æ33ñVòn»kbï, s, 9, 2023.@@@@@.@@ |
17) | ŒªñN, Ÿ, åÎ^ç, rØ]k, Ln@l, |JGº, Rè », åì_Í, äÑWã. ×E\ÊÌMR1¶ÝÊÉîÃKhXN[jO@ÌJÆMAIT×E§äªq̯è. æ65ñVRL@»š¢_ï, , 9, 2023.@@@@@.@@ |
16) | Yanaka, K., Hirano, Y., Qiun, X.Y., Suzuki, H., Kakeya, H., Matsuura, T., Furutani, Y. A small chemical compound iCDM-34 identified by an in silico screening suppresses HBV DNA through activation of aryl hydrocarbon receptor, 2023 Interbational HBV Meeting, Kobe, Sep. 2023.@@@.@@ |
15) | |JGº. P~JoCIW[ð@²Æµœªqvt@CO, 2023NxáèxZpuKï, ¶ÈwÈwpÏv€ wp€xîÕ`¬ æ[f®šxvbgtH[iADAMsj, ŒÃ®, 9, 2023. iµÒuj |
14) | |JGº. VRšnòP~JoCIW[ÌÅOüFYwAgÉæéãòiÌÀp»Éü¯Ä, sCmx[Vp[Nð¬Z~i[iåÃFsT[`p[Nj, åã, 7, 2023. iµÒuj |
13) | |JGº. V|WE1EuWIð˲¯IiáªqEªqERÌjv\VRšnòFAXpM¬yfð˲. æ27ñú{ªñªqWI¡ÃwïwpWï, ²ê, 6, 2023. iµÒuj |
12) | Pan, Y., Suzuki, T., Sakai, K., Hirano, Y., Ikeda, H., Hattori, A., Dohmae, N., Nishio, K., Kakeya, H. Identification of bisabosqual A as an asparagine synthetase (ASNS) inhibitor towards the development of molecular-targeted anticancer drug. The 17th Annual Meeting of Japanese Society for Chemical Biology, Osaka, May, 2023. |
11) | Kakeya, H. Development of an innovative anticancer drug TBP1901, an injectable prodrug of curcumin. 2023 NSFC*1-JSPS-CAS*2 Forum: Translational Medicine and Innovative Drug Research. Tianjin, China, Jun. 2023. (*1 Natural Science Foundation of China, *2 Chinese Academy of Science) [keynote lecture] |
10) | ŒªñN, Ÿ, åÎ^ç, Ln@l, |JGº, Rè », åì_Í, äÑWã. MR1Ì×E\ÊÊðwWÆ·éKhXN[jO@ÌJÆMAIT×EW [^[̯è. ú{P~JoCIW[wï@æ17ñNï, åã, 5, 2023.@@ |
9) | Pan, Y., Suzuki, T., Sakai, K., Hirano, Y., Ikeda, H., Hattori, A., Dohmae, N., Nishio, K., Kakeya, H. Screening and identification of an asparagine synthetase (ASNS) inhibitor as a molecular-targeted anticancer drug. The 143rd Annual Meeting of Pharmaceutical Society of Japan. Hokkaido, Mar. 2023.@@@@@ |
8) | öè œ, ºÔum, qij, |JGº, A£Pv. DL-A~m_x»Lbgðp¢œA~ChÀÌAspcîÌZ~»EÙ«»Ìo@ÌJ\Ÿ³ÉÖ^·éÃW^pN¿Eyv`hÌúffEŸ³JjYÌðŸÉü¯Ä\. æ14ñJapan@Bioanalysis Forum (JBF) V|WE, , 3, 2023. |
7) | Ikeda, H., Shibasaki, M., Kodama, K., Kawami, M., Imoto, M., Kakeya, H. Screening for anticancer lead compounds through a new strategy for targeting cancer stem cells. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
6) | Sun, Y., Hashizume, D., Kakeya, H. Synthetic study on 2-(1H-imidazol-4-yl)-1,3,4-oxadiazole scaffolds for drug discovery. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
5) | Kuranaga, T., Tamura, M., Ikeda, H., Terada, S., Nakagawa, Y., Kakeya, H. Reactivity-guided identification and total synthesis of an unstable anticancer macrolide presaccharothriolide Z. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
4) | Kakeya, H., Abe, T., Horisawam Y., Kikuchi, O., Ozawa-Umeta, H., Kishimoto, A., Imaizumi, A., Hashimoto, T., Shirakawa, K., Takaori-Kondo, A., Yusa, K., Asakura, T., Kanai, M. Pharmacologic characterization of TBP1901, an innovative prodrug form of curcumin, and CRISPR-Cas9 screen for therapeutic targets of curcumin. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
3) | Koyama, A., Kuranaga, T., Morimoto, R., Kakeya, H. Acyl sulfamide-mediated amidation for biomimetic peptide synthesis. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
2) | Pan, Y., Suzuki, T., Sakai, K., Hirano, Y., Ikeda, H., Hattori, A., Dohmae, N., Nishio, K., Kakeya, H. Chemical biology research on an asparagine synthetase (ASNS) inhibitor as a molecular-targeted anticancer drug. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
1) | Àc õ, |àV³Ÿ, qij, |JGº. VKU±Ì»òðp¢œD,L-A~m_ÌŽxªÍ@J. æ28ñLC&MSeNmvU, ICJÃ, 1, 2023. [xXgv[e[VÜixXge[}Üj] |
15) | öè œ, ºÔum, qij, |JGº, A£Pv. õwªx»ÜD-FDLDAðp¢œA~ChÀÌAXpM_cîÌZ~»EÙ«»Ì¯è. VA~m_ªÍ€ïæ12ñwpuï, , 12, 2022. [DG\Ü] |
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14) | Àc õ, |àV³Ÿ, qij, |JGº. VKU±Ì»òðp¢œ¶Ì¿yÑ×E|{ãŽD,L-A~m_ÌŽxªÍ. VA~m_ªÍ€ïæ12ñwpuï, , 12, 2022. |
13) | Yasuda, Y., Takezawa, M., Kuranaga, T., Kakeya, H. Highly sensitiveanalysis of D-and L-amino acids in biological samples using new derivatization reagents. The 37th Annual Meeting of the Japanese Society for the study of Xenobiotics, Kanagawa, Nov. 2022.@ |
12) | ŒªñN, Ÿ, åÎ^ç, Ln@l, |JGº, Rè », åì_Í, äÑWã. XvbgVtF[[ðpµœXN[jO@ÉæéVKMR1Kh̯èÆ»Ì\¢«Ö€. æ39ñfBViP~Xg[V|WE, 11, 2022, ICJÃ.@@@@@ |
11) | Ozaki, M., Shimotsuma, M., Kuranaga, T., Kakeya, H., Hirose, T. Identification of DL-and DL-iso-form of aspartic acid residues in amyloid b peptide using a chiral resolution labeling reagent. The 59th Japanese Peptide Symposium, Miyagi, Oct. 2022. |
10) | Ikeda, H., Imoto, M., Kakeya, H. Identification of the polyether ionophore lenoremycin through a new screening strategy targeting cancer stem cells. The 81st Annual Meeting of the Japanese Cancer Association. Kanagawa, Sep. 2022. [selected as a late-breaking poster]@@@@@ |
9) | Kura, Y., Develasco, M.A., Sakai, K., Fujita K., Bannno, E., Fujita, Y., Hashimoto, M., Nishimoto, M., Nozawa, M., Yoshimura, K., Kakeya, H., Umemura, H., Nishio, K. Chemopreventive potential of curcumin monoglucuronide in mouse Pten-null prostate cancer. The 81st Annual Meeting of the Japanese Cancer Association. Yokohama, Sep. 2022.@@@@@ |
8) | qij, cºü¿, rcñd, c V, ìYî, |JGº. »w¬ðìgµœóRªñ«VRšvTbJXIhZ̯è. æ64ñVRL@»š¢_ï, ê, 9, 2022.@@@@@ |
7) | |JGº, qij, rcñd, Ÿ, ŒºTê, ä{³Æ. ÷¶šÔ»wR~ jP[VÌðÆLp¶š«KhÌJ. VwpÌæ€u»wR~ jP[VÌteBAvæèÜÆßV|WE, s, 7, 2022. |
6) | |JGº. VRšnòP~JoCIW[ÌÅOü. k¢åwæ100ñKMCFZ~i[iKitasato Microbial Chemistry Frontierj, , 6, 2022. iµÒuj |
5) | Îì¶m, àcç°, åŒÞ, ¡ìãÄ, éØT, P, °OŒ, |JGº, cç³³O. ×EàÅÌñ{\[yv`h¬yfÌIðIx»šæѪð@\Ì©. ú{P~JoCIW[wï@æ16ñNï, xR, 5, 2022.@@ |
4) | ²XØá, ŒºTê, ŒRWv, ªãczq, |JGº, gc«. FKBP12ÉæéZEXIjãÓ§äÌ»wâ`wIðÍ. ú{_|»wï2022Nxåï, siICj, 3, 2022. |
3) | Îì¶m, ¡ìãÄ, àcç°, éØT, P, °OŒ, |JGº, cç³³O. ×EàÅÌñ{\[yv`h¬yfÌIðIP~JxOšæѪðßöÌ©. ú{òwïæ142Nï. ŒÃ®iICj, 3, 2022.@@ |
2) | Watari, S., Kaneko, K., Iwata, S., Nagao, N., Onaka, H., Shinzato, N., Kakeya, H. Syetematic screening of new microbial metabolites by combined-culture of actinomycetes. Japan-the Netherlands Microbiology Symposium 2022, Mar. 2022 (Kochi/on-line).@@@@@ |
1) | Kakeya, H. Chemical communication research on microbes toward the development of novel antibiotics. Japan-the Netherlands Microbiology Symposium 2022, Mar. 2022 (Kochi/on-line). (Invited lecture)@@@@@ |
18) | Kakeya, H. Chemical communication research toward the development of novel antibiotics. (#182 Antibiotics Discovery), PACIFICHEM2021, Hawaii, USA, Dec. 2021. (Invited lecture)@@@@ |
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17) | Kakeya, H. Chemical communication research toward the development of new anticancer drugs. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
16) | Omura, S., Khadka, S., Sato, F., Nakamura, Y., Nishio, K., Kakeya, H., Tsunoda, I. Curcumin mooglucuronide (CMG) treatment alters the gut microbiota, regulating an autoimmune model for multiple sclerosis. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
15) | Ikeda, H., Muroi, M., Kondoh, Y., Ishikawa, S., Kakeya, H., Osada, H., Imoto, M. Miclxin, a novel MIC60 inhibitor, induces apoptosis via mitochondrial stress in beta-catenin mutant tumor cells. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
14) | Matsumoto, T., Jiang, Y., Kuranaga, T., Lu, S., Wang, W., Onaka, H. Kakeya, H. Discovery of longicatenamides A-D produced by combined-culture of Streptomyces sp. KUSC_F05 and Tsukamurella pulmonis TP-B0596. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
13) | Kuranaga, T., Minote, M., Morimoto, R., Pan, C., Ogawa, H., Kakeya, H. Highly sensitive amino acid labeling reagents inspired by a scarce natural product yaku'amide B. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
12) | Minote, M., Kuranaga, T., Morimoto, R., Pan, C., Ogawa, H., Kakeya, H. Design, synthesis , and application of highly sensitive labeling reagents inspired by a scarce natural product. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
11) | Œ³ñC, Yulu Jiang, qij Shun Lu, Weicheng Wang, öGN, |JGº. úüÛRMJei~hA-DÉÖ·é€FÙ®÷¶šÌ¡|{Éæé¶YA\¢èA¶š«AyÑS¬. æ63ñVRL@»š¢_ï, åãinCubhj, 9, 2021.@@@@@ |
10) | Kura, Y., Velasco, M.D., Sakai, K., Fujita, Y., Hashimoto, M., Kakeya, H., Uemura, H., Nishio, K. Curcumin monoglucuronide modulates the tumor microenvironment of Pten-null prostate tumors and exhits antitumor activity The 80th Annunal Meeting of the Japan Cancer Asscociation. Sep. Yokohama, 2021. |
9) | Îì¶m, ¡ì@ãÄ, àcç°, éØT, °O@Œ, |JGº, cç³³O. ×EàÅÌñ{\[yv`h¬yfÌIðIP~JxO. æ15ñoCIÖA»wV|WE, 9, 2021.@@ |
8) | ²XØá, ŒºTê, ŒRWv, ªãczq, |JGº, gc@«. ªôyêÉš¯éZãÓ§ä@\Ì»wâ`wIðÍ. yêâ`wtH[æ54ñ€ñï, ŒÃ®, 9, 2021.@ |
7) | |JGº, qij, rcñd, ŒºTê, ä{³Æ. ÷¶šÔ»wR~ jP[VÌðE§äÆLp¶š«KhÌJ. VwpÌæ€u»wR~ jP[VÌteBAvEæ8ñöJV|WE. siICj 7, 2021. |
6) | ŒªñN, {çq, @Ÿ, |JGº, Rè@», åÎ^ç, åì_Í, äÑWã. MAIT×EÌ«»ðS€MR1KhÌTõ€. VwpÌæ€u»wR~ jP[VÌteBAvEæ8ñöJV|WE. siICj ,7, 2021.@@ |
5) | rcñd, ì©ü¢, ä{³Æ, |JGº. ªñ²×EðWIƵœRªñÜV[YÌTõ€. ú{P~JoCIW[wï@æ15ñNï. ªiICj, 6, 2021.@@ |
4) | X{ÁŸ, Œ³ñC, ¥èR¢, öò«s, Rc³ŸY, qij, |JGº. LC-MSðp¢œ«ðºÌDŽxA~m_ªÍ. nò§bï 2020 in s. siICj, 6, 2021. |
3) | ŒªñN, {çq, @Ÿ, |JGº, Rè@», åÎ^ç, åì_Í, äÑWã. MAIT×E«»Ü5-OP-RUÌ\¢«Ö€. ú{P~JoCIW[wï@æ15ïNïòwï. ªiICj, 6, 2021.@@ |
2) | rcñd, ì©ü¢, ä{³Æ, |JGº. ªñ²×EðWIƵœRªñÜV[YTõnÌ\z. ú{òwïæ141Nï. s, 3, 2021.@@ |
1) | ðäÞ, ŽLŸ, ÃJ@T, éØT, °O@Œ, ¬ÑŽ, @Ÿ, Žc@_, |JGº. s][iðL·éVKá_fU±öqHIF-1jQÜÌJ€. ú{òwïæ141Nï. L, 3, 2021.@@ |
16) | |JGº. ©RÉwÔ¶»w€Fªqv[uJÆnò. såwwÛZ³çiZ^[E¶»w€jbgæ10ñöJV|WE. s, 12, 2020. @@ |
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15) | |JGº, qij. nòEçòÖ̧íF©RÉwÔP~JoCIW[€. såwuŠé«á·vIC2020. s, 10, 2020. @@ |
14) | Pan, C., Kuranaga, T., Liu, C., Lu, S., Shinzato, N., Kakeya, H. Discovery of sulfur-containing cyclic lipopeptides thioamycolamides A-E, produced by the rare ctinomycete Amycolatopsis sp., The 62nd Symposium on the Chemistry of Natural Products, Nagoya, Sep. 2020.@@ |
13) | ¥èR¢, ¬ìÍé©, X{ÁŸ, àN ³ª, qij, |JGº. óVRšÌ\¢ð`[tƵœŽxx»ÜÌJ. ú{òwïæ140Nï. s, 3, 2020.iunCCgj @@ |
12) | cºü¿, ìYî, qij, |JGº. VRvhbO^RªñÜ[h»šTbJXIhBÌS¬€. ú{òwïæ140Nï. s, 3, 2020.@@@ |
11) | |@d, ŒºTê, àq«î, Shan Lu, |JGº. VRL@»šsaccharothriolide BÉ zðŸœvhbOZpÌJ€. ú{òwïæ140Nï. s, 3, 2020.@@@ |
10) | X{ÁŸ, qij, e{qK, |JGº. ÀpIinverseyv`h¬@ÌJ. ú{òwïæ140Nï. s, 3, 2020.@@ |
9) | ¡Ÿ, Ÿ, áX, ¬ìS÷, àN ³ª, |JGº. ErL`»yfUSP47ÆCateninD1̪ñ««»Éš¯é@\AÖ. ú{òwïæ140Nï. s, 3, 2020.@@ |
8) | |JGº. AJf~AnòðÚwµœnòP~JoCIW[€. TSMTP (Translational Science and Medicine Training Program) Symposium in Sapporo, Dy, 2, 2020. iµÒuj@@@@ |
7) | Kaneko, K., Nagao, N., Onaka, H., Shinzato, N., Kakeya, H. Detection of combined-culture specific constituents by the Molecular Networking and multivariate analyses. The 4th Kyoto Biomolecular Mass Spectrometry Society (KBMSS), Kyoto, Feb. 2020. |
6) | |JGº, Ý{[O, ~c-¬àVµ, ŽLŸ, gc¹», qij, ¡òú, Ž{³, àäëj. n«vhbO^ªqWIRªñÜCMGÌJ€. såwfBJCmx[ViMiPjìzåw@vOEãòn€ð¬T, s, 1, 2020.@@@ |
5) | qij, ¬ìÍé©, ¥èR¢, X{ÁŸ, àN³ª, |JGº. HCmVRšð@\`[tɵœŽxx»Ü. såwfBJCmx[ViMiPjìzåw@vOEãòn€ð¬T, s, 1, 2020.@@@@@@@ |
4) | Ÿ, àN³ª, ª[Ÿ, cŽ, ¡Ÿ, ¬ìS÷, |JGº. P~JoCIW[ðîÕƵœErL`»yfUSP47̶@\ðÍ. såwfBJCmx[ViMiPjìzåw@vOEãòn€ð¬T, s, 1, 2020.@@@@ |
3) | qij, Ÿ, |JGº. nòP~JoCIW[€. såwfBJCmx[ViMiPjìzåw@vOEãòn€ð¬T, s, 1, 2020.@@@@ |
2) | |JGº. Lp¶š«KhÌJðuüµœ»wR~ jP[V€. L@¬Ìj [gh2020iL@¬»wŠïÖŒxåÃj, åã, 2, 2020. iµÒuj@@@@ |
1) | Kakeya, H. Continuing Fascination with Discovery Science: Phenotypic Screening to Chemical Biology. Mona Symposium 2020: Natural Product Chemistry and Medicinal Chemistry. Kingston, Jamaica, Jan. 2020. (plenary lecture) |
32) | |JGº. ÷¶šÔ»wR~ jP[VÌðÆLp¶š«KhÌJ. VwpÌæ€u»wR~ jP[VÌteBAvEæ6ñöJV|WE. ¡l, 12, 2019. iµÒuj@@@ |
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31) | Kakeya, H. Chemical comunication research toward the development of useful chemical probes. The 4th A3 Roundtable Meeting on Asia Chemical Probe Research, Sendai, Nov. 2019. (Plenary lecture)@@@@ |
30) | Kakeya, H. Natural products-prompted chemical biology: Phenotypic screening and a new platform for target identification. The 6th Tishler-Omura Sympoium, Tokyo, Oct. 2019. (plenary lecture) [postponed due to the Typhoon no.19]@@@@ |
29) | Li, X., Hattori, A., Takahashi, S., Goto, Y., Harada, H., Kakeya, H. Inhibition of UCHL1 blocks proliferation and metastasis in HIF01 dependent tumor malignancy. 31th EORTC-NCI-AACR Symposium: International Conference on Molecular Targets and Cancer Therapeutics. Boston, MA, USA, Oct. 2019.@@@@ |
28) | Kakeya, H, Kishimoto, A., Umeta, H., Imaizumi, A., Kanai, M. Development of an injectable water-soluble anticancer drug CMG for oxaliplatin-resistant colorectal cancer with KRAS mutation. 31th EORTC-NCI-AACR Symposium: International Conference on Molecular Targets and Cancer Therapeutics. Boston, MA, USA, Oct. 2019.@ |
27) | Furutani, Y., Sudoh, M., Kakeya, H., Kojima, S. A small chemical compound CDM-3008 modulates cccDNA and suppresses HBV through induction of interferon-stimulated genes. 2019 International HBV Meeting. Melbourne, Australia, Oct. 2019.@@@@@ |
26) | Kuranaga, T., Kakeya, H. Highly sensitive labeling reagents inspired by a scarce marine natural product. 10th Korea-Japan Chemical Biology Symposium. Ishikawa, Oct. 2019.@@@@@ |
25) | Kanai, M., Kishimoto, A., Umeta, H., Imaizumi, A., Kakeya, H. Symposia 20 "Frontier in Molecular Target Therapy of Cancer": Development of a water-soluble prodrug CMG which inhibits proteasome activity through DYRK2 dependent manner. The 78th Annual Meeting of the Japanese Cancer Association, Kyoto, Sep. 2019. (invited)@@@@@ |
24) | Li, X., Hattori, A., Goto, Y., Harada, H., Kakeya, H. Involvment of UCHL1 in the HIF-1-dependent tumor cell malignancy in 3D cell culture model. The 78th Annual Meeting of the Japanese Cancer Association, Kyoto, Sep. 2019.@@@@@ |
23) | |JGº, qij. ©RÉwÔòÃè. såwAJf~bNfC2019, s, 9, 2019.@@@@ |
22) | ŽLŸ, Ñ@GŸ, Poznaks, V. |JGº. á_fU±öqHIF-1jQ«ðL·éÂófvVyv`hverucopeptinÌS¬. æ61ñVRL@»š¢_ï, L, 9, 2019.@@@@@ |
21) | Kakeya, H. Frontier research on chemical communications unveils the mystery of life science. The 27th International Society of Heterocyclic Chemistry Congress. Kyoto, Sep. 2019. (invited)@@@@ |
20) | cºü¿, ìYî, qij, |JGº. Rªñš¿TbJXIhBÌû©IS¬€. æ39ñL@¬Z~i[uŸúÌL@¬ðS€lÌœßÉv, åã, 8, 2019.@@@@@ |
19) | |JGº. ©RÉwÔTCGXuÀF »wR~ jP[VÌteBA€. såwI[vLpX. s, 8, 2019.@@@@ |
18) | ÃJ@T, Ëû^q, ^äxq, óûËq, ¬ÑJI, {¡³K, éØ¡a, |JGº, ¬ê. cccDNAð}§·éC^[tFláªq»šCDM-3008Ììp@\. æ29ñREBXÃ@wïwpWïEï, _Þì, 7, 2019.@@@@@ |
17) | àäëj, Ý{[O, ~c@µ, ¡ò@ú, |JGº. ILTv`ïR«ÌKRASå°ªñÉηéCMGËÜðp¢œVK¡Ã@ÌJ. æ17ñú{Õ°îáwïwpWï, s, 7, 2019.@@@@@ |
16) | |JGº. ÷¶šÔ»wR~ jP[VÌpÉæéVK¶š«KhÌJ€. æ19ñú{`¿ÈwïNïEæ71ñú{×E¶šwïåï ¯Nåï. ºÉ, 6, 2019.@iµÒuj@@@@@@ |
15) | |JGº, ŒºTê, qij, ì³T, ä{³Æ. ÷¶šÔ»wR~ jP[VÌðE§äÆLp¶š«KhÌJ. VwpÌæ€u»wR~ jP[VÌteBAvEæ5ñöJV|WE, åã, 6, 2019.@@@@@ |
14) | ãìãÄŸ, |JGº, ãu¬, äÑWã, âV¡@T, ²¡á, åŽN¶. [wwK@ÆPCAðÍðgÝí¹œP~JXy[XÌ». VwpÌæ€u»wR~ jP[VÌteBAvEæ5ñöJV|WE, åã, 6, 2019.@ |
13) | |JGº. uV|WEEªñÆhåÌ»wR~ jP[VÌðƧäv. n«vhbO^ªqWIRªñÜCMGÌJ€. æ23ñú{ªñªqWI¡ÃwïwpWï. åã, 6, 2019. iµÒuj@@@@@ |
12) | cºü¿, ìYî, qij, |JGº. Rªñ«ðL·é÷¶šãÓYšTbJXIhBÌS¬€. æ86ñú{ªÍ»wïL@÷ʪ̀§kïEæ110ñvª©®§äwïÍwÊvªï æ36ñ¯V|WE. s, 6, 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
11) | àq«î, ·öìfÔ, @Ÿ, |JGº. á_fU±öqiHIFjjQ»šverucopeptin̶¬â`qNX^[̯èÆVKÞÌÌTõ. æ86ñú{ªÍ»wïL@÷ʪ̀§kïEæ110ñvª©®§äwïÍwÊvªï æ36ñ¯V|WE. s, 6, 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
10) | |JGº. uV|WEE»wR~ jP[VÌteBAv. ÷¶šÔ»wR~ jP[VÌpÉæéVKLp¶š«KhÌJ€. æ19ñú{`¿ÈwïNïEæ71ñú{×E¶šwï ¯Nåï. ºÉ, 6, 2019. iµÒuj@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
9) | ÃJ@T, Ëû^q, ^äxq, óûËq, {¡³K, éØ¡a, |JGº, ¬ê. C^[tFlÌ«ðÂáªq»šCDM-3008ÌRHBV«ÌðÍ. æ26ñÌ×E€ï. ¡l, 5, 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
8) | |JGº. uV|WEEªñ÷¬Â«ÌðÆ»ÌÉü¯œòwIAv[`ÆÍHHIF-1¿ÌðƧäÉü¯Äv. á_fVOiðWIƵœnòP~JoCIW[. ú{òwïæ139Nï. çt, 3, 2019. iµÒuj@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
7) | |JGº. ·úe[}V|WEu¶œÈwÉš¯éªq»wÌv[Xv. »wR~ jP[VªDèÈ·¶œÈw. ú{»wïæ99tGNïi2019j. _Ë, 3, 2019. iµÒuj |
6) | ó rœ, öèŸY, ŒºTê, |JGº, öGN. ¡|{Éš¯éStreptomyces sp. HEK616Éæé5aTHQs̶Y@\, ú{_|»wï2019Nxåï. , 3, 2019. |
5) | Kakeya, H. Development of cryptic antifungal 5aTHQs targting cell membrane signaling. Asian Chemical Biology Initiative (ACBI) 2019 Yangon Meeting. Yangon, Myanmer, Jan. 2019. (invited)@@@@@@@@@@@@@@@@@@@@ |
4) | |JGº. uV|WEEVRšnò`ú{ÌÝ𶩵œVª¬`v@VRšnòÌ ðúµÄF÷¶šÔ»wR~ jP[VÌp. æ402ñCBIwïiîñvZ»w¶šwïjuï. , 1, 2019. iµÒuj@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
3) | Kakeya, H., Takahashi, N., Kishimoto, A., Imaizumi, A., Kanai, M. Development of an innovative water-soluble anticancer drug, curcumin mono-beta-D-glucuronide (CMG). The 1st International Symposium on Chemical Communication (ISCC2019). Tokyo, Jan. 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
2) | Nonaka, M., Fukuda, M.N., Kakeya, H. Rapid screening of antibody-binding peptides by combination of T7 phage display and next-generation sequencing technologies. The 1st International Symposium on Chemical Communication (ISCC2019). Tokyo, Jan. 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
1) | Jiang, Y., Lu, S., Hirai, G., Kato, T., Onaka, H., Kakeya, H. Towards the development of chemical communication molecules among microbes. The 1st International Symposium on Chemical Communication (ISCC2019). Tokyo, Jan. 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
33) | Kakeya, H., Kishimoto, A., Imaizumi, A., Kanai, M. Development of a synthetic water-soluble curcumin mono-beta-D-glucuronide (CMG), as an innovative anticancer prodrug targeting KRAS-NF-kappaB signaling pathway. 30th EORTC-NCI-AACR Symposium: International Conference on Molecular Targets and Cancer Therapeutics. Dublin, Ireland, Nov. 2018. |
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32) | Nonaka, M., Kakeya, H., Fukuda, M. Drug delivery to malignant brain tumor by a peptide specific to Annexin A1. 30th EORTC-NCI-AACR Symposium: International Conference on Molecular Targets and Cancer Therapeutics. Dublin, Ireland, Nov. 2018. |
31) | |JGº. ãòiV[hªqÌœl«noÆ×EàWITõE¯è. åebNtH[. , 10, 2018. iµÒuj |
30) | Jiang, Y. L., Lu, S., Hirai, G., Kato, T., Onaka, H., Kakeya, H. Enhancement of saccharothriolides production and discovery of new derivatives by combined culture of a rare actinomycete Saccharothrix sp. and Tsukamurella sp. The 22th Symposium on Development and Application of Naturally Occurring Drug Materials. Kumamoto, Oct. 2018. |
29) | ŒºTê, RŽî, JG, öèŸY, ó rœ, öGN, |JGº. ÷¶šÌ¡|{ÅŸçêé5aTHQÌea«Æ¶š«. æ60ñVRL@»š¢_ï. ª, 9, 2018. |
28) | âºD¡, ²¡º, ùìTî, ¬ŒTá, ìû³k, |JGº, ·cTV, Œ÷. A|g[VXU±«VRšcytotrienin A̬€. æ60ñVRL@»š¢_ï. ª, 9, 2018. |
27) | |JGº, ì³T, qij. VRšnòP~JoCIW[. såwAJf~bNfC2018, s, 9, 2018. |
26) | ŽçG, Shan Lu, Yulu Jiang, Å, ŒºTê, Ÿ, |JGº. æ91ñú{¶»wïåï. s, 9, 2018. |
25) | ŒŽñ^, Ÿ, |JGº. Calpain7Ì×EàÇÝÌðÍ. æ91ñú{¶»wïåï. s, 9, 2018. |
24) | ª[Ÿ, Ÿ, |JGº. yfœ¬x_IðÍðp¢œErL`»yfUSP47ÌC[ÌæÌ@\ðÍ. æ91ñú{¶»wïåï. s, 9, 2018. |
23) | |JGº. VRšnòP~JoCIW[`úüÛÉ£¹çêÄ`. 2018Nxiæ33ñjú{úüÛwïåï. , 9, 2018. iµÒuj |
22) | ¶cÀ¹, É¡€, ŒºTê, gc «, |JGº. œuÇ`¬â×EL·Éš¯éXtBS¿Ìdv«. yêâ`wtH[[æ51ñ€ñï. ª, 9, 2018. (|X^[ÜðóÜ) |
21) | |JGº. ©RÉwÔTCGXuÀF »wR~ jP[VªqÌäÉé. såwI[vLpX. s, 8, 2018. |
20) | |JGº. _òÌn»E€J®üƻܻZpZ~i[FVK_òÌJðuüµœP~JoCIW[€. V[GV[oÅZ~i[. , 7, 2018.iµÒuj |
19) | Jiang, Y.L., Lu, S., Hirai, G., Kato, T., Onaka, H., Kakeya, H. Enhancement of saccharothriolide (STLs) production by combined-culture of Saccharothrix sp. and Tsukamurella sp. The 29th Meeting on Discovery and Development of New Drugs. Shizuoka, Jul. 2018. |
18) | cºSç, Shan Lu, cŽ, |JGº. á_fU±öqiHIFsj«»š¿ÌP£E\¢èÆìp@ðÍ. æ29ñVòn¬kbï. ê, 7, 2018. |
17) | |JGº. VRšnòP~JoCIW[Ìçí¡. æ53ñVRš»wkbï. åã, 7, 2018.iµÒuj |
16) | ràPé, Cheng-Quin Pan, ¶cÀ¹, ŒºTê, |JGº. ¶ÌVOiÉìp·éVRšÌTõ€. æ53ñVRš»wkbï. åã, 7, 2018. |
15) | É¡k¢, qij, |JGº, e{qK. ZIl~hF̬€. æ53ñVRš»wkbï. åã, 7, 2018. |
14) | |JGº, ŒºTê, qij, ì³T, ä{³Æ. ÷¶šÔ»wR~ jP[VÌðÆLp¶š«KhÌJ. VwpÌæ€u»wR~ jP[VÌteBAvEæ3ñöJV|WE. , 6, 2018. |
13) | |JGº. u»wR~ jP[VÌteBAvðN_ɵœnòP~JoCIW[. VwpÌæ€u¿NIeBªð«Ÿ©·¶œ»Ûvæ4ñÌæïc. ºÉ, 6, 2018. iÁÊuj |
12) | ÃJ@T, |JGº, ¬ê. [NVbvuB^ÌVK¡ÃòÌTõÌ»óvFhbOt[ÌÀ»ðÚwµœcccDNA}§ÜCDM-3008ÆGeJrÆ̹pÉæéHBVÄ«»Ì}§. åã, 6, 2018. iÁÊuj |
11) | Lu, S., Nishimura, S., Ito, M., Kato, T., Kakeya, H. Discovery of pre-saccharothriolide X from the rare actinomycet Saccharothrix sp. The 13th Annual Meeting of Japanese Society for Chemical Biology, Tokyo, Jun. 2018. |
10) | Kakeya, H. Microbial metabolites targeting microenvironment: a cell membrane sigaling modulator and a hypoxia-response modulator. The 9th Japan-Korea chemical biology symposium, Incheon, Korea, May, 2018. (invited) |
9) | Ogawa, Y., Kakeya, H. Screening of sensitizers derived from microbial metabolites to induce apoptosis in pancreatic cancer cells. The 9th Japan-Korea chemical biology symposium, Incheon, Korea, May, 2018. |
8) | Nonaka, M., Kakeya, H., Fukuda, M. Identification of binding peptides against IgE from human myeloma U266 cells. The 9th Japan-Korea chemical biology symposium, Incheon, Korea, May, 2018. |
7) | Li, X.B., Goto, Y., Hattori, A., Harada, H., Kakeya, H. Study on the UCHL1-HIF-1 axis toward development of molecular targeted anticancer drugs. The 22th Annual Meeting of the Japanese Association for Molecular Target Therapy of Cancer (JAMTTC), Tokyo, May, 2018. |
6) | Kanai, M., Imaizumi, A., Kakeya, H. Development of a water-soluble curcumin monoglucronide (CMG) as a novel anticancer prodrug targeting KRAS-NF-kappa B signaling pathway. Global Academic Programs (GAP) conference, Stockholm, Sweden, May, 2018. (invited) |
5) | |JGº. u·úéæEP~JoCIW[€Á¬Ìœß̶š«ªqÌ©íªv\÷¶šÔ»wR~ jP[VÌäɧÞ\. ú{»wïæ98tGNï. çt, 3, 2018. iµÒuj |
4) | èr¶, {NŸ, Ÿ, ¬ê, |JGº. TGF-ÀVOi`BjQÜKUSC-Y244ÍTGF-ÀÉæéãçÔt]·ð}§·é. ú{òwïæ138Nï, àò, 3, 2018. |
3) | |JGº. uV|WEF±ê©çÌVRšTCGXv\P~JXy[Xg[íªF÷¶š¡|{@yÑPDSS (Precurso-Directed in situ Synthesis)@\, ú{_|»wï2018Nxåï. ŒÃ®, 3, 2018. iµÒuj |
2) | |JGº. ÷¶šÔ»wR~ jP[VÌpÉæéP~JXy[Xg[íª. VwpÌæ€u»wR~ jP[VÌteBAvEæ2ñöJV|WE. s, 2, 2018. iµÒuj |
1) | Lu, S., Nishimura, S., Ito, M., Kato, T., Kakeya, H. Expansion of chemical space in saccharothriolides: Precursor-directed in situ synthesis (PDSS) in a rare actinomycete Saccharothrix sp. Natural Product Discovery & Development in the Genomic Era (Natural Products 2018), Clearwater, FL, USA. Jan. 2018. |
26) | |JGº. n_òCmx[Vðn·éP~JoCIW[ûª. _òfUC€ïiåÃFú{_òwïE_òfUC€ïj. , 11, 2017. iµÒuj |
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25) | ¡ò ú, ŽLŸ, õàpé, àäëj, Ž{ ³, qìI¡, ÃcFÍ, |JGº. @\«HifÞÌãòiÖÌWJðÚwµœnòP~JoCIW[. æ7ñHiòwV|WE. s, 10, 2017. iµÒuj |
24) | ŽLŸ, Ñ GŸ, Poznaks, V., |JGº. ãò»wIWJðwüµœverucopeptinÌS¬€. æ35ñfBViP~Xg[V|WE. ŒÃ®, 10, 2017. |
23) | Furutani, Y., Toguchi, M., kakeya, H., Kojima, S. Combinatorial treatment of CDM/iCDM and entecavir for efficient suppression of cccDNA. 2017 International HBV Meeting: The Molecular Biology of Hepatitis B viruses, Washington, DC, USA. Sep. 2017. |
22) | ŒºTê, gº Ê, RŽî, |JGº. VRL@»šÌ\¢ðÍÆNMRVOiÌd¡. æ18ñNMR€ï. aÌR, 9, 2017. iµÒuj |
21) | ¶cÀ¹, É¡€, ŒºTê, |JGº. XtBS¿Ì@\ðŸðÚwµœ»wâ`wIðÍ.FGLm}CVÞÌæŸÆ»Ì\»^. yêâ`wtH[æ50ñ€ñï. , 9, 2017. |
20) | ŒºTê, ¿q«l, |JGº, ŒiÎ÷, å÷³q, ¶£`v, Carvalho, S., Cortes, J., Ribas, J. Xe[ðWIÉ·éR^Û»šZIl~hÉæé×EÇÙí. yêâ`wtH[æ50ñ€ñï. , 9, 2017. |
19) | ººsl, öèŸY, RŽî, ŒºTê, ó rœ, |JGº, öGN. ¡|{ÉæÁĶY³êéegqhLm»šÌðÍ. æ32ñú{úüÛwïåï, ·ì, 9, 2017. |
18) | |JGº. ©RÉwÔTCGXuÀF÷¶šÔ»wR~ jP[VÌäÉé. såwI[vLpX. s, 8, 2017. |
17) | àäëj, ¬àV µ, ¡ò ú, ŽLŸ, |JGº. [NVbvuAJf~ARªñòJÌiWvFvhbO^NN~ðp¢œVKRªñòÌJ. æ15ñú{Õ°îáwïwpWï. ºÉ, 7, 2017. |
16) | ¬ìÍé©, @áX, @Ÿ, ã¡eq, XéêÍã, œªáÁ°, Žc@_, |JGº. ªqWIRªñÜJðwüµœErL`»yfUCHL1jQÜÌTõ€. æ28ñVòn¬kbïuŸ³ÆnòÌCmx[Vv. ê, 7, 2017. |
15) | ¶cÀ¹, É¡€, ¡cqœ, ŒºTê, |JGº. ×E¿ðWIƷ黚ÌXN[jOyѻ̫]¿. æ28ñVòn¬kbïuŸ³ÆnòÌCmx[Vv. ê, 7, 2017.(DG\Üi§ãÜjðóÜ) |
14) | Lu, S., Nishimura, S., Ito, M., Kato, T., Kakeya, H. Novel natural products, saccharothriolides, from rare actinomycete Saccharothrix sp. and precursor-directed in situ synthesis (PDSS) of thier analogs. The 10th Anniversary Symposium of Division of Bioinformatics and Chemical Genomics, Graduate School of Pharmaceutical Sciences, Kyoto University, Kyoto, July, 2017. |
13) | àq«î, | d, ·öìfÔ, Îì¶m, gœìa÷, Ü\ëV, |JGº. P~JXy[Xg[ðwüµœ¶¬HwI€. såwåw@òw€Èãòn¬îñÈwêU10üNLOV|WE. s, 7, 2017. |
12) | ª[Ÿ, cŽ, Ÿ, |JGº. ErL`»yfUSP47Ì|rL`œÁ»@\ÌðŸÆjQÜTõnÌ\z. såwåw@òw€Èãòn¬îñÈwêU10üNLOV|WE. s, 7, 2017. |
11) | ŽLŸ, Ñ@GŸ, Viktors Poznacks, |JGº. á_fU±öqiHIFsjjQÜJðwüµœverucopeptinÌS¬€. såwåw@òw€Èãòn¬îñÈwêU10üNLOV|WE. s, 7, 2017. |
10) | |JGº. ÷¶š¡|{@ÌpÉæénòP~JoCIW[. æ12ñ»w¶Ôw€ï. Ù, 6, 2017. iµÒuj |
9) | ÃJ@T, |JGº, ¬ê. V|WEuB^Ì€ÌVWJvFcccDNA}§ÜCDM/iCDMÆGeJrÆ̹pøÊÌðÍ. æ53ñú{Ìwïï. L, 6, 2017. |
8) | Lu, S., Nishimura, S., Ito, M., Kato, T., Kakeya, H. Generation of saccharothriolide analogs by precursor-directed in situ synthesis (PDSS) and their SAR study. The 12th Annual Meeting of Japanese Society for Chemical Biology, Sapporo, June, 2017. |
7) | ŒºTê, É¡€, ŽLŸ, |JGº. T|jÆXe[̪qÔÝìpÉš¯éY» fœÊÆ _îÌdv«. ú{P~JoCIW[wï æ12ñNï, Dy, 6, 2017. |
6) | |JGº. ©RÉwÑAŽðRð«A·èðné. ú{wpU»ïiJSPSjuú{Éš¯éP~JoCIW[ÌVWJvÉÖ·éYwŠÍ€ÏõïiJSPSæ189ÏõïjEH29Nxæ1ñèáï, , 5, 2017.iµÒuj |
5) | Li, X.B., Takahashi, S., Hattori, A., Goto, Y., Morinobu, A., Hiraoka, M., Harada, H., Kakeya, H. Chemical biology research on the UCHL1-HIFs axis toward development of molecular targeted anticancer drugs. SKO Symposium 2017 (Joint Symposium 2017 of Seoull Univ., Kyoto Univ., and Osaka Univ.), Osaka, May, 2017. |
4) | @áX, Ÿ, ã¡eq, XéêÍã, , œªáÁ°, Žc@_, |JGº. åw@¶V|WEuòwªñ€ÌWÆ¢ðæ±·éáèªñ€Ò̧ívFUCHL1-HIF«»oHðWIƵœªqWIRªñÜJ€. ú{òwïæ137Nï. åä, 3, 2017. iµÒuj |
3) | Ñ@±œ, ŽLŸ, ìYî, Ëû^q, ²¡Tü, ÃJ@T, ¬ê, |JGº. VKB^Ì¡Ãòn»Éü¯œCDMsÌ\¢«Ö€. ú{òwïæ137Nï. åä, 3, 2017. |
2) | |JGº. uV|WEF_|»w©çM·é¢ã^VRš»wv\AJf~AnòÉš¯é\»^XN[jOÆ¢ãVRš»w\. ú{_|»wï2017Nxåï. s, 3, 2017. iµÒuj |
1) | |JGº. nòP~JoCIW[€ûªF\»^XN[jOÆV[hªqJ. rbOf[^ì®^nòVXe€_Eæ3ñV|WE. cä`måw. ¡l, 3, 2017. iµÒuj |
24) | @áX, ã¡eq, Ÿ, œªáÁ°, Žc@_, |JGº. VKªqWIRªñÜJðwüµœUCHL1-HIF«»oHjQÜXN[jOnÌ\z. æ75ñú{àwïwpï. ¡l, 10, 2016. |
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23) | ŒºTê, RŽî, JG, öèŸY, ó rœ, öGN, |JGº. ÷¶šÌ¡|{ÅŸçêé5aTHQÆstreptoaminalÌ\¢Æ\¢. æ21ñVRòšÌJÆpV|WE. çt, 10, 2016.iµÒuj |
22) | Kojima, S., Furutani, Y., Kakeya, H. Screening of novel cccDNA modulator compounds, iCDMs.The 2016 International HBV Meeting: The Molecular Biology of Hepatitis B Viruses. Seuol, Korea, Sep. 2016. |
21) | Îì¶m, ¡ì@ãÄ, }亟, éØT, °O@Œ, |JGº. ñ{\[«yv`h¬yfÌIðIx»ZpÌJÆv¬@\ðÍVXeÌ\z. æ58ñVRL@»š¢_ï. åä, 9, 2016. |
20) | Œ{×M, úäìa_, ¢iëO, |JGº, ÑYñY. XvCVOjQÜRQN-18690A (18-deoxyherboxidiene)ÌS¬. æ58ñVRL@»š¢_ï. åä, 9, 2016. |
19) | ª[Ÿ, ÂØ@L, @Ÿ, |JGº. ErL`»yfUSP47Ì|rL`œÁ»ÉÖíéªqàÌæ̯è. æ89ñú{¶»wïåï. åä, 9, 2016. |
18) | ãÉî, ¬ÑSq, @Ÿ, |JGº. ErL`»yfjQÉæéHIF-1»x̧ä. æ89ñú{¶»wïåï. åä, 9, 2016. |
17) | Îì¶mA}亟A¡ì@ãÄA|JGº. ñ{\[«yv`h¬yfÌÔ I@\ðÍZpÌJ. æ10ñoCIÖA»wV|WE. Îì, 9, 2016. |
16) | |JGº. uVµ¢R^ÛòV[hJÆKgåíªv\R^ÛòJÌœßÌP~JoCIW[€ûªFV[hªqJÆJjYðÍ. ZpîñŠïZ~i[. , 8, 2016.iµÒuj |
15) | Kakeya, H. Development of new anticancer drugs targeting TGF-À and HIF signaling pathway. 2016 BIO International Convention. San Francisco, CA, USA, Jun. 2016. |
14) | |JGº. nòP~JoCIW[F¶Ìà÷¬Â«VOi̧ä. VKfÞTõ€ïEæ15ñZ~i[. ¡l, 6, 2016. iµÒuj |
13) | JG, RŽî, ŒºTê, |JGº. ¶ÌÆÝìp·é5aTHQÞÌ\¢«Ö€Æuõv[uJ. ú{P~JoCIW[wï æ11ñNï. s, 6, 2016. |
12) | ¬ê, |JGº, ÃJ T, èp÷, ŒYam. ¢ã¶œîÕZpðp¢œB^̧³ÌœßÌnò€. æ26ñREBXÃ@wïï. €m, 5, 2016. |
11) | ¬ê, ÃJ T, |JGº. V|WEEB^Ì€ÌUp-To-DateFC^[tFl«ðÂáªq»šCDMÉæécccDNA}§ìpÌðÍ. æ52ñú{Ìwïï. çt, 5, 2016. |
10) | |JGº. TGF-ÀšæÑá_fVOiðWIƵœVKªñ¡ÃòÌJ€. æ15ñÛoCIeNmW[WŠïiBIOtech 2016j. , 5, 2016. |
9) | Kakeya, H. Microbial metabolites-prompted chemical biology: Phenotypic screening and a new platform for target identification. The Fifth Symposium of RIKEN-Max Planck Joint Research Center for System Chemical Biology. Berlin, Germany, Apr. 2016. iµÒuj |
8) | ŽLŸ, Ñ@GŸ, |JGº. á_fU±öqiHIFjjQ«ðL·éÂófvVyv`hverucopeptinÌS¬€. ú{òwïæ136Nï. ¡l, 3, 2016. |
7) | RŽî, ŒºTê, öèŸY, ó rœ, öGN, |JGº. åw@¶V|WEF¿«VRšÌp\úüÛ¡|{tæè©oµœVKAJChQÉÖ·é€. ú{òwïæ136Nï. ¡l, 3, 2016. iµÒuj |
6) | Cornelio, K., Matsumori, N., Murata, M., Nishimura, S., Kakeya, H., Yoshida, M., Matsunaga, S. Examination of apossible mechanism for the membrane translocation of the marine sponge-derived bioactive metabolite TNM-A. ú{»wï96tGNïi2016j, s, 3, 2016. |
5) | ººml, öèŸY, RŽî, ŒºTê, ó rœ, |JGº, öGN. ¡|{ÁÙIɶY³êéegqhLm¶¬â`qÌðÍ. ú{_|»wï2016Nxåï. Dy, 3, 2016. |
4) | Nishimura, S., Ito, A., Kakeya, H. Strict recognition of membrane lipids by a sea cucumber saponin, holotoxin B. Gordon Research Conference-Marine Natural Products-, Ventra, CA, USA, Mar., 2016. |
3) | gº@Ê, ŒºTê, å˹D, @Ÿ, |JGº. Eá_fU±öq(HIF)jQ«ðL·éverucopeptinÌ\¢ðÍÆìp@ðÍ, VwpÌæ€uVRšP~JoCIW[FªqWIÆ«§ävnæ~jV|WEisj, s, 2, 2016. |
2) | Kakeya, H. Academic drug discovery research: Phenotypic screening and target identification. University of Bordeaux-Kyoto University Mini-Symposium on Biomolecular Science. Kyoto, Jan. 2016. iµÒuj |
1) | Nishimura, S., Moriyama, A., Katagiri, N., Takahashi, N., Kakeya, H. In vivo linking of membrane lipids and membrane proteins using amphiphilic lipid probes. The 8th Takeda Science Foundation Symposium on PharmaSciences: Biomolecule-Based Medicinal Science: Featuring Mid-Size Drugs. Osaka, Jan. 2016. |
31) | Kakeya, H. Natural products-based academic drug discovery. International symposium on natural products chemistry and chemical biology 2015. Hawaii, USA, Dec., 2015. iµÒuj |
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30) | Kakeya, H. Natural products-prompted chemical biology; Phenotypic screening and target identification. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. iµÒuj |
29) | Lu, S., Nishimura, S., Hirai, G., Ito, M., Kawahara, T., Izumikawa, M., Sodeoka, M., Shin-ya, K., Tsuchida, T., Kakeya, H. Saccharothliolides A-C, novel phenyl-substituted 10-membered macrolides from a rare actinomycete Saccharothrix sp., identified by HPLC-MS profiling of microbial metabolites. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
28) | Takahashi, N., Hayashi, H., Kakeya, H. Synthetic study on the antitumor cyclodepcipeptide metabolite, verucopeptin. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
27) | Sugiyama, R., Nishimura, S., Ozaki, T., Asamizu, S., Onaka, H., Kakeya, H. 5-Alkyl-1,2,3,4-tetrahydroquinolines (5aTHQs), new membrane-interacting lipophilic metabolites, produced by combined-culture of Streptomyces nigrescens and Tsukamurella pulmonis. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
26) | Nishimura, S., Sugiyama, R., Fujita, K., Ito, S., Sakanishi, K., Iwabuchi, Y., Kanoh, N., Matsumori, N., Kakeya, H. Structure and function of heronamides, polyene macrolactams from marine-derived actinomycetes . The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
25) | Ishikawa, F., Miyamoto, K., Konno, S., Kasai, S., Kakeya, H. Accurate detection and manipulation of adenylation domain functions in nonribosomal peptide synthetases by an enzyme-linked immunosorbent assay system using active site-directed probes for adenylation domains. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
24) | Konno, S., Ishikawa, F., Suzuki, T., Dohmae, N., Kakeya, H. Profiling of nonribosomal peptide synthetase activities using active site-directed proteomic probes for adenylation domains. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
23) | Nishimura, S., Kakeya, H. Sterol-targeting antibiotics and the balance of membrane trafficking. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
22) | Yoshimura, A., Nishimura, S., Otsuka, S., Hattori, A., Kakeya, H. Studies on the microbial metabolite verucopeptin, an inhibitor of HIF-signaling pathway. SKO Symposium 2015 (Joint Symposium 2015 of Seuol Univ., Kyoto Univ., and Osaka Univ.), Seoul, Nov., 2015. |
21) | }亟, Îì¶m, |JGº. ñ{\[«yv`h¬yfÌ|óãCüðWIƵœ»wv[uÌJ. æ65ñú{òwïßExïEåï. 10, åã, 2015. |
20) | Îì¶m, ¡ìãÄ, }亟, éØT, °OŒ, |JGº. ¬¬ªq»šQÉæéAfj[VhCÌIðIW¯»šæÑvt@COÖÌWJ. æ9ñoCIÖA»wV|WE. 9, F{, 2015.iuÜðóÜj |
19) | Œ÷, ÉrÆ, DŸ, âŒqœ, âºD¡, ¡cqœ, RŽî, ŒºTê, |JGº. Heronamides A-C ÌS¬Æ\¢üùAšæÑ\¢«Ö. æ57ñVRL@»š¢_ï. ¡l, 9, 2015. |
18) | Lu, S., Nishimura, S., Hirai, G., Ito, M., Kawahara, T., Izumikawa, M., Sodeoka, M., Shin-ya, K., Tsuchida, T., Kakeya, H. Studies on Saccharothriolides A-C, Novel Phenyl-substituted 10-Membered Macrolidesfrom a Rare Actinomycete Saccharothrix sp. 57th Symposium on the chemistry of natural products. Yokohama, Sep. 2015. |
17) | lûcIã, ¡cqœ, ûPËG¢, ŒºTê, œª^°, Žc_, |JGº. IDH3¿\HIF-1oHð§ä·é¶š«š¿ÌTõ€. æ26ñVòn»kbï. ê, 9, 2015. (DG\Üi§ãÜjðóÜ) |
16) | |JGº. ¿ln¢^nòP~JoCIW[, æ7ñòwÌ¢ðlŠésV|WEuòEHEãAgÉæé¿ln¢^nò€ÌteBAv, s, 8, 2015. |
15) | |JGº. såwI[vLpXEòwEÍ[öÆ. nòEçòÖ̧íF©RÉwÔP~JoCIW[€. s, 8, 2015. |
14) | |JGº. V|WEunòÌ«v. nòP~JoCIW[FV[hªqJƪqvt@CO. æ63ñú{»wÃ@wïï. , 6, 2015. iµÒuj |
13) | ¡ìãÄ, Îì¶m, éØT, °O Œ, |JGº. Afj[VhCÉηé«Êwü^v[uðp¢œñ{\[«yv`h¬yf«Ìvt@CO. æ15ñú{`¿ÈwïNï, ¿, 6, 2015. |
12) | Nishimura, S., Sugiyama, R., Fujita, K., Kakeya, H. Abnormal cell wall deposition by heronamides, small molecules targeting phospholipids possessing saturated hydrocarbon chain. Pombe 2105 (8th International Fission Yeast Meeting), Kobe, Japan, June, 2015. |
11) | }亟, Îì¶m, |JGº. ñ{\[«yv`h¬yfÌSÌ^pN¿ðWIƵœáªqv[uÌJ. ú{P~JoCIW[wïEæ10ñNï, åä, 6, 2015. |
10) | ¡ìãÄ, Îì¶m, éØT, °OŒ, |JGº. Afj[VhCÉηé«Êwü^v[uðpµœñ{\[«yv`h¬yf«Ìvt@CO. ú{P~JoCIW[wïEæ10ñNï, åä, 6, 2015.[DG|X^[ÜðóÜ] |
9) | |JGº. ¶Ìà÷¬Â«VOiðWIƵœnòP~JoCIW[. nòòtH[Eæ58ñkbï. , 5, 2015. iµÒuj |
8) | |JGº. ·úe[}V|WEiú{»wïECujOZbVju¶¬}Vi[ÆVRšP~JoCIW[ÌZÉæéVWJv. æ±IVRšP~JoCIW[F\»^XN[jOÆWITõE¯è. ú{»wïæ95tGNï. çt, 3, 2015. iµÒuj |
7) | Kakeya, H. Technologies bridging metabolome and clock -Chemical biology for drug discovery; seed molecules development and target identification-. International Symposium on RNA and Clock: Epigenetic Landscape in Biological Rhythms. Hyogo, Mar. 2015. iµÒuj |
6) | ¡cqœ, RŽî, ŒºTê, |JGº. Heronamide AšæÑB̶¬@\ÉÖ·é€. ú{òwïæ135Nïi_Ëj. _Ë, 3, 2015. |
5) | ¡ìãÄAÎì¶mAéØTA°OŒA|JGº. Afj[VhCÉηé«Êwü^v[uÌJ. ú{òwïæ135Nïi_Ëj. _Ë, 3, 2015. [DG\ÜðóÜ] |
4) | }亟, Îì¶m, |JGº, ñ{\[«yv`h¬yfÌØv`WSÌ^pN¿ðWIƵœv[uÌJ€. ú{òwïæ135Nïi_Ëj. _Ë, 3, 2015. |
3) | Îì¶m, ¡ìãÄ, |JGº. «Êwü^v[uÍAfj[VhCðIðIÉW¯·é. æ17ñ¶œ»w€ï, m, 1, 2015. |
2) | Sugiyama, R., Nishimura, S., Ozaki, T., Onaka, H., Kakeya, H. 5-Alkyl-1,2,3,4-tetrahydroquinolines, membrane-interacting lipophilic metabolites, found in a unique combined culture of Streptomyces sp. and Tsukamurella pulmonis. Natural Products 2015; Natural product discovery & development in the post genomic era [Organized by Society for Industrial Microbiology and Biotechnology (SIMB)], San Diego, CA, USA, Jan. 2015. |
1) | Kakeya, H., Yoshimura, A., Sugiyama, R., Kishimoto, S., Nishimura, S., Hattori, A., Ishikawa, F., Yomoda, Y., Lu, S., Katagiri, N., Shimada, S., Seto, E., Hayashi, H., Takahashi, N., Harada, H. Chemical Biology for modulators targeting cancer microenvironment and cell membrane signaling. Natural Products 2015; Natural product discovery & development in the post genomic era [Organized by Society for Industrial Microbiology and Biotechnology (SIMB)] , San Diego, CA, USA, Jan. 2015. |
32) | |JGº. V|WEEmgÌVWJF nòV[YJðwüµœVRšP~JoCIW[ -\»^XN[jOÆWITõE¯è-. æ20ñVRòšÌJÆpV|WE. , 11, 2014.iµÒuj |
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31) | Îì¶m, ¡ìãÄ, |JGº. Afj[VhCÉηée[[ChP~JxO@ÌJ. æ20ñVRòšÌJÆpV|WE. , 11, 2014. |
30) | Nishimura, S., Sugiyama, R., Matsumori, N., Kakeya, H. Marine natural products targeting cell membrane. 3rd Annual Conference of the International Chemical Biology Society (ICBS2014), San Francisco, CA, USA, Nov. 2014. |
29) | Ý{^¡, ŒºTê, Ÿ, gœìa÷, Ü\ëV, |JGº. AVOAjW\¢ðL·éVKVftHAchlorocatechelinÞÌP£E\¢èAS¬AšæѶš«. æ56ñVRL@»š¢_ï. m, 10, 2014. |
28) | ¡ìãÄ, Îì¶m, |JGº. «Êwü^v[uðp¢œAfj[VhCÌIðIW¯». æ8ñoCIÖA»wV|WE. 9, ªR, 2014. |
27) | Îì ¶m, {{ á, ¡ì ãÄ, }ä ºŸ, |J Gº. i»ªqHwðwüµœAfj[VhCÉηéELISA@ÌJ. æ8ñoCIÖA»wV|WE. 9, ªR, 2014. |
26) | ¿q«l, ŒºTê, zqq, gc«, |JGº. AÉæé×EXe[b`hCÌÇݧä@\ÌðŸ. yêâ`wæ47ñ€ñï. , 9, 2014. |
25) | Kakeya, H. Chemical biology for drug discovery and target identification. IUPAC2014 & 248th ACS (American Chemical Society) National Meeting, San Francisco, CA, USA, Aug. 2014. (µÒu) |
24) | ÂØL, pÑÔ, ¬ÑSq, Ÿ, |JGº.@ErL`»yfUSP47Ì«»Éš¯éC[ÌæÌð. æ19ñú{aÔveA[[wïwpWï. åã, 8, 2014. |
23) | |JGº. såwI[vLpXEòwEÍ[öÆ. nòEçòɧÞP~JoCIW[. s, 8, 2014. |
22) | XR², ŒºTê, |JGº. ¶ÌðWIÆ·éVRšÌìp@ðÍðwüµœLiDEL@ÌJ. ú{P~JoCIW[wïEæ9ñNï. åã, 6, 2014.[DG|X^[ÜðóÜ] |
21) | öèŸY, RŽî, ŒºTê, ó rœ, |JGº, öGN. ¡|{ðpµœVKegqhLmÞÌP£Æ»Ì¶¬ÉÖ·é€. 2014Nxiæ29ñjú{úüÛwï. ïé, 6, 2014. |
20) | Konno, S., Ishikawa, S., Kakeya, H. Chemical labeling of adenylation domains in nonribosomal peptide synthetase. Gordon Research Conferences: Bioorganic Chemistry-Global Challenges in the 21st Century-. Andover, NH, USA, June, 2014. |
19) | Ishikawa, F., Konno, S., Kakeya, H Highly selective detection method for nonribosomal peptide synthetase using cocktails of active-site probes for adenylation domains. Gordon Research Conferences: Bioorganic Chemistry-Global Challenges in the 21st Century-. Andover, NH, USA, June, 2014. |
18) | |JGº. nòV[YJðwüµœVRšP~JoCIW[. VRšP~JoCIW[ -ªqWIÆ«§ä-Eæ6ñöJV|WE. €m, 5, 2014.iµÒuj |
17) | Ý{^¡, ŒºTê, Ÿ, gœìa÷, Ü\ëV, |JGº. VKVftHAchlorocatechelinÞÌP£E\¢èÆS\]¿. ¶ÈÈu»wÃ@îÕx®v æ3ñV|WEuAJf~A©çÌRªñÜnòÉü¯Äv. «ê, 5, 2014 |
16) | cŽ, gºÊ, ÀcM, ŽLŸ, ŒºTê, Ÿ, |JGº. ªñªqWInòðwüµœá_fU±öq(HIF)jQÜÌTõEJ€. ¶ÈÈu»wÃ@îÕx®v æ3ñV|WEuAJf~A©çÌRªñÜnòÉü¯Äv. «ê, 5, 2014. |
15) | |JGº. V|WEEVRšP~JoCIW[(2)FPEoCIP~Xg[F÷¶š@\ðpµœnòP~JoCIW[€. ú{òwï134Nï. F{, 3, 2014.iµÒuj |
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14) | Ý{^¡, ŒºTê, Ÿ, gœìa÷, Ü\ëV, |JGº. Streptomyces®úüÛæè©oµœfŽqÜLVKVftHAÌP£E\¢è. ú{òwï134Nï. F{, 3, 2014. [DG\ÜðóÜ], [Nï\nCCgÉÌð] |
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13) | RŽî, ŒºTê, öèŸY, öGN, |JGº. egqhLmiðL·éVKúüÛãÓšÌ\¢œl«Æ¶š«. ú{òwï134Nï. F{, 3, 2014. [DG\ÜðóÜ] |
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12) | gºÊ, ŒºTê, åËÑD, Ÿ, |JGº. á_fU±öq(HIF)«»oHðjQ·éverucopeptinÌìp@ðÍ. ú{òwï134Nï. F{, 3, 2014. |
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11) | ÀcM, êcLü, rìŸ, cŽ, Ÿ, ŒºTê, åÎ^ç, ¡äMF, |JGº. VKá_fU±öqHIFjQÜÌTõÆ\¢«Ö€. ú{òwï134Nï. F{, 3, 2014. |
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10) | ŽLŸ, |JGº. Rîá«ÂófvVyv`hverucopeptinÌS¬€. ú{òwï134Nï. F{, 3, 2014. |
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9) | ¡ìãÄ, Îì¶m, |JGº. õea«v[uðpµœAfj[VhCÉηéKh˶IW¯». ú{òwï134Nï. F{, 3, 2014 |
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8) | ëìŸF, ŒºTê, Á¡œ, |JGº. Chaetoglobosin DÍROSY¶Éæè×EÌZ»ðjQ·é. ú{òwï134Nï. F{, 3, 2014. |
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7) | ¬ÑSq, Ÿ, ÂØL, |JGº. EUrm1»«ÌošæѪq¯è. ú{òwï134Nï. F{, 3, 2014. |
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6) | ÂØ@L, p@ÑÔ, ¬Ñ@Sq, @Ÿ, |J@Gº. ErL`»yf(USP)47̪qàhCÌ@\ðÍ. ú{òwï134Nï. F{, 3, 2014. |
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5) | ªºMq, »ìzê, â×j, œìG, ÀØër, nç³Yê, yäC, ¡níL, Ži, Œäl, à_cFq, ¡òú, Ž{³, |JGº, ac[¹, ÃÍ, ·Jì_ñ, X{Bç. ³ì×tNXI[o[2dÓ±ÉæÁÄTheracurminÍŒÌNN~»ÜæèàDêœzûøŠÌüãªÝçêœ. ú{òwï134Nï. F{, 3, 2014. |
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4) | Sugiyama, R., Nishimura, S., Matsumori, N., Tsunematsu, Y., Hattori, A., Kakeya, H. Mode of action of heronamides, polyene macrolactams from a marine-derived Streptomyces sp. Gordon Research Conferences: Marine natural products- from discovery to human health-. Ventura, CA, USA, Mar. 2014. |
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3) | |JGº. nòEçòɧÞP~JoCIW[FòwÖÌUi¢ŽÈj¢. kq|NeXäy, s{§kwZ. 3, 2014.iµÒuj |
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2) | Yoshimura, A., Nishimura, S., Otsuka, S., Hattori, A. Kakeya, H. Mode of action of vercopeptin, an inhibitor of HIF-signaling pathway isolated from an actinomycete. The 12th International Student Seminar (12th ISS), Kyoto Univeristy. Kyoto, Feb. 2014. |
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1) | |JGº. œ¬25NxsòÈåwæ2ñnòÈwteBAV|WE. nòP~JoCIW[F\»^XN[jOÆWI¯è. s, 2, 2014.iµÒuj |
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21) | ëìŸF, ŒºTê, Á¡ œ, |JGº. ZãÓÍAN`jQÜÖÌŽó«ðãž³¹é. æ5ñHiòwV|WE. s, 11, 2013. |
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20) | ŒºTê, ¿q«l, zqq, gc«, |JGº. Xe[b`×EhCÌ`¬@\ÌðÍ. æ5ñHiòwV|WE. s, 11, 2013. [DG\ÜðóÜ] |
19) | {{á, Îì¶m, Ñ@L, |JGº. óÛNeosartorya®Rvjî]ÚyfÉÖ·é€. æ5ñHiòwV|WE. 11, s, 2013. |
18) | }亟, ðäCX, PŒYŸ, Ÿ, ŒºTê, |JGº. TGF-ÀVOijQ«ðL·éVRšgvgyv`AÌWIªqTõ€. æ5ñHiòwV|WE. s, 11, 2013.@[DG\ÜðóÜ] |
17) | Kakeya, H. Natural Products-Initiated Chemical Biology; Screening, Discovery, and Target Identification. 13th International Conference on the Chemistry and other bioactive compounds (ICCA-13), Yamanashi, Sep. 2013. (Invited Lecture) |
16) | RŽî, ŒºTê, ŒXMŸ, PŒYŸ, Ÿ, ºc¹Y, |JGº. CmRúüÛª¶Y·éheronamideÞÌP£Æ¶š«. æ55ñVRL@»š¢_ï. s, 9, 2013. |
15) | ¡ìãÄ, Îì¶m, |JGº. Afj[VhCðWIƵœõea«v[uÌJ. æ7ñoCIÖA»wV|WE. €m, 9, 2013. |
14) | {×N, Îì¶m, {{á, Icëj, ¡ìãÄ, |JGº. Andrimid̶¬yfÌ@\ðÍ. æ7ñoCIÖA»wV|WE. €m, 9, 2013. |
13) | Nishimura, S., Tokukura, M., Ochi, J., Yoshida, M., Kakeya, H. Sterol-rich membrane domains and the balance of membrane traffic. Pombe 2013 (7th International fission yeast meeting), June, London, UK, 2013. |
12) | {{á, Îì¶m, Ñ@L, |JGº. óÛNeosartorya sp. Rvjî]ÚyfÌ@\ðÍ. ú{P~JoCIW[wïEæ8ñNï. , 6, 2013. |
11) | Îì¶m, |JGº. AdenylationhCðWIƵœea«v[uÌJ. ú{P~JoCIW[wïEæ8ñNï. , 6, 2013. |
10) | Îì¶m, |JGº. LC-MS/MSðp¢œáªqv[uÉηéWI^pN¿Ì¯è. æ13ñú{`¿Èwï. ¹æ, 6, 2013. |
9) | É¡º, |JGº, gc«. ESUMO»yfSENP1jQÜÌTõ. æ17ñú{ªñªqWI¡ÃwïEwpWï. s, 6, 2013. |
8) | gº@Ê, ŒºTê, Ÿ, |JGº. á_fU±öq(HIF)«»oHðjQ·éúüÛRverucopeptinÌâΧÌzuÌè. æ17ñú{ªñªqWI¡ÃwïEwpWï. s, 6, 2013. |
7) | ëìŸF, ŒºTê, |JGº. A~m_ãÓðϲ·éVR»šÌTõ€. æ17ñú{ªñªqWI¡ÃwïEwpWï. s, 6, 2013. |
6) | {{á, Îì¶m, Ñ@L, |JGº. ªq@\Ï·ðwüµœ óÛNeosartorya sp. Rvjî]ÚyfÌ@\ðÍ. ú{òwïæ133Nï. _Þì, 3, 2013. |
5) | Îì¶m, |JGº. Lp¶¬yf̯èE@\ðÍðwüµœ»wc[ÌJ\AdenylationhCðWIƵœea«v[uÌJ\. ú{òwïæ133Nï. _Þì, 3, 2013. |
4) | RŽî, ŒºTê, PŒYŸ, Ÿ, |JGº. VK|G}NN^ÌP£E\¢èƻ̶š«. ú{òwïæ133Nï. _Þì, 3, 2013. |
3) | gº@Ê, ŒºTê, Ý{^¡, Ÿ, |JGº. 1,3-dimethylœó\¢Ì§Ìzuè@ÌØFtumescenamide CÆverucopeptinðáÉ. ú{òwïæ133Nï. _Þì, 3, 2013. |
2) | pÑÔ, Ÿ, ÂØL, ¬ÑSq, Xgpq, |JGº. ErL`»yf(USP)47Ì«»@\ÌðÍ. ú{òwïæ133Nï. _Þì, 3, 2013. |
1) | X{Bç, »ìzê, â×j, œìG, ÀØër, nç³Yê, yäC, éØŽü, RàÝä«, ¡níL, åËìF, à_cFq, ¡òú, ìSi, sjª, {M¥, |JGº, ac[¹, ·Jì_ñ. 4»Ü³ì×tNXI[o[2dÓ±ÉæèAZN~zù¿Ì¢zûøŠªÀسêœ. ú{òwïæ133Nï. _Þì, 3, 2013. |
20) | pÑÔ, Ÿ, ÂØL, ¬ÑSq, Xgpq, |JGº. ErL`»yf(USP)47Ì«»Éš¯éªqàrL`lhCÌð. æ85ñú{¶»wï. 12, ª, 2012. |
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19) | Ÿ, Œì¢q, pÑÔ, ¬ÑSq, Xgpq, |JGº. ErL`»yfUCH-L3Í_»XgXÌWI^pN¿Å é. æ85ñú{¶»wï. 12, ª, 2012. |
18) | |JGº. µÒuFVRš»wðîÕƵœnòP~JoCIW[. áè€ÒÌœßÌL@»wDyZ~i[. 11, kC¹, 2012. |
17) | ðäCX, ŒºTê, Ÿ, Ÿcñ€, yëv, ªºÏ, |JGº. 3À-Hydroxysteroid dehydrogenase (3À-HSD) jQÜÌJ€. æ30ñfBViP~Xg[V|WE. 11, , 2012. |
16) | Kanou, A., Nishimura, S., Kakeya, H. Chemical genetics for dissecting the crosstalk between cell metabolism and cell morphology. The 1st International Symposium on Chemical Biology of Natural Products: Target ID and Regulation of Bioactivity. Kyoto, Oct., 2012. |
15) | gºÊ, åËÑD, ŒºTê, Ÿ, |JGº. á_fU±öq(HIF)«»oHðjQ·éverucopeptinÉÖ·é€. æ19ñVRòšÌJÆpV|WE. 10, åã, 2012. |
14) | Jû¢}, ðäCX, ŒºTê, Ÿ, |JGº. GBF1jQ«ðL·égolgicide A Ì\¢«Ö€. æ62ñú{òwïßExïEåï, 10, ºÉ, 2012.[DG|X^[\ÜðóÜ] |
13) | gºÊ, åËÑD, ŒºTê, Ÿ, ·cTV, |JGº. á_fU±öq(HIF)«»oHðjQ·éverucopeptinÌ»wIðÍ€. æ54ñVRL@»š¢_ï. 10, , 2012. |
12) | ÓÅ, Ÿ, |JGº. á_fU±öq(HIF)jQÜTõÌœßÌnCRecEXN[jOnÌ\z. æ16ñú{ªñªqWI¡ÃwïEwpWï. ª, 6, 2012. |
11) | RŽî, ŒºTê, X[óq, öGN, |JGº. úüÛÌ¡|{ÉæÁÄŸçêéVKegqhLmU±ÌÉÖ·é€. ú{P~JoCIW[wï æ7ñNï. 6, s, 2012. |
10) | Ÿ, Œì¢q, pÑÔ, ¬ÑSq, Xgpq, |JGº. Activity-based ProfillingÉæé_»XgXŽó«ErL`»yf̯è. ú{P~JoCIW[wï æ7ñNï. 6, s, 2012. |
9) | Hu, X.-T., Hattori, A., Tokiwa, R., Kakeya, H. A high content screening system to develop novel HIF-1 inhibitors disrupting its heterodimeric formation. Organization for Oncology and Translational Research (OOTR) 8th Annual Meeting, Kyoto, Japan, Apr. 2012.[DG|X^[\ÜðóÜ] |
8) | Piao, J.-H., Tashiro, A., Nishikawa, M., Moriyoshi, E., Hattori, A., Kakeya, H. Enzymatic properties of recombinant human ubiquitin specific protease 47. Organization for Oncology and Translational Research (OOTR) 8th Annual Meeting, Kyoto, Japan, Apr. 2012. |
7) | }亟, ðäCX, PŒYŸ, Ÿ, åÎ^ç, ¡äMF, ŒºTê, |JGº. VKTGF-ÀVOi`BjQÜtryptopeptin AšæѪqv[u̬€. ú{òwïæ132Nï. Dy, 3, 2012. |
6) | RŽî, ŒºTê, X[óq, öGN, |JGº. úüÛª¶Y·éVKegqhLmU±ÌÌP£E\¢ðÍ. ú{òwïæ132Nï. Dy, 3, 2012. |
5) | ÓÅ, Ÿ, íÕç, |JGº. ñªquõâVXeðpµœá_fU±öq(HIF)jQÜ«]¿nÌ\z. ú{òwïæ132Nï. Dy, 3, 2012. |
4) | Œì¢q, ¬ÑSq, pÑÔ, Xgpq, Ÿ, |JGº. ErL`»yfUCH-L3Í_»XgXºÅs«»³êé. ú{òwïæ132Nï. Dy, 3, 2012. |
3) | pÑÔ, cãß, Œì¢q, Xgpq, Ÿ, |JGº. qgUSP47ÌErL`»yf«ÌðÍ. ú{òwïæ132Nï. Dy, 3, 2012 |
2) | ŒºTê, |JGº. V|WEuVRš»wÌVµ¢ª¬vF¶ÌððÍ·é»wâ`w. ú{òwïæ132Nï. Dy, 3, 2012. iµÒuj |
1) | |JGº. V|WEuHi@\wÆòwFÚ_Æá_©çwÔÌAv[`FhàÌÆèhEhàÌÃèhðîÕƵœP~JoCIW[€. ú{_|»wï2011Nxåï. s, 3, 2012. iµÒuj |
15) | |JGº. nòP~JoCIW[F©RÉwÔhòhÃè. ÈwEZptFX^ in s. s, 12, 2011. |
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14) | Morimoto, T., Wada, H., Sunagawa, Y., Fujita, M., Kakeya, H., Sasaki, H., Imaizumi, A., Hashimoto, T., Akao, M., Osakada, G., Kambara, H., Doi, O., Shiomi, H., Kimura, T., Shimatsu, A., Hasegawa, K., Effects of highly absorptive curcumin on systolic and diastolic function in hypertensive patients with left ventricular hypertrophy. Heart failure: Pharmacologic Therapy in Advanced Preclinical and Clinical Trials. American Association Scientific Sessions 2011. Orland, FL, USA, Nov. 2011. |
13) | Hattori, A., Tashiro, A., Piao, J.-H., Moriyoshi, E., Kakeya, H. Characterization of enzymatic properties of recombinant human specific protease 47. 7th General Meeting of the International Proteolysis Society. San Diedo, CA, USA, Oct. 2011. |
12) | Ý{^¡, PŒYŸ, ŒºTê, Ÿ, |JGº. úüÛªY¶·éVKÂó|fvVyv`hpentadepsin AÉÖ·é€. æ53ñVRL@»š¢_ï. åã. 9, 2011. |
11) | Espiritu, R.A., Matsumori, N., Murata, M., Nishimura, S., Kakeya, H., Matsunaga, S., Yoshida, M. Interaction of the marine sponge cyclic peptide theonellamide A with lipid bilayers investigated by membrane-permeabilizing activities and solid state 2H NMR. 14th Asian Chemical Congress 2011. Bangkok, Thailand, Sep. 2011. |
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9) | åìTi, Ÿ, ãc³¹, eRi, gMB°, |JGº. qgC7orf24Ìâ`q»ÍA]ÊJn_ßTÌ3ÌCCAATzñɧä³êé. æ84ñú{¶»wï. s, 9, 2011. |
8) | Ÿ, pÑÔ, cãß, Xgpq, |JGº. OUCBð|[^[Ép¢œErL`»yf«ªè@Ì\z. æ84ñú{¶»wï. s, 9, 2011. |
7) | i{C÷, Ÿ, |JGº, |{Ài, {Žœ, Ü ðÅÌA±œðpµœpH˶«VKDNAAL»ÜÌÝv. æ9ñ¢ãðS€L@»wV|WE. , 5, 2011. |
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4) | Ÿ, cãß, Xgpq, pÑÔ, |JGº. ErL`»yf«ÌVµ¢ªè@Ìm§. ú{òwïæ131Nï. ê, 3, 2011. |
3) | PŒYŸ, Ÿ, åÎ^ç, ¡äMF, ŒºTê, |JGº. úüÛ̶Y·éVKRªñÜ[h»štryptopeptinÌ»w\¢è. ú{òwïæ131Nï. ê, 3, 2011. |
2) | |JGº. ÁÊV|WEVRš»wÆP~JoCIW[uVK¶š«VRL@ªqÌJñÆP~JoCIW[€v. ú{òwïæ131Nï. ê, 3, 2011.iµÒuj |
1) | |JGº. á_fU±öq(HIF)Ì@\§äš¿ÌTõE]¿. ªñx®u»wÃ@îÕx®v-AJf~A©çÌRªñÜnòÖü¯Ä-. s, 3, 2011. |
12) | Tsunematsu, Y., Oishi, S., Fujii, N., Nishimura, S., Hattori, A., Kakeya, H. Tryptopeptin A, a novel TGF-beta signaling inhibitor from Streptomyces sp. International Chemical Congress of Pacific Basin Societies 2010 (PACIFICHEM 2010). Hawaii, USA, Dec., 2010. |
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11) | Nishimura, S., Matsunaga, S., Kakeya, H., Yoshida, M. Mode of action of theonellamides, antifungal bicyclic peptides from a marine sponge. International Chemical Congress of Pacific Basin Societies 2010 (PACIFICHEM 2010). Hawaii, USA, Dec., 2010. |
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9) | åìTi, Ÿ, ãc³¹, eRi, gMB°, |JGº. C7orf24/GGCTÌ]ÊÍNF-YÉæè«»³êé. æ83ñú{¶»wïåïEæ33ñú{ªq¶šwïNï¯åï: Biochemistry and Molecular Biology 2010 (BMB2010). 12, _Ë, 2010. |
8) | ŒºTê, zqq, LcSq, ŒRWv, ŒiÎ÷, gc«, |JGº. CYR^Ûš¿theonellamideÌìp@ðŸ. æ60ñú{òwïßExïEåï. 10, åã, 2010. |
7) | PŒYŸ, åÎ^ç, ¡äMF, ŒºTê, Ÿ, |JGº. úüÛª¶Y·éVKTGF-ÀVOi`BjQÜÌP£E\¢ðÍƬ. æTQñVRL@»š¢_ï. 9, ê, 2010. [§ãÜðóÜ] |
6) | Ñ@L, ºñN, åuN, ³œ, ·cTV, |JGº. VKÇV¶jQš¿Ì¶¬â`qQÌN[jO. 2010Nxiæ25ñjú{úüÛwïåï. 9, , 2010. |
5) | åγ«, {NŸ, šÐ³}, Ž jY, ·cTV, Ÿ, |JGº. VKá_fU±öq(HIF)jQÜÌn»€. æ1Sñú{ªñªqWI¡ÃwïEwpWï. 7, , 2010. |
4) | {NŸ, šÐ³}, Ÿ, |JGº. VKscaffoldðL·éTGF-ÀVOi`BÕfòÌn»€. æ1Sñú{ªñªqWI¡ÃwïEwpWï. 7, , 2010. |
3) | ŒºTê, zqq, LcSq, ŒRWv, ŒiÎ÷, gc«, |JGº. Xe[ðWIÆ·étheonellamideÌìp@ðÍ. ú{P~JoCIW[wï æ5ñNï. 5, _Þì, 2010. |
2) | Ohno, Y., Hattori, A., Ueda, M., Kageyama, S., Yoshiki, T., Kakeya, H. Involvement of NF-Y in transcriptional regulation if the human C7orf24/GGCT gene. Organisation for Oncology and Translational Research (OOTR) 6th Annual Conference. Kyoto, Japan, Feb., 2010. [DG|X^[\ÜðóÜ] |
1) | {NŸ, Ÿ, |JGº.@VKÌŸ³¡ÃòÌJ€FhHit to ProbehÌíªÆÀØ. uTGF-À«»œðWIƵœÌŸ³ÌVKff@, ¡ÃE\h@ÌJv€ÇV|WE. 2, åã, 2010. |
7) | Á¡Œ÷, ØC, |JGº, ·cTV. Aspergillus fumigatusÉš¯épseurotin¶¬â`qNX^[ÌðÍ. æ9ñ óÛªq¶šwRt@X. , 11, 2009. |
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6) | Nishimura, S., Matsuyama, A.., Yoshida, M., Matsunaga, S., Kakeya, H. Regulation of sterol localization revealed by chemical genetics using theonellamide. The 5th International Fission Meeting. Tokyo, Oct. 2009. |
5) | |JGº. V|WEuQmòwÆnòvFP~JoCIW[€ðîÕƵœAJf~AÉš¯énò€. æ68ñú{àwïwpï. ¡l, 10, 2009iµÒuj. |
4) | ŒºTê, ŒRWv, ŒiÎ÷, |JGº, gc«. Xe[ðWIÆ·étheonellamideÞªU±·éªôyêÌ`ÔÙí. yêâ`wtH[æ42ñ€ñï. }g, 7, 2009. |
3) | åìTi, Ÿ, |JGº. VKàÖAöqqgC7orf24Ì]ʧä@\ÌðÍ. æ13ñú{àªqWI¡Ãwï. ¿, 6, 2009. |
2) | Ÿ, PŒYŸ, åËÑD, {NŸ, ŒºTê, îqO, åÎ^ç, ¡äMF, Ž jY, ·cTV, |JGº. HIF-1@\§ä»šÌ]¿n\zÆTõ€. ú{òwïæ129Nï. s, 3, 2009. |
1) | Kakeya, H. Natural products-initiated chemical biology. Organic Chemistry Seminar in University of Louis Pasteur. Strasbourg, France, Apr. 2009 (Invited Lecture). |
5) | |JGº. ÷¶š¹ðîÕƵœP~JoCIW[€. æ17ñVRòšÌJÆpV|WE. V|WE1\u÷¶šöÝ\ÍÌÄF¯-nòÆîb€ÖÌpv. œ, 11, 2008.iµÒuj |
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4) | îqOA|JGºAÉ¡üçäA{œ`º. ŸÌC¬ª¶¬ÉÖ^·éey¬yfâ`qÌðÍ€. æ55ñú{¶òwïNï. ·è, 9, 2008. |
3) | ÑYñYA¯iAÎìElARûêYAcºFTA¡ä_MAŒJmãA«êA|JGºA·cTV. AT}CVnRîáVRšATCggGjAÌS¬. æ50ñVRL@»š¢_ï. œ, 9, 2008. |
2) | |JGº. "àÌÆè"ðîÕƵœP~JoCIW[€. æ128ñú{òwïV|WE VRšp[FwàÌÆèC¬C@\ðŸx`åwVRšòw€`. ¡l, 3, 2008.iµÒuj |
1) | |JGº. nòV[YJðwüµœVKVRL@»šÌJñEn»ÆP~JoCIW[€. \SEÇa¡ÃÌlbTX\Õ°SÇĶ€ï. s, 1, 2008.iµÒuj |
6) | |JGº. LpVRL@»šÌJñÆP~JoCIW[€. L@¬»wŠïuKïiœ¬19NxãúiHjj. , 11, 2007.iµÒuj |
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5) | _Rm, |JGº, PäY, NäGŸ, ·cTV. Epoxyquinol B inhibits the NF- B signaltransduction pathway through the TAK1 activity. æ66ñú{àwï. ¡l, 10, 2007. |
4) | ŒàV³F, RûêY, ¯i, |JGº, ¬ì£b, ·cTV. PanepophenatnrinÌsÄS¬yÑ»Ì\¢«Ö€. æ49ñVRL@»š¢_ï. Dy, 9, 2007. |
3) | Á¡Œ÷AØCAó©sOA|JGºA·cTV. Aspergillus fumigatus̶Y·é×EüújQÜgvX^`̶¬â`qNX^[̯è. æ2ñú{P~JoCIW[€ï. s, 5, 2007. |
2) | Kakeya, H., Kamiyama, H., Osada, H. Chemical biology of epoxyquinol B, an anti-angiogenic small molecule. RIKEN International Symposium on Chemcial Biology 2007 (RIKEN ISCB 2007). Kanagawa, Japan, Jan., 2007. |
1) | Hayashi, Y., Matsuzawa, M., Yamaguchi, J., Shoji, M., Kakeya, H., Onose, R., Osada, H. Total synthesis and structure activity relationship of (+)-panepophenanthrin, a ubiquitin-activating enzyme inhibitor. The Takeda Science Foundation Symposium on Pharma Sciences: On the Frontiers of Chemical Biology. Tokyo, Japan, Dec., 2007. |