| 6) | žcyl, qij, ühĺ÷, gcšť, żcVŹ, |JGş. VKŞń˛×EXtFCh`ŹjQÜXgvgXtFAĚSŹ. ú{ňwďć146Nďiĺăj, ĺă, 3, 2026.@@ |
|---|---|
| 5) | zKšl, qij, Çěž, ŕcŽ, |JGş. RŰÜcZi~hCĚŔHIŹoH̢¨ćŃ\˘ŤÖ¤. ú{ňwďć146Nďiĺăj, ĺă, 3, 2026.@@ |
| 4) | ŕ , n i, ´ł ˝, Îěa÷, F{ěĆ, |JGş, sŁ_u. ActVA-ORFlyfÉćéA[JbvO˝đîľ˝itgLmť¨ĚńĘť. ú{ňwďć146Nďiĺăj, ĺă, 3, 2026.@@ |
| 3) | źcäťç, rcńd, Ę J, |JGş. Şń˛×EXtFCh`ŹjQŤđLˇéPKS-NRPSnCubhVRť¨ĚŠĆěp@đÍ. ú{ňwďć146Nďiĺăj, ĺă, 3, 2026.@@ |
| 2) | Rc׏, AŁPv, şÔum, rcžÄ˘, ěŁM, Ň ¤, FiČO, qij, |JGş, öč ˝. ´xxťÜD-FDLDAđp˘˝ŔčŻĘĚWŻUąĚť@ÉćéAcnC}[ałŇ´ĚD/L-SerĆD/L-ProĚčĘŞÍ. ć17ńJBFV|WE, şÉ, 3, 2026. (*JBF: Japan Bioanalysis Forum) |
| 1) | Kakeya, H. (TBA). Asian Chemical Biology Initiative (ACBI) 2026 Chiang Mai Meeting, Chiang Mai, Thailand, Jan. 2026. (invited) |
| 47) | |JGş. VR¨nňP~JoCIW[ɨŻéhmgh¤ĚçíĄ. ú{P~JoCIW[wďEYwAgĎőď2025Nxć3ńčáĎőď, ĺă, 12, 2025.iľŇuj |
|---|---|
| 46) | Kakeya, H. On-gel combined-culture screening and discovery of new microbial metabolites of actinomycetes for drug discovery. PACIFICHEM 2025, Hawaii, USA, Dec. 2025. [Natural Products in the 'Omics Era' (#ORG018)] (invited) |
| 45) | Kakeya, H. Natural products-inspired chemical biology: Development of highly sensitive labeling reagents for amino acids, short peptide fragments, and scarce natural products. PACIFICHEM 2025, Hawaii, USA, Dec. 2025. [Recent Advances in Chemical Biology - in Memory of Koji Nakanishi, the Pioneer in Natural Product Chemistry on the Occasion of his 100 Year Birthday (#ORG024)] (invited) |
| 44) | Zhang, L., Pan, Y., Hattori, A., Uekusa, H., Suzuki, T., Dohmae, N., Hirano, Y., Kakeya, H. Discovery of lysine-reactive metabolites as covalent asparagine synthetase inhibitors from Stachybotrys sp. PACIFICHEM 2025, Hawaii, USA, Dec. 2025. [Bio-active Molecular Design Interwoven by AI Technology, Chemical Biology and Organic Synthesis (#ORG004)] |
| 43) | Mimura, A., Ikeda, H., Shibasaki, M., Suo, T., Hashimoto, J., Shin-ya, K., Imoto, M., Kakeya, H. Isolation, structural determination, and biological activity of novel cancer stem cell inhibiots streptospherins A-F. The 11th Japan-Korea Chemical Biology Symposium. Chungbuk, Korea, Dec. 2025. |
| 42) | Ikeda, H., Imoto, M., Kakeya, H. Establishment of a new screening strategy targeting cancer stem cells (CSCs) and development of the CSC inhibitors. The 11th Japan-Korea Chemical Biology Symposium. Chungbuk, Korea, Dec. 2025. |
| 41) | Yanagisawa, K., Kaneko, K., Ikeda, H., Iwata, S., Muranaka, A., Koshino, H., Nagao, N., Watari, S., Nishimura, S., Shinzato, N., Onaka, H., Kakeya, H. Discovery of actinoquinonal A and its congeners from the combined-culture of Streptomyces sp. and their production profile. The 11th Japan-Korea Chemical Biology Symposium. Chungbuk, Korea, Dec. 2025. |
| 40) | ŕcŽ, qij, 罞Y, |JGş. VKR^ŰÜAtBI[ĚűŠISŹ. ć42ńfBViP~Xg[V|WE, ż, 11, 2025. |
| 39) | źŞńN, ăěsĺ, čş, HtG÷, Ź`öş, ž, Ln@l, |JGş, Rč ť, Îŕ_ ×, ĺě_Í, äŃWă. ÂőŤőG}đp˘˝diaryltetrazoleÉćéśĚŞqĚxť˝ĚJ. ć42ńfBViP~Xg[V|WE, ż, 11, 2025. |
| 38) | öč ˝, Rc׏, AŁPv, rcžÄ˘, ěŁM, Ň ¤, FiČO, qij, |JGş. ´xUąĚťňD-FDLDAđp˘˝ADłŇ´ĚD/L-ZĆD/L-vĚčĘŞÍ. ú{A~m_wďć19ńwpĺď, ¤m, 11, 2025. |
| 37) | źŞńN, ăěsĺ, úąş, HtG÷, űöş, ž, Ln@l, |JGş, Rč ť, Îŕ_ ×, ĺě_Í, äŃWă. ÂőŤőG}đp˘˝eg][ĆJ{_ĚJbvO˝ÉćéśĚŞqĚxť. ć51ń˝ĆŹĚiŕV|WE, L, 11, 2025. |
| 36) | Matsui, M., Ikeda, H., Sakai, K., Nishio, K., Imoto, M., Kakeya, H. Discovery of an anticancer seed targeting cancer stem cells and analysis of its mode of action. 37th AACR-NCI-EORTC International Conference on Molecular Targets and Cancer Therapeutics, MA, USA, Oct. 2025. |
| 35) | Kakeya, H., Abe, T., Horisawa, Y., Kikuchi, O., Ozawa-Umezawa, H., Kishimoto, A., Katsuura, Y., Imaizumi, A., Hashimoto, T., Shirakawa, K., Takaori-Kondo, A., Yusa, K., Asakura, T., Kanai, M. Development of an innovative anticancer drug TBP1901, an injectable prodrug of curcumin, for the treatment of multiple myeloma. 37th AACR-NCI-EORTC International Conference on Molecular Targets and Cancer Therapeutics, MA, USA, Oct. 2025. |
| 34) | Rc׏, AŁPv, şÔum, rcžÄ˘, qij, |JGş, öč ˝. ´xLxťÜD-FDLDAđp˘˝yHiĆyůżĚD/L-A~m_ĚčĘŞÍ. ć19ń^{[V|WE, _Ë, 10, 2025. @ |
| 33) | öč˝, Rc׏, AŁPv, şÔum, rcžÄ˘, ěŁM, Ň ¤, FiČO, qij, |JGş. ´xLxťÜD-FDLDAđp˘˝ŻĘĚWŻUąĚť@Éćé´ĚD/L-ZĆD/L-vĚčĘŞÍ. ć19ń^{[V|WE, _Ë, 10, 2025. @ |
| 32) | żcVŹ,@qij, ´ úă, |JGş. Ëśę^A~hđîľ˝VKĹA~hť˝. ć75ńú{ňwďÖźxďEĺď, s, 10, 2025.@ |
| 31) | źcäťç, rcńd, Ę@J, |JGş. Şń˛×EXtFCh`ŹđjQˇéPKS-NRPSnCubhVRť¨ĚŠ. ć75ńú{ňwďÖźxďEĺď, s, 10, 2025.@ |
| 30) | rcńd, ÄčçO, Oş Ň, ühĺ÷, qij, ´{şq, VĆęj, ä{łĆ, |JGş. VKŞń˛×EtFA`ŹjQÜXgvgXtFŢĚJĆ\˘ŤÖ¤. ć75ńú{ňwďÖźxďEĺď, s, 10, 2025.@ |
| 29) | Furutani, Y., Yanaka, K., Kukimoto, M., Kobayashi, K., Nagamori, S., Shirouzu, M., Aizaki, H., Ochi, S., Kakeya, H., Matsuura, T. Development of an orally available JAK1 activator CDM-2020 that suppresses HBV through the induction of inteferon-stimulated genes. 2025 International HBV Meeting, Berlin, Germany, Sep. 2025. |
| 28) | ŕcŽ, qij, 罞Y, |JGş. VKR^ŰÜAtBI[Ě\˘ůł¨ćŃSʤ. ć67ńVRL@ť¨˘_ď, {é, 9, 2025. |
| 27) | Mimura, A., Ikeda, H., Shibasaki, M., Suo, T., Hashimoto, J., Shin-ya, K., Imoto, M., Kakeya, H. Isolation, structural determination, and biological activity of streptospherins A-F, new inhibitors targeting cancer stem cells. The 5th Research Network Salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2025. |
| 26) | ĂJ T, öD, A{rq, ŹŃJI, iXűu, üq, čp÷, zqŹ}, |JGş, źYma. áŞqJAKŤťÜCDM-2020ĚJ. ć33ńú{RECXĂ@wď, , 8, 2025. |
| 25) | Ą{ŘXq, rcńd, ŹŃ´, ä§ĺ, ü]ę_, ´c _, |JGş. ÷ś¨ăÓY¨RĚá_fUąöqW [^[ĚJ¤. ć35ńVňnťkbď, ĂŞ, 7, 2025. |
| 24) | Oş@Ň, rcńd, ÄčçO, ühĺ÷, ´{şq, VĆęj, ä{łĆ, |JGş. VKŞń˛×EXtFA`ŹjQÜXgvgXtFŢĚPُťA\˘đÍAyŃś¨Ť. ć35ńVňnťkbď, ĂŞ, 7, 2025. [¤§ăÜ]@@ |
| 23) | źäüRó, rcńd, âäaq, źöal, ä{łĆ, |JGş. Şń˛×EXtFA`ŹjQĚŠĆěp@đÍ. ć29ńú{ŞńŞqWIĄĂwď, Dy, 7, 2025.@ |
| 22) | qij, ŹR@¤, ´ úă, żcVŹ, |JGş. ńG}ITXeiuA~hť˝ĚJĆp. ć126ńL@ŹV|WE, s, 6, 2025.@ |
| 21) | öč˝, oFü, Rc׏, ÖűI, AŁPv, ěŁM, Ň ¤, qij, |JGş, FiČO, şÔum. PBrJĆ´xUąĚťňL-FDVDAđp˘˝VOldÉLC-MSÉćéH÷ĚC~_][Wyv`hĆÖAăÓ¨ĚčĘŞÍ. ć42ńú{÷Ęh{fwďwpWď, s, 6, 2025. @ |
| 20) | Keck, D., Yamada, Y., Hirose, T., Shimotsuma, M., Ikeda, A., Kawase, T., Tsuji, A., Tomonaga, S., Kuranaga, T., Kakeya, H., Ozaki, M., Quantitative analysis of D/L-Ser and D/L-Pro in serum using a highly sensitive chiral resolution labeling reagents D-FDLDA. HPLC 2025, Bruges, Belgium, Jun. 2025.@ |
| 19) | öč˝, Rc׏, AŁPv, şÔum, rcžÄ˘, ěŁM, Ň ¤, FiČO, qij, |JGş. ´xxťÜD-FDLDAđp˘˝AcnC}[ałŇ´ĚD-SerĆD-ProĚčĘ@Ěm§. ú{A~m_wďć8ńYwAgV|WE. , 6, 2025. @ |
| 18) | Zhang, L., Pan, Y., ž, AGT, éŘT, °O ź, ˝ěGT, |JGş. StachybotrysŽ^ŰR̤LŤAXpMŹyfjQÜĚTőĆJ¤. ú{P~JoCIW[wď@ć19ńNď, s, 6, 2025. |
| 17) | Ş{Ťu, Xcĺă, HtG÷, ž, Ln@l, |JGş, ĺě_Í, äŃWă. CD1aSŠŤT×Eđ§äˇéżKhĚTő¤. ú{P~JoCIW[wď@ć19ńNď, s, 6, 2025. |
| 16) | rcńd, Ą{ŘXq, ä§ĺ, ü]ę_, ´c _, |JGş. VR¨öÝóÔđpľ˝á_fUąöqW [^[ĚJ¤. öÝóÔŞqÝvEć3ńöJV|WE, Ąl, 5, 2025.@ |
| 15) | Ş{Ťu, Xcĺă, HtG÷, ž, Ln@l, |JGş, ĺě_Í, äŃWă. CD1aÉńŚłęéKhĚTőč@ĚJĆ\˘ŤÖ¤¤. öÝóÔŞqÝvEć3ńöJV|WE, Ąl, 5, 2025. |
| 14) | öč˝, oFü, Rc׏, ÖűI, AŁPv, ěŁM, Ň ¤, qij, |JGş, FiČO, şÔum. PBrJĆxťÜL-FDLDAđp˘˝Ž¨íĚŮČéH÷ĚC~_][Wyv`hĆÖAť¨ĚčĘŞÍ@Ěm§. ć79ńú{h{EHĆwďĺď, ¤m, 5, 2025. @ |
| 13) | Rc׏, öč ˝, AŁPv, rcžÄ˘, qij,@|JGş, şÔum. ´xUąĚťňD-FDLDAđp˘˝ŻĘĚWŻUąĚť@ÉćéśĚA~¨ćŃOěĚA~m_ĚčĘ. ć79ńú{h{EHĆwďĺď, ¤m, 5, 2025. @ |
| 12) | |JGş. ú{ňwďÜEóÜuFnňđuüľ˝VR¨P~JoCIW[¤. ú{ňwďć145NďiŞj, Ş, 3, 2025. ióÜuj@ |
| 11) | |JGş. V|WEumgTCGX@AbvgDfCgvFhmghđîŐĆľ˝VR¨nňP~JoCIW[. ú{ňwďć145NďiŞj, Ş, 3, 2025. iľŇuj@ |
| 10) | Oş@Ň, rcńd, ÄčçO, ühĺ÷, ´{şq, VĆęj, ä{łĆ, |JGş. VKŞń˛×EXtFA`ŹjQÜXgvgXtFAĚśYŤüăĆVKŢĚĚŠ. ú{ňwďć145NďiŞj, Ş, 3, 2025. |
| 9) | úĺŕVaó, ŕqŤî, rcńd, âcŔ, şúĆ, zěLá, ˇöěfÔ, n i, źşTę, V˘Žç, öGN, |JGş. úüŰĚĄ|{ÉćčYśłęéVKsmitgLmnť¨ĚPŁE\˘đÍĆťĚYśÉÖˇé¤. ú{ňwďć145NďiŞj, Ş, 3, 2025. [wśDG\ÜiűŞ\Ěj]@ |
| 8) | Zhang, L., Pan, Y., ž, AGT, ˝ěGT, |JGş. ^ŰStachybotrysŽŞśYˇéVK¤LŤAXpMŹyfjQÜĚJ¤. ú{ňwďć145NďiŞj, Ş, 3, 2025. |
| 7) | źäüRó, rcńd, ÄčçO, âäaq, źöal, ä{łĆ, |JGş. Şń˛×EXtFA`ŹjQŤđLˇéúüŰăÓY¨ĚŠĆěp@đÍ. ú{ňwďć145NďiŞj, Ş, 3, 2025. [wśDG\ÜiűŞ\Ěj]@@ |
| 6) | rcńd, ä§ĺ, Ą{ŘXq, ŹŃ´, ü]ę_, ´c _, |JGş. ŤžłĄĂɨŻéPKCż/mTORCVOiđîľ˝HIF-1żŤťíŞ. ú{ňwďć145NďiŞj, Ş, 3, 2025.@ |
| 5) | n i, ´{ ˝, Îěa÷, F{ěĆ, |JGş, sŁ_u. AN`mWśŹÉÖ^ˇéVK_ťyfActVA-ORF3ĚAlphaFoldđpľ˝@\đͤ. ú{ňwďć145NďiŞj, Ş, 3, 2025.@ |
| 4) | Ş{Ťj, Xcĺă, HtG÷, ž Ln@l, |JGş, ĺě_Í, äŃWă. żR´ńŚ^pNżCD1aÉFŻłęé|yv`hDDM-838Ě\˘ŤÖ¤. ú{ňwďć145NďiŞj, Ş, 3, 2025.@ |
| 3) | Kakeya, H. Natural product-inspired chemical biology: Development of an agrochemical seed targeting the scab-forming actinomycete. Asian Chemical Biology Initiative (ACBI) 2025 Hanoi Meeting, Hanoi, Vietnam, Jan. 2025. (invited) |
| 2) | Kakeya, H. Natural product-inspired chemical biology: Development of highly sensitive labeling reagents for amino acids, scarce natural products, and amylooid beta fragment peptides. The 5th Intenational Conference on Natural Product Discovery and Development in the Genomic Era. San Diego, CA, USA, Jan. 2025. |
| 1) | Yanagisawa, K., Kaneko, K., Ikeda, H., Iwata, S., Muranaka, A., Koshino, H., Nagao, N., Watari, S., Nishimura, S., Shinzato, N., Onaka, H., Kakeya, H. Discovery of a new pyranonaphthoquinone, actinoquinonal A: Combined-culture of Streptomyces sp. 23-50 with Tsukamurella pulmonis TP-B0596 triggers a shunt of the mevalonate pathway of Streptomyces sp. 23-50. The 5th Intenational Conference on Natural Product Discovery and Development in the Genomic Era. San Diego, CA, USA, Jan. 2025. [DG\Üi|X^[\)FThe Carol D. Litchfield Honorable Mention Student Poster Presentation] |
| 33) | öč˝, oFü, ÖűI, AŁPv, ěŁM, Ň ¤, qij, |JGş, FiČO, şÔum. PBrJĆxťÜL-FDLDAđp˘˝H÷ĚC~_][Wyv`hĆÖAť¨ĚčĘ. ć14ńVA~m_ŞÍ¤ď, , 12, 2024. @ |
|---|---|
| 32) | Rc׏, öč ˝, AŁPv, rcžÄ˘, qij,@|JGş, şÔum. ´xxťÜD-FDLDAđp˘˝r[ĚśĚA~ިćŃÖAť¨ĚęÄŞÍ. ć14ńVA~m_ŞÍ¤ď, , 12, 2024. @ |
| 31) | ühĺ÷, qij, gcšť, ŹR ¤, rcńd, ÄčçO, |JGş. VKŞń˛×EXtFA`ŹjQÜXgvgXtFAĚ\˘čyŃSʤ. ć41ńfBViP~Xg[V|WE, s, 11, 2024. |
| 30) | Ş{Ťu, Xcĺă, HtG÷, ž Ln@l, |JGş, ĺě_Í, äŃWă. CD1aSŠŤT×Eđ§äˇéjŰR|yv`hDDM-838Ě\˘ŤÖ¤. ć41ńfBViP~Xg[V|WE, s, 11, 2024. |
| 29) | Zhang, L., Pan, Y., Hattori, A., Uekusa, H., Kakeya, H.Discovery of new meroterpenoids produced by Stachybotrys ruwenzoriensis RF-6853 as asparagine synthetase inhibitors. Seoul Univ.-Kyoto Univ.-Osaka Univ. Symposium 2024 (SKO Symposium 2024). Seoul, Korea, Nov., 2024. |
| 28) | Rc׏, öč˝, şÔum, rcžÄ˘, qij, |JGş, AŁPv. ´xxťÜD-FDLDAđp˘˝r[Ě sA~ިćŃÖAť¨ĚęÄŞÍ. ć120ńú{Hiqśwďwpuď, ¤m, 11, 2024. |
| 27) | öč˝, oFü, ÖűI, şÔum, ěŁM, Ň ¤, qij, |JGş, FiČO,@AŁPv. xťÜL-FDVDAĆPBrJđp˘˝Ž¨íEgDEiíĚŮČéH÷ĚC~_][Wyv`hĆ\ŹA~m_A^EĚčĘŞÍ. ć120ńú{Hiqśwďwpuď, ¤m, 11, 2024. |
| 26) | öč˝, oFü, rcžÄ˘, qij, |JGş, AŁPv. ´xőwŞxťÜL-FDLDAđp˘˝yHiEůżĚDL-A~m_ĚčĘŞÍ@ĚJ. ć120ńú{Hiqśwďwpuď, ¤m, 11, 2024. |
| 25) | Kakeya, H., Pan, Y., Zhang, L., Suzuki, T., Sakai, K., Hirano, Y., Ikeda, H., Hattori, A., Dohmae, N., Nishio, K. Identification and a mode of action of bisabosqual A, a novel asparaginase synthetase (ASNS) inhibitor, towards the development of molecular-targeted anticancer drug. 36th EORTC-NCI-AACR Symposium on Molecular Targets and Cancer Therapeutics. Barcelona, Spain, Oct. 2024. (EORTC, the European Organization for Research and Treatment of Cancer; NCI, the National Cancer Institute; AACR, the American Association for Cancer Research) |
| 24) | úĺŕVaó, ŕqŤî, rcńd, âcŔ, şúĆ, zěLá, ˇöěfÔ, n i, źşTę, V˘Žç, öGN, |JGş. úüŰĚĄ|{Ć^{[đÍÉćéVKRŞńÜV[YĚJ¤. ć74ńú{ňwďÖźxďEĺď, şÉ, 10, 2024.[DGÜiűŞ\Ěj]@@ |
| 23) | rcńd, ěŠü˘, ÄčçO, Oş Ň, |JGş. Şń˛×EđWIơé÷ś¨ńăÓY¨ĚŠĆěp@đÍ. ć74ńú{ňwďÖźxďEĺď, şÉ, 10, 2024.@ |
| 22) | ŹR ¤, qij, X{Áž, źłńC, |JGş. Ëśę^A~hđîľ˝yv`hŹ@ĚJĆŞqÂóyv`hŹÖĚp. ć74ńú{ňwďÖźxďEĺď, şÉ, 10, 2024. [DGÜiűŞ\Ěj]@ |
| 21) | Ikeda, H., Iseki, S., Kobayashi, S., Irie, K., Harada, H., Kakeya, H. Upregulation of HIF-1ż via the PKCż/mTORC signaling pathway is a potential therapeutic strategy for ishemia-related diseases. The 4th network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2024. |
| 20) | Furutani, Y., Tanaka, K., Nagamori, S., Kobayashi, K., Aizaki, H., Ochi, S., Kakeya, H., Matsuura, T. Development of cccDNA modulators, CDMs, that specifically activate interferon-related signals and inhibit HBV replication. 2024 International HBV Meeting: Biology of the Hepatitis B and Viruses. Chicago, IL, USA, Sep. 2024@ |
| 19) | öč˝, oFü, ÖűI, şÔum, ěŁM, Ň ¤, qij, |JGş, FiČO,@AŁPv. xťÜL-FDVDAĆPBrJđp˘˝Ž¨íEgDEiíĚŮČéH÷ĚC~_][Wyv`hĆ\ŹA~m_A^EĚęÄŞÍ. ú{A~m_wďć18ńwpĺďiJSAAS2024j, éĘ, 9, 2024. |
| 18) | żcVŹ, rcńd, qij, ĽčR˘, ŕNłŞ, Jű§, V˘Žç, öGN, |JGş. VKAmCLXUąÜALZ^~hAĚPŁE\˘đÍyŃSŹ. ć66ńVRL@ť¨˘_ď, s, 9, 2024. |
| 17) | ŕqŤî, O}{Ô, Yulu Jiang, ´Lž, |JGş. A¨aQť¤Ša´öŰđWIơé_ňV[YJ¤FcZi~hCĚŠĆěp@đÍ. ć66ńVRL@ť¨˘_ď, s, 9, 2024. |
| 16) | Kakeya, H. Natural product-inspired chemical biology: Development of highly sensitive labeling reagents for amino acids and scarce natural products. International Congress on Natural Products Research 2024 (ICNPR 2024), Krakow, Poland, Jul. 2024.@@ |
| 15) | úĺŕVaó, ŕqŤî, rcńd, âcŔ, şúĆ, zěLá, ˇöěfÔ, n i, źşTę, V˘Žç, öGN, |JGş. úüŰĚĄ|{ÉćéVKRŞńÜV[YĚJ¤. ć34ńVňnťkbď, ČŘ, 7, 2024. [¤§ăÜ]@@@ |
| 14) | rcńd, ä{łĆ, |JGş. Şń˛×EđWIơém}CVĚŻčEěp@. ć28ńú{ŞńŞqWIĄĂwď, , 6, 2024.@@ |
| 13) | Furutani, Y., Kakeya, H., Matsuura, T. Development of novel small molecules that activate innate immunity and inhibit HBV replication. The 60th Annual Meeting of the Japan Society of Hepatology, Kumamoto, Jun, 2024. |
| 12) | ŕqŤî, O}{Ô, Yulu Jiang, ´Lž, |JGş. úüŰăÓY¨cZi~hCĚRť¤Ša´öŰŤĆťĚĎŤťŞŕ˝çˇj[NČ\ť^É¢Ä. ú{P~JoCIW[wď@ć18ńNď, , 5, 2024. |
| 11) | Kakeya, H. Separation and identification of the D/L-forms of amino acids and short-chain peptides using highly sensitive labeling reagents for research of cardiovascular disease. The 9th Annual Scientific Meeting of JCVA (Japan Cardiovascular Association), Shizuoka, May 2024. |
| 10) | öč ˝, oFü, şÔum, ěŁM, Ň@¤, qij, |JGş, FiČO, AŁPv. ´xxťÜL-FDVDAĆPBrJđp˘˝HiĚC~_][Wyv`hĆ\ŹA~m_A^EĚęÄŞÍ. ć78ńú{h{EHĆwďĺď, Ş, 5, 2024. |
| 9) | Ý{[O, ŹŠRI, ac[š, ó´Nq, RAę, öčT, ÂRL÷, YŰG, Ąňú, ´{ł, ťězę, X{Bç, ŕäëj, |JGş, ˇJě_ń. łÇóEyÇĚV^RiECX´őÇłŇɨŻéoűzűNN~iNN[W jĚÇÖĚiW}§řĘđءévZ{ÎĆńdÓłěםärą. ú{ňwďć144NďiĄlj, Ąl, 3, 2024.@@ |
| 8) | ühĺ÷, qij, gcšť, rcńd, ÄčçO, |JGş. VKŞń˛×EXtFA`ŹjQÜXgvgXtFAĚSʤ. ú{ňwďć144NďiĄlj, Ąl, 3, 2024. |
| 7) | żcVŹ, qij, ĽčR˘, rcńd, ŕNłŞ, |JGş. VKAmCLXUąÜALZ^~hAĚŽS\˘čyŃSʤ. ú{ňwďć144NďiĄlj, Ąl, 3, 2024. |
| 6) | ŕcŽ, qij, 罞Y, |JGş. VKR^ŰÜAtBI[ĚSʤ. ú{ňwďć144NďiĄlj, Ąl, 3, 2024. |
| 5) | rcńd, ÄčçO, ŞcĘG, DRŔă, ühĺ÷, gcšť, qij, VĄęq, ~řęv, ä{łĆ, |JGş. VKŞń˛×EXtFA`ŹjQÜXgvgXtFAĚPŁE\˘đÍ. ú{ňwďć144NďiĄlj, Ąl, 3, 2024. |
| 4) | |JGş. VR¨nňP~JoCIW[đîŐĆľ˝ŞqWIRŞńÜJ¤. ŞńĄĂCmx[VÉüŻÄ. sĺw¤@E¨żE×E_@ĘqimăäZ^[, s, 3, 2024.iľŇuj |
| 3) | Kakeya, H. Natural products-inspired chemical biology-Development of a novel asparagine synthetase inhibitor for cancer chemotherapy-, Asian Chemical Biology Initiative (ACBI) 2024 Istanbul Meeting, Istanbul, Turkey, Mar. 2024. iinvitedj@@ |
| 2) | Matsuoka, T., Hattori, A., Oishi, S., Araki, M., Ma, B., Fujii, T., Arichi, N., Okuno, Y., Kakeya, H., Yamasaki, S., Ohno, H., Inuki, S. Establishment of an MR1-presentation reporter screening system to identify MAIT cell modulation. CD1-MR1 2024, Tasmania, Australia, Feb., 2024. |
| 1) | öč ˝, şÔum, qij, |JGş, AŁPv, . ´xőwŞxťÜL-FDVDAđp˘˝śĚżEHiŠçĚA~m_Ě´xŞÍ@Ěm§. ć15ńJapan@Bioanalysis Forum (JBF) V|WE, s, 3, 2024. |
| 37) | Kakeya, H. Natural products-inspired chemical biology-Development of highly sensitive labeling reagents-, Asian Chemical Biology Initiative (ACBI) 2023 Kuala Lumpur Meeting, Kuala Lumpur, Malaysia, Dec. 2023. iinvitedj |
|---|---|
| 36) | |JGş, VR¨nňP~JoCIW[FVKA~m_Eyv`hŞÍ@ĚJĆp. ć13ńVA~m_ŞÍ¤ď, , 12, 2023. iľŇuj@@ |
| 35) | AŁPv, öč ˝, oFü, şÔum, rcžÄ˘, qij, |JGş. ´xőwŞxťÜD-FDLDAđp˘˝yHiĚDL-A~m_ŞÍ. ć13ńVA~m_ŞÍ¤ď, , 12, 2023. |
| 34) | öč ˝, şÔum, qij, |JGş, AŁPv. ´xőwŞxťÜL-FDVDAđp˘˝A~m_Ě\˘ŮŤĚĆőwŮŤĚĚęÄŞÍ. ęÄŞÍ@Ěm§. ć13ńVA~m_ŞÍ¤ď, , 12, 2023. |
| 33) | Sun, Y., Hashizume, D., Kakeya, H. Synthetic study of 2-(1H-imidazole-4-yl)-1,3,4-oxadiazole scaffolds for pharmaceuticals. The 40th Medicinal Chemistry Symposium. Nagoya, Nov., 2023. |
| 32) | Koyama, A., Kuranaga, T., Morimoto, R., Matsumoto, T., Kakeya, H. Acyl sulfonamide-mediated amidation and its application to the synthesis of middle molecular natural peptidic molecules. The 60th Japanese Peptide Symposium, Shiga, Nov. 2023. |
| 31) | Kuranaga, T., Morimoto, R., Pan, C., Ogawa, H., Kakeya, H. Design, synthesis, and application of highly sensitive labeling reagent for amino acids. The 60th Japanese Peptide Symposium, Shiga, Nov. 2023. |
| 30) | Ozaki, M., Shimotsuma, M., Kuranaga, T., Kakeya, H., Hirose, T. Identification of DL-amino acids containing threonine and isoleucine stereoisomers in peptides using an original chiral resolution labeling reagent. The 60th Japanese Peptide Symposium, Shiga, Nov. 2023. |
| 29) | |JGş. VR¨P~JoCIW[đîŐĆľ˝năňČw¤. ć9ńňw̢đlŚésV|WEFnăňČwęUJwLOV|WE, s, 11, 2023. iľŇuj |
| 28) | Pan, Y., Suzuki, T., Sakai, K., Hirano, Y., Ikeda, H., Hattori, A., Dohmae, N., Nishio, K., Kakeya, H. Identification of an asparagine synthetase inhibitor bisabosqual A as an anticancer seed. The 3rd network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
| 27) | Kodama, K., Ikeda, H., Shibasaki, M., Kawami, M., Imoto, M., Kakeya, H. Screening and identification of anticancer lead compounds through a novel strategy targeting cancer stem cells. The 3rd network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
| 26) | Kakeya, H., Ozaki, M., Shimotsuma, M., Kuranaga, T., Hirose, T. Development of a new chiral resolution labeling reagent and aplication to separation of amyloid b fragment peptides with racemized and isomerized aspartic acid residues. The 3rd network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
| 25) | Koyama A., Kuranaga, T., Morimoto, R., Matsumoto, T., Kakeya, H. A novel peptide C-terminal modification and its application to the synthesis of middle molecular cyclic peptides. The 3rd network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
| 24) | Sun, Y., Hashizume, D., Kakeya, H. Studies on 2-(1H-imidazol-4-yl)-1,3,4-oxadiazole scaffolds for pharmacological molecules. The 3rd network salon, Medical Innovation Program, Kyoto University, Kyoto, Sep. 2023. |
| 23) | AŁPv, öč ˝, oFü, şÔum, qij, |JGş. ´xőwŞxťÜD-FDLDAđp˘˝HiĚDL-A~m_ŞÍ. ú{A~m_wďć17ńwpĺď (JSAA2023), Ş, 9, 2023. |
| 22) | öč ˝, şÔum, qij, |JGş, AŁPv, . ´xőwŞxťÜL-FDVDAđp˘˝SA~m_ęÄŞÍ@Ěm§. ú{A~m_wďć17ńwpĺď (JSAA2023), Ş, 9, 2023. |
| 21) | oFü, öč ˝, şÔum, qij, |JGş, AŁPv. őwŞxťÜL-FDVDAđp˘˝yv`hĚThrĆIlȩĚŮŤĚĚŻč. ú{A~m_wďć17ńwpĺď (JSAA2023), Ş, 9, 2023. |
| 20) | ŹR ¤, qij, X{Áž, źłńC, |JGş. Gsťđ}§ˇéyv`hC[Cü@ĆŞqÂóyv`hŹÖĚp. ć65ńVRL@ť¨˘_ď, , 9, 2023.@@@@@.@@ |
| 19) | Ę J, rcńd, ÄčçO, ěŠü˘, ä{łĆ, |JGş. Şń˛×EđWIĆľ˝RŞńÜV[YĚJ¤. ć33ńVňnťkbď. s, 9, 2023. [¤§ăÜ]@@ |
| 18) | ŹR ¤, qij, X{Áž, źłńC, |JGş. Şqyv`hnňđuüľ˝VKyv`hŹ@ĚJ. ć33ńVňnťkbď, s, 9, 2023.@@@@@.@@ |
| 17) | źŞńN, ž, ĺÎ^ç, rŘ]k, Ln@l, |JGş, Rč ť, ĺě_Í, äŃWă. ×E\ĘĚMR1śÝĘÉîĂKhXN[jO@ĚJĆMAIT×E§äŞqĚŻč. ć65ńVRL@ť¨˘_ď, , 9, 2023.@@@@@.@@ |
| 16) | Yanaka, K., Hirano, Y., Qiun, X.Y., Suzuki, H., Kakeya, H., Matsuura, T., Furutani, Y. A small chemical compound iCDM-34 identified by an in silico screening suppresses HBV DNA through activation of aryl hydrocarbon receptor, 2023 Interbational HBV Meeting, Kobe, Sep. 2023.@@@.@@ |
| 15) | |JGş. P~JoCIW[đ@˛Ćľ˝Şqvt@CO, 2023NxáčxZpuKď, śČwČwpĎv¤ wp¤xîŐ`Ź ć[fލxvbgtH[iADAMsj, źĂŽ, 9, 2023. iľŇuj |
| 14) | |JGş. VR¨nňP~JoCIW[ĚĹOüFYwAgÉćéăňiĚŔpťÉüŻÄ, sCmx[Vp[NđŹZ~i[iĺĂFsT[`p[Nj, ĺă, 7, 2023. iľŇuj |
| 13) | |JGş. V|WE1EuWIđ˲ŻIiáŞqEŞqERĚjv\VR¨nňFAXpMŹyfđ˲. ć27ńú{ŞńŞqWIĄĂwďwpWď, ˛ę, 6, 2023. iľŇuj |
| 12) | Pan, Y., Suzuki, T., Sakai, K., Hirano, Y., Ikeda, H., Hattori, A., Dohmae, N., Nishio, K., Kakeya, H. Identification of bisabosqual A as an asparagine synthetase (ASNS) inhibitor towards the development of molecular-targeted anticancer drug. The 17th Annual Meeting of Japanese Society for Chemical Biology, Osaka, May, 2023. |
| 11) | Kakeya, H. Development of an innovative anticancer drug TBP1901, an injectable prodrug of curcumin. 2023 NSFC*1-JSPS-CAS*2 Forum: Translational Medicine and Innovative Drug Research. Tianjin, China, Jun. 2023. (*1 Natural Science Foundation of China, *2 Chinese Academy of Science) [keynote lecture] |
| 10) | źŞńN, ž, ĺÎ^ç, Ln@l, |JGş, Rč ť, ĺě_Í, äŃWă. MR1Ě×E\ĘĘđwWơéKhXN[jO@ĚJĆMAIT×EW [^[ĚŻč. ú{P~JoCIW[wď@ć17ńNď, ĺă, 5, 2023.@@ |
| 9) | Pan, Y., Suzuki, T., Sakai, K., Hirano, Y., Ikeda, H., Hattori, A., Dohmae, N., Nishio, K., Kakeya, H. Screening and identification of an asparagine synthetase (ASNS) inhibitor as a molecular-targeted anticancer drug. The 143rd Annual Meeting of Pharmaceutical Society of Japan. Hokkaido, Mar. 2023.@@@@@ |
| 8) | öč ˝, şÔum, qij, |JGş, AŁPv. DL-A~m_xťLbgđp˘˝A~ChŔĚAspcîĚZ~ťEŮŤťĚo@ĚJ\žłÉÖ^ˇéĂW^pNżEyv`hĚúffEžłJjYĚđžÉüŻÄ\. ć14ńJapan@Bioanalysis Forum (JBF) V|WE, , 3, 2023. |
| 7) | Ikeda, H., Shibasaki, M., Kodama, K., Kawami, M., Imoto, M., Kakeya, H. Screening for anticancer lead compounds through a new strategy for targeting cancer stem cells. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
| 6) | Sun, Y., Hashizume, D., Kakeya, H. Synthetic study on 2-(1H-imidazol-4-yl)-1,3,4-oxadiazole scaffolds for drug discovery. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
| 5) | Kuranaga, T., Tamura, M., Ikeda, H., Terada, S., Nakagawa, Y., Kakeya, H. Reactivity-guided identification and total synthesis of an unstable anticancer macrolide presaccharothriolide Z. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
| 4) | Kakeya, H., Abe, T., Horisawam Y., Kikuchi, O., Ozawa-Umeta, H., Kishimoto, A., Imaizumi, A., Hashimoto, T., Shirakawa, K., Takaori-Kondo, A., Yusa, K., Asakura, T., Kanai, M. Pharmacologic characterization of TBP1901, an innovative prodrug form of curcumin, and CRISPR-Cas9 screen for therapeutic targets of curcumin. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
| 3) | Koyama, A., Kuranaga, T., Morimoto, R., Kakeya, H. Acyl sulfamide-mediated amidation for biomimetic peptide synthesis. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
| 2) | Pan, Y., Suzuki, T., Sakai, K., Hirano, Y., Ikeda, H., Hattori, A., Dohmae, N., Nishio, K., Kakeya, H. Chemical biology research on an asparagine synthetase (ASNS) inhibitor as a molecular-targeted anticancer drug. Future Drug Discovery Empowered by Chemical Biology, Nara, Feb. 2023. |
| 1) | Ŕc ő, |ŕVłž, qij, |JGş. VKUąĚťňđp˘˝D,L-A~m_Ě´xŞÍ@J. ć28ńLC&MSeNmvU, ICJĂ, 1, 2023. [xXgv[e[VÜixXge[}Üj] |
| 15) | öč ˝, şÔum, qij, |JGş, AŁPv. őwŞxťÜD-FDLDAđp˘˝A~ChŔĚAXpM_cîĚZ~ťEŮŤťĚŻč. VA~m_ŞÍ¤ďć12ńwpuď, , 12, 2022. [DG\Ü] |
|---|---|
| 14) | Ŕc ő, |ŕVłž, qij, |JGş. VKUąĚťňđp˘˝śĚżyŃ×E|{ă´D,L-A~m_Ě´xŞÍ. VA~m_ŞÍ¤ďć12ńwpuď, , 12, 2022. |
| 13) | Yasuda, Y., Takezawa, M., Kuranaga, T., Kakeya, H. Highly sensitiveanalysis of D-and L-amino acids in biological samples using new derivatization reagents. The 37th Annual Meeting of the Japanese Society for the study of Xenobiotics, Kanagawa, Nov. 2022.@ |
| 12) | źŞńN, ž, ĺÎ^ç, Ln@l, |JGş, Rč ť, ĺě_Í, äŃWă. XvbgVtF[[đpľ˝XN[jO@ÉćéVKMR1KhĚŻčĆťĚ\˘ŤÖ¤. ć39ńfBViP~Xg[V|WE, 11, 2022, ICJĂ.@@@@@ |
| 11) | Ozaki, M., Shimotsuma, M., Kuranaga, T., Kakeya, H., Hirose, T. Identification of DL-and DL-iso-form of aspartic acid residues in amyloid b peptide using a chiral resolution labeling reagent. The 59th Japanese Peptide Symposium, Miyagi, Oct. 2022. |
| 10) | Ikeda, H., Imoto, M., Kakeya, H. Identification of the polyether ionophore lenoremycin through a new screening strategy targeting cancer stem cells. The 81st Annual Meeting of the Japanese Cancer Association. Kanagawa, Sep. 2022. [selected as a late-breaking poster]@@@@@ |
| 9) | Kura, Y., Develasco, M.A., Sakai, K., Fujita K., Bannno, E., Fujita, Y., Hashimoto, M., Nishimoto, M., Nozawa, M., Yoshimura, K., Kakeya, H., Umemura, H., Nishio, K. Chemopreventive potential of curcumin monoglucuronide in mouse Pten-null prostate cancer. The 81st Annual Meeting of the Japanese Cancer Association. Yokohama, Sep. 2022.@@@@@ |
| 8) | qij, cşüż, rcńd, c V, ěYî, |JGş. ťwŹđěgľ˝óRŞńŤVR¨vTbJXIhZĚŻč. ć64ńVRL@ť¨˘_ď, ĂŞ, 9, 2022.@@@@@ |
| 7) | |JGş, qij, rcńd, ž, źşTę, ä{łĆ. ÷ś¨ÔťwR~ jP[VĚđĆLpś¨ŤKhĚJ. VwpĚć¤uťwR~ jP[VĚteBAvćčÜĆßV|WE, s, 7, 2022. |
| 6) | |JGş. VR¨nňP~JoCIW[ĚĹOü. k˘ĺwć100ńKMCFZ~i[iKitasato Microbial Chemistry Frontierj, , 6, 2022. iľŇuj |
| 5) | Îěśm, ŕcç°, ĺźŢ, ĄěăÄ, éŘT, P, °Oź, |JGş, cçłłO. ×EŕĹĚń{\[yv`hŹyfĚIđIxť¨ćŃŞđ@\ĚŠ. ú{P~JoCIW[wď@ć16ńNď, xR, 5, 2022.@@ |
| 4) | ˛XŘá, źşTę, źRWv, Şăczq, |JGş, gcŤ. FKBP12ÉćéZEXIjăÓ§äĚťwâ`wIđÍ. ú{_|ťwď2022Nxĺď, siICj, 3, 2022. |
| 3) | Îěśm, ĄěăÄ, ŕcç°, éŘT, P, °Oź, |JGş, cçłłO. ×EŕĹĚń{\[yv`hŹyfĚIđIP~JxO¨ćŃŞđßöĚŠ. ú{ňwďć142Nď. źĂŽiICj, 3, 2022.@@ |
| 2) | Watari, S., Kaneko, K., Iwata, S., Nagao, N., Onaka, H., Shinzato, N., Kakeya, H. Syetematic screening of new microbial metabolites by combined-culture of actinomycetes. Japan-the Netherlands Microbiology Symposium 2022, Mar. 2022 (Kochi/on-line).@@@@@ |
| 1) | Kakeya, H. Chemical communication research on microbes toward the development of novel antibiotics. Japan-the Netherlands Microbiology Symposium 2022, Mar. 2022 (Kochi/on-line). (Invited lecture)@@@@@ |
| 18) | Kakeya, H. Chemical communication research toward the development of novel antibiotics. (#182 Antibiotics Discovery), PACIFICHEM2021, Hawaii, USA, Dec. 2021. (Invited lecture)@@@@ |
|---|---|
| 17) | Kakeya, H. Chemical communication research toward the development of new anticancer drugs. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
| 16) | Omura, S., Khadka, S., Sato, F., Nakamura, Y., Nishio, K., Kakeya, H., Tsunoda, I. Curcumin mooglucuronide (CMG) treatment alters the gut microbiota, regulating an autoimmune model for multiple sclerosis. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
| 15) | Ikeda, H., Muroi, M., Kondoh, Y., Ishikawa, S., Kakeya, H., Osada, H., Imoto, M. Miclxin, a novel MIC60 inhibitor, induces apoptosis via mitochondrial stress in beta-catenin mutant tumor cells. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
| 14) | Matsumoto, T., Jiang, Y., Kuranaga, T., Lu, S., Wang, W., Onaka, H. Kakeya, H. Discovery of longicatenamides A-D produced by combined-culture of Streptomyces sp. KUSC_F05 and Tsukamurella pulmonis TP-B0596. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
| 13) | Kuranaga, T., Minote, M., Morimoto, R., Pan, C., Ogawa, H., Kakeya, H. Highly sensitive amino acid labeling reagents inspired by a scarce natural product yaku'amide B. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
| 12) | Minote, M., Kuranaga, T., Morimoto, R., Pan, C., Ogawa, H., Kakeya, H. Design, synthesis , and application of highly sensitive labeling reagents inspired by a scarce natural product. (#79 Chemical Communications through Natural and Synthetic Bioactive Compounds), PACIFICHEM2021, Hawaii, USA, Dec. 2021.@@ |
| 11) | źłńC, Yulu Jiang, qij Shun Lu, Weicheng Wang, öGN, |JGş. úüŰRMJei~hA-DÉÖˇé¤FŮŽ÷ś¨ĚĄ|{ÉćéśYA\˘čAś¨ŤAyŃSŹ. ć63ńVRL@ť¨˘_ď, ĺăinCubhj, 9, 2021.@@@@@ |
| 10) | Kura, Y., Velasco, M.D., Sakai, K., Fujita, Y., Hashimoto, M., Kakeya, H., Uemura, H., Nishio, K. Curcumin monoglucuronide modulates the tumor microenvironment of Pten-null prostate tumors and exhits antitumor activity The 80th Annunal Meeting of the Japan Cancer Asscociation. Sep. Yokohama, 2021. |
| 9) | Îěśm, Ąě@ăÄ, ŕcç°, éŘT, °O@ź, |JGş, cçłłO. ×EŕĹĚń{\[yv`hŹyfĚIđIP~JxO. ć15ńoCIÖAťwV|WE, 9, 2021.@@ |
| 8) | ˛XŘá, źşTę, źRWv, Şăczq, |JGş, gc@Ť. ŞôyęɨŻéZăÓ§ä@\Ěťwâ`wIđÍ. yęâ`wtH[ć54ń¤ńď, źĂŽ, 9, 2021.@ |
| 7) | |JGş, qij, rcńd, źşTę, ä{łĆ. ÷ś¨ÔťwR~ jP[VĚđE§äĆLpś¨ŤKhĚJ. VwpĚć¤uťwR~ jP[VĚteBAvEć8ńöJV|WE. siICj 7, 2021. |
| 6) | źŞńN, {çq, @ž, |JGş, Rč@ť, ĺÎ^ç, ĺě_Í, äŃWă. MAIT×EĚŤťđS¤MR1KhĚTő¤. VwpĚć¤uťwR~ jP[VĚteBAvEć8ńöJV|WE. siICj ,7, 2021.@@ |
| 5) | rcńd, ěŠü˘, ä{łĆ, |JGş. Şń˛×EđWIĆľ˝RŞńÜV[YĚTő¤. ú{P~JoCIW[wď@ć15ńNď. ŞiICj, 6, 2021.@@ |
| 4) | X{Áž, źłńC, ĽčR˘, öňŤs, RcłžY, qij, |JGş. LC-MSđp˘˝ŤđşĚD´xA~m_ŞÍ. nň§bď 2020 in s. siICj, 6, 2021. |
| 3) | źŞńN, {çq, @ž, |JGş, Rč@ť, ĺÎ^ç, ĺě_Í, äŃWă. MAIT×EŤťÜ5-OP-RUĚ\˘ŤÖ¤. ú{P~JoCIW[wď@ć15ďNďňwď. ŞiICj, 6, 2021.@@ |
| 2) | rcńd, ěŠü˘, ä{łĆ, |JGş. Şń˛×EđWIĆľ˝RŞńÜV[YTőnĚ\z. ú{ňwďć141Nď. s, 3, 2021.@@ |
| 1) | đäŢ, ´Lž, ĂJ@T, éŘT, °O@ź, ŹŃ´, @ž, ´c@_, |JGş. s][iđLˇéVKá_fUąöqHIF-1jQÜĚJ¤. ú{ňwďć141Nď. L, 3, 2021.@@ |
| 16) | |JGş. ŠRÉwÔśťw¤FŞqv[uJĆnň. sĺwwŰZłçiZ^[Eśťw¤jbgć10ńöJV|WE. s, 12, 2020. @@ |
|---|---|
| 15) | |JGş, qij. nňEçňÖ̧íFŠRÉwÔP~JoCIW[¤. sĺwuŚéŤáˇvIC2020. s, 10, 2020. @@ |
| 14) | Pan, C., Kuranaga, T., Liu, C., Lu, S., Shinzato, N., Kakeya, H. Discovery of sulfur-containing cyclic lipopeptides thioamycolamides A-E, produced by the rare ctinomycete Amycolatopsis sp., The 62nd Symposium on the Chemistry of Natural Products, Nagoya, Sep. 2020.@@ |
| 13) | ĽčR˘, ŹěÍéŠ, X{Áž, ŕN łŞ, qij, |JGş. óVR¨Ě\˘đ`[tĆľ˝´xxťÜĚJ. ú{ňwďć140Nď. s, 3, 2020.iunCCgj @@ |
| 12) | cşüż, ěYî, qij, |JGş. VRvhbO^RŞńÜ[hť¨TbJXIhBĚSʤ. ú{ňwďć140Nď. s, 3, 2020.@@@ |
| 11) | |@d, źşTę, ŕqŤî, Shan Lu, |JGş. VRL@ť¨saccharothriolide BÉ zđž˝vhbOZpĚJ¤. ú{ňwďć140Nď. s, 3, 2020.@@@ |
| 10) | X{Áž, qij, e{qK, |JGş. ŔpIinverseyv`hŹ@ĚJ. ú{ňwďć140Nď. s, 3, 2020.@@ |
| 9) | Ąž, ž, áX, ŹěS÷, ŕN łŞ, |JGş. ErL`ťyfUSP47ĆCateninD1ĚŞńŤŤťÉ¨Żé@\AÖ. ú{ňwďć140Nď. s, 3, 2020.@@ |
| 8) | |JGş. AJf~AnňđÚwľ˝nňP~JoCIW[¤. TSMTP (Translational Science and Medicine Training Program) Symposium in Sapporo, Dy, 2, 2020. iľŇuj@@@@ |
| 7) | Kaneko, K., Nagao, N., Onaka, H., Shinzato, N., Kakeya, H. Detection of combined-culture specific constituents by the Molecular Networking and multivariate analyses. The 4th Kyoto Biomolecular Mass Spectrometry Society (KBMSS), Kyoto, Feb. 2020. |
| 6) | |JGş, Ý{[O, ~c-ŹŕVľ, ´Lž, gcšť, qij, Ąňú, ´{ł, ŕäëj. nŤvhbO^ŞqWIRŞńÜCMGĚJ¤. sĺwfBJCmx[ViMiPjězĺw@vOEăňn¤đŹT, s, 1, 2020.@@@ |
| 5) | qij, ŹěÍéŠ, ĽčR˘, X{Áž, ŕNłŞ, |JGş. HCmVR¨đ@\`[tÉľ˝´xxťÜ. sĺwfBJCmx[ViMiPjězĺw@vOEăňn¤đŹT, s, 1, 2020.@@@@@@@ |
| 4) | ž, ŕNłŞ, Ş[ž, c´, Ąž, ŹěS÷, |JGş. P~JoCIW[đîŐĆľ˝ErL`ťyfUSP47Ěś@\đÍ. sĺwfBJCmx[ViMiPjězĺw@vOEăňn¤đŹT, s, 1, 2020.@@@@ |
| 3) | qij, ž, |JGş. nňP~JoCIW[¤. sĺwfBJCmx[ViMiPjězĺw@vOEăňn¤đŹT, s, 1, 2020.@@@@ |
| 2) | |JGş. Lpś¨ŤKhĚJđuüľ˝ťwR~ jP[V¤. L@ŹĚj [gh2020iL@ŹťwŚďÖźxĺĂj, ĺă, 2, 2020. iľŇuj@@@@ |
| 1) | Kakeya, H. Continuing Fascination with Discovery Science: Phenotypic Screening to Chemical Biology. Mona Symposium 2020: Natural Product Chemistry and Medicinal Chemistry. Kingston, Jamaica, Jan. 2020. (plenary lecture) |
| 32) | |JGş. ÷ś¨ÔťwR~ jP[VĚđĆLpś¨ŤKhĚJ. VwpĚć¤uťwR~ jP[VĚteBAvEć6ńöJV|WE. Ąl, 12, 2019. iľŇuj@@@ |
|---|---|
| 31) | Kakeya, H. Chemical comunication research toward the development of useful chemical probes. The 4th A3 Roundtable Meeting on Asia Chemical Probe Research, Sendai, Nov. 2019. (Plenary lecture)@@@@ |
| 30) | Kakeya, H. Natural products-prompted chemical biology: Phenotypic screening and a new platform for target identification. The 6th Tishler-Omura Sympoium, Tokyo, Oct. 2019. (plenary lecture) [postponed due to the Typhoon no.19]@@@@ |
| 29) | Li, X., Hattori, A., Takahashi, S., Goto, Y., Harada, H., Kakeya, H. Inhibition of UCHL1 blocks proliferation and metastasis in HIF01 dependent tumor malignancy. 31th EORTC-NCI-AACR Symposium: International Conference on Molecular Targets and Cancer Therapeutics. Boston, MA, USA, Oct. 2019.@@@@ |
| 28) | Kakeya, H, Kishimoto, A., Umeta, H., Imaizumi, A., Kanai, M. Development of an injectable water-soluble anticancer drug CMG for oxaliplatin-resistant colorectal cancer with KRAS mutation. 31th EORTC-NCI-AACR Symposium: International Conference on Molecular Targets and Cancer Therapeutics. Boston, MA, USA, Oct. 2019.@ |
| 27) | Furutani, Y., Sudoh, M., Kakeya, H., Kojima, S. A small chemical compound CDM-3008 modulates cccDNA and suppresses HBV through induction of interferon-stimulated genes. 2019 International HBV Meeting. Melbourne, Australia, Oct. 2019.@@@@@ |
| 26) | Kuranaga, T., Kakeya, H. Highly sensitive labeling reagents inspired by a scarce marine natural product. 10th Korea-Japan Chemical Biology Symposium. Ishikawa, Oct. 2019.@@@@@ |
| 25) | Kanai, M., Kishimoto, A., Umeta, H., Imaizumi, A., Kakeya, H. Symposia 20 "Frontier in Molecular Target Therapy of Cancer": Development of a water-soluble prodrug CMG which inhibits proteasome activity through DYRK2 dependent manner. The 78th Annual Meeting of the Japanese Cancer Association, Kyoto, Sep. 2019. (invited)@@@@@ |
| 24) | Li, X., Hattori, A., Goto, Y., Harada, H., Kakeya, H. Involvment of UCHL1 in the HIF-1-dependent tumor cell malignancy in 3D cell culture model. The 78th Annual Meeting of the Japanese Cancer Association, Kyoto, Sep. 2019.@@@@@ |
| 23) | |JGş, qij. ŠRÉwÔňĂč. sĺwAJf~bNfC2019, s, 9, 2019.@@@@ |
| 22) | ´Lž, Ń@Gž, Poznaks, V. |JGş. á_fUąöqHIF-1jQŤđLˇéÂófvVyv`hverucopeptinĚSŹ. ć61ńVRL@ť¨˘_ď, L, 9, 2019.@@@@@ |
| 21) | Kakeya, H. Frontier research on chemical communications unveils the mystery of life science. The 27th International Society of Heterocyclic Chemistry Congress. Kyoto, Sep. 2019. (invited)@@@@ |
| 20) | cşüż, ěYî, qij, |JGş. RŞń¨żTbJXIhBĚűŠISʤ. ć39ńL@ŹZ~i[užúĚL@ŹđS¤lĚ˝ßÉv, ĺă, 8, 2019.@@@@@ |
| 19) | |JGş. ŠRÉwÔTCGXuŔF ťwR~ jP[VĚteBA¤. sĺwI[vLpX. s, 8, 2019.@@@@ |
| 18) | ĂJ@T, Ëű^q, ^äxq, óűËq, ŹŃJI, {ĄłK, éŘĄa, |JGş, Źę. cccDNAđ}§ˇéC^[tFláŞqť¨CDM-3008Ěěp@\. ć29ńREBXĂ@wďwpWďEď, _Ţě, 7, 2019.@@@@@ |
| 17) | ŕäëj, Ý{[O, ~c@ľ, Ąň@ú, |JGş. ILTv`ďRŤĚKRASĺ°ŞńÉΡéCMGËÜđp˘˝VKĄĂ@ĚJ. ć17ńú{Ő°îáwďwpWď, s, 7, 2019.@@@@@ |
| 16) | |JGş. ÷ś¨ÔťwR~ jP[VĚpÉćéVKś¨ŤKhĚJ¤. ć19ńú{`żČwďNďEć71ńú{×Eś¨wďĺď ŻNĺď. şÉ, 6, 2019.@iľŇuj@@@@@@ |
| 15) | |JGş, źşTę, qij, ěłT, ä{łĆ. ÷ś¨ÔťwR~ jP[VĚđE§äĆLpś¨ŤKhĚJ. VwpĚć¤uťwR~ jP[VĚteBAvEć5ńöJV|WE, ĺă, 6, 2019.@@@@@ |
| 14) | ăěăÄž, |JGş, ăuŹ, äŃWă, âVĄ@T, ˛Ąá, ĺ´Nś. [wwK@ĆPCAđÍđgÝíš˝P~JXy[XĚÂť. VwpĚć¤uťwR~ jP[VĚteBAvEć5ńöJV|WE, ĺă, 6, 2019.@ |
| 13) | |JGş. uV|WEEŞńĆhĺĚťwR~ jP[VĚđƧäv. nŤvhbO^ŞqWIRŞńÜCMGĚJ¤. ć23ńú{ŞńŞqWIĄĂwďwpWď. ĺă, 6, 2019. iľŇuj@@@@@ |
| 12) | cşüż, ěYî, qij, |JGş. RŞńŤđLˇé÷ś¨ăÓY¨TbJXIhBĚSʤ. ć86ńú{ŞÍťwďL@÷ʪͤ§kďEć110ńvŞŠŽ§äwďÍwĘvŞď ć36ńŻV|WE. s, 6, 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
| 11) | ŕqŤî, ˇöěfÔ, @ž, |JGş. á_fUąöqiHIFjjQť¨verucopeptinĚśŹâ`qNX^[ĚŻčĆVKŢĚĚTő. ć86ńú{ŞÍťwďL@÷ʪͤ§kďEć110ńvŞŠŽ§äwďÍwĘvŞď ć36ńŻV|WE. s, 6, 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
| 10) | |JGş. uV|WEEťwR~ jP[VĚteBAv. ÷ś¨ÔťwR~ jP[VĚpÉćéVKLpś¨ŤKhĚJ¤. ć19ńú{`żČwďNďEć71ńú{×Eś¨wď ŻNĺď. şÉ, 6, 2019. iľŇuj@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
| 9) | ĂJ@T, Ëű^q, ^äxq, óűËq, {ĄłK, éŘĄa, |JGş, Źę. C^[tFlĚŤđÂáŞqť¨CDM-3008ĚRHBVŤĚđÍ. ć26ńĚ×E¤ď. Ąl, 5, 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
| 8) | |JGş. uV|WEEŞń÷ŹÂŤĚđĆťĚÉüŻ˝ňwIAv[`ĆÍHHIF-1żĚđƧäÉüŻÄv. á_fVOiđWIĆľ˝nňP~JoCIW[. ú{ňwďć139Nď. çt, 3, 2019. iľŇuj@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
| 7) | |JGş. ˇúe[}V|WEuś˝ČwɨŻéŞqťwĚv[Xv. ťwR~ jP[VŞDčȡś˝Čw. ú{ťwďć99tGNďi2019j. _Ë, 3, 2019. iľŇuj |
| 6) | ó r˝, öčžY, źşTę, |JGş, öGN. Ą|{ɨŻéStreptomyces sp. HEK616Éćé5aTHQsĚśY@\, ú{_|ťwď2019Nxĺď. , 3, 2019. |
| 5) | Kakeya, H. Development of cryptic antifungal 5aTHQs targting cell membrane signaling. Asian Chemical Biology Initiative (ACBI) 2019 Yangon Meeting. Yangon, Myanmer, Jan. 2019. (invited)@@@@@@@@@@@@@@@@@@@@ |
| 4) | |JGş. uV|WEEVR¨nň`ú{ĚÝ𜊾˝VŞŹ`v@VR¨nňĚ đúľÄF÷ś¨ÔťwR~ jP[VĚp. ć402ńCBIwďiîńvZťwś¨wďjuď. , 1, 2019. iľŇuj@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
| 3) | Kakeya, H., Takahashi, N., Kishimoto, A., Imaizumi, A., Kanai, M. Development of an innovative water-soluble anticancer drug, curcumin mono-beta-D-glucuronide (CMG). The 1st International Symposium on Chemical Communication (ISCC2019). Tokyo, Jan. 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
| 2) | Nonaka, M., Fukuda, M.N., Kakeya, H. Rapid screening of antibody-binding peptides by combination of T7 phage display and next-generation sequencing technologies. The 1st International Symposium on Chemical Communication (ISCC2019). Tokyo, Jan. 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
| 1) | Jiang, Y., Lu, S., Hirai, G., Kato, T., Onaka, H., Kakeya, H. Towards the development of chemical communication molecules among microbes. The 1st International Symposium on Chemical Communication (ISCC2019). Tokyo, Jan. 2019.@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@@ |
| 33) | Kakeya, H., Kishimoto, A., Imaizumi, A., Kanai, M. Development of a synthetic water-soluble curcumin mono-beta-D-glucuronide (CMG), as an innovative anticancer prodrug targeting KRAS-NF-kappaB signaling pathway. 30th EORTC-NCI-AACR Symposium: International Conference on Molecular Targets and Cancer Therapeutics. Dublin, Ireland, Nov. 2018. |
|---|---|
| 32) | Nonaka, M., Kakeya, H., Fukuda, M. Drug delivery to malignant brain tumor by a peptide specific to Annexin A1. 30th EORTC-NCI-AACR Symposium: International Conference on Molecular Targets and Cancer Therapeutics. Dublin, Ireland, Nov. 2018. |
| 31) | |JGş. ăňiV[hŞqĚ˝lŤnoĆ×EŕWITőEŻč. ĺebNtH[. , 10, 2018. iľŇuj |
| 30) | Jiang, Y. L., Lu, S., Hirai, G., Kato, T., Onaka, H., Kakeya, H. Enhancement of saccharothriolides production and discovery of new derivatives by combined culture of a rare actinomycete Saccharothrix sp. and Tsukamurella sp. The 22th Symposium on Development and Application of Naturally Occurring Drug Materials. Kumamoto, Oct. 2018. |
| 29) | źşTę, R´î, JG, öčžY, ó r˝, öGN, |JGş. ÷ś¨ĚĄ|{Ĺžçęé5aTHQĚeaŤĆś¨Ť. ć60ńVRL@ť¨˘_ď. Ş, 9, 2018. |
| 28) | âşDĄ, ˛Ąş, ůěTî, ŹźTá, ěűłk, |JGş, ˇcTV, ź÷. A|g[VXUąŤVR¨cytotrienin AĚŹ¤. ć60ńVRL@ť¨˘_ď. Ş, 9, 2018. |
| 27) | |JGş, ěłT, qij. VR¨nňP~JoCIW[. sĺwAJf~bNfC2018, s, 9, 2018. |
| 26) | ´çG, Shan Lu, Yulu Jiang, Ĺ, źşTę, ž, |JGş. ć91ńú{śťwďĺď. s, 9, 2018. |
| 25) | ź´ń^, ž, |JGş. Calpain7Ě×EŕÇÝĚđÍ. ć91ńú{śťwďĺď. s, 9, 2018. |
| 24) | Ş[ž, ž, |JGş. yf˝Źx_IđÍđp˘˝ErL`ťyfUSP47ĚC[ĚćĚ@\đÍ. ć91ńú{śťwďĺď. s, 9, 2018. |
| 23) | |JGş. VR¨nňP~JoCIW[`úüŰÉŁšçęÄ`. 2018Nxić33ńjú{úüŰwďĺď. , 9, 2018. iľŇuj |
| 22) | ścŔš, ÉĄ¤, źşTę, gc Ť, |JGş. ˝uÇ`Źâ×ELˇÉ¨ŻéXtBSżĚdvŤ. yęâ`wtH[[ć51ń¤ńď. Ş, 9, 2018. (|X^[ÜđóÜ) |
| 21) | |JGş. ŠRÉwÔTCGXuŔF ťwR~ jP[VŞqĚäÉé. sĺwI[vLpX. s, 8, 2018. |
| 20) | |JGş. _ňĚnťE¤JŽüƝܝZpZ~i[FVK_ňĚJđuüľ˝P~JoCIW[¤. V[GV[oĹZ~i[. , 7, 2018.iľŇuj |
| 19) | Jiang, Y.L., Lu, S., Hirai, G., Kato, T., Onaka, H., Kakeya, H. Enhancement of saccharothriolide (STLs) production by combined-culture of Saccharothrix sp. and Tsukamurella sp. The 29th Meeting on Discovery and Development of New Drugs. Shizuoka, Jul. 2018. |
| 18) | cşSç, Shan Lu, c´, |JGş. á_fUąöqiHIFsjŤť¨żĚPŁE\˘čĆěp@đÍ. ć29ńVňnŹkbď. ĂŞ, 7, 2018. |
| 17) | |JGş. VR¨nňP~JoCIW[ĚçíĄ. ć53ńVR¨ťwkbď. ĺă, 7, 2018.iľŇuj |
| 16) | rŕPé, Cheng-Quin Pan, ścŔš, źşTę, |JGş. śĚVOiÉěpˇéVR¨ĚTő¤. ć53ńVR¨ťwkbď. ĺă, 7, 2018. |
| 15) | ÉĄk˘, qij, |JGş, e{qK. ZIl~hFĚŹ¤. ć53ńVR¨ťwkbď. ĺă, 7, 2018. |
| 14) | |JGş, źşTę, qij, ěłT, ä{łĆ. ÷ś¨ÔťwR~ jP[VĚđĆLpś¨ŤKhĚJ. VwpĚć¤uťwR~ jP[VĚteBAvEć3ńöJV|WE. , 6, 2018. |
| 13) | |JGş. uťwR~ jP[VĚteBAvđN_Éľ˝nňP~JoCIW[. VwpĚć¤użNIeBŞđŤžŠˇś˝ťŰvć4ńĚćďc. şÉ, 6, 2018. iÁĘuj |
| 12) | ĂJ@T, |JGş, Źę. [NVbvuB^ĚVKĄĂňĚTőĚťóvFhbOt[ĚŔťđÚwľ˝cccDNA}§ÜCDM-3008ĆGeJrĆĚšpÉćéHBVÄŤťĚ}§. ĺă, 6, 2018. iÁĘuj |
| 11) | Lu, S., Nishimura, S., Ito, M., Kato, T., Kakeya, H. Discovery of pre-saccharothriolide X from the rare actinomycet Saccharothrix sp. The 13th Annual Meeting of Japanese Society for Chemical Biology, Tokyo, Jun. 2018. |
| 10) | Kakeya, H. Microbial metabolites targeting microenvironment: a cell membrane sigaling modulator and a hypoxia-response modulator. The 9th Japan-Korea chemical biology symposium, Incheon, Korea, May, 2018. (invited) |
| 9) | Ogawa, Y., Kakeya, H. Screening of sensitizers derived from microbial metabolites to induce apoptosis in pancreatic cancer cells. The 9th Japan-Korea chemical biology symposium, Incheon, Korea, May, 2018. |
| 8) | Nonaka, M., Kakeya, H., Fukuda, M. Identification of binding peptides against IgE from human myeloma U266 cells. The 9th Japan-Korea chemical biology symposium, Incheon, Korea, May, 2018. |
| 7) | Li, X.B., Goto, Y., Hattori, A., Harada, H., Kakeya, H. Study on the UCHL1-HIF-1 axis toward development of molecular targeted anticancer drugs. The 22th Annual Meeting of the Japanese Association for Molecular Target Therapy of Cancer (JAMTTC), Tokyo, May, 2018. |
| 6) | Kanai, M., Imaizumi, A., Kakeya, H. Development of a water-soluble curcumin monoglucronide (CMG) as a novel anticancer prodrug targeting KRAS-NF-kappa B signaling pathway. Global Academic Programs (GAP) conference, Stockholm, Sweden, May, 2018. (invited) |
| 5) | |JGş. uˇúéćEP~JoCIW[¤ÁŹĚ˝ßĚś¨ŤŞqĚŠíŞv\÷ś¨ÔťwR~ jP[VĚäɧŢ\. ú{ťwďć98tGNď. çt, 3, 2018. iľŇuj |
| 4) | črś, {Nž, ž, Źę, |JGş. TGF-ŔVOi`BjQÜKUSC-Y244ÍTGF-ŔÉćéăçÔt]ˇđ}§ˇé. ú{ňwďć138Nď, ŕň, 3, 2018. |
| 3) | |JGş. uV|WEFąęŠçĚVR¨TCGXv\P~JXy[Xg[íŞF÷ś¨Ą|{@yŃPDSS (Precurso-Directed in situ Synthesis)@\, ú{_|ťwď2018Nxĺď. źĂŽ, 3, 2018. iľŇuj |
| 2) | |JGş. ÷ś¨ÔťwR~ jP[VĚpÉćéP~JXy[Xg[íŞ. VwpĚć¤uťwR~ jP[VĚteBAvEć2ńöJV|WE. s, 2, 2018. iľŇuj |
| 1) | Lu, S., Nishimura, S., Ito, M., Kato, T., Kakeya, H. Expansion of chemical space in saccharothriolides: Precursor-directed in situ synthesis (PDSS) in a rare actinomycete Saccharothrix sp. Natural Product Discovery & Development in the Genomic Era (Natural Products 2018), Clearwater, FL, USA. Jan. 2018. |
| 26) | |JGş. n_ňCmx[VđnˇéP~JoCIW[űŞ. _ňfUC¤ďiĺĂFú{_ňwďE_ňfUC¤ďj. , 11, 2017. iľŇuj |
|---|---|
| 25) | Ąň ú, ´Lž, őŕpé, ŕäëj, ´{ ł, qěIĄ, ĂcFÍ, |JGş. @\ŤHifŢĚăňiÖĚWJđÚwľ˝nňP~JoCIW[. ć7ńHiňwV|WE. s, 10, 2017. iľŇuj |
| 24) | ´Lž, Ń Gž, Poznaks, V., |JGş. ăňťwIWJđwüľ˝verucopeptinĚSʤ. ć35ńfBViP~Xg[V|WE. źĂŽ, 10, 2017. |
| 23) | Furutani, Y., Toguchi, M., kakeya, H., Kojima, S. Combinatorial treatment of CDM/iCDM and entecavir for efficient suppression of cccDNA. 2017 International HBV Meeting: The Molecular Biology of Hepatitis B viruses, Washington, DC, USA. Sep. 2017. |
| 22) | źşTę, gş Ę, R´î, |JGş. VRL@ť¨Ě\˘đÍĆNMRVOiĚdĄ. ć18ńNMR¤ď. aĚR, 9, 2017. iľŇuj |
| 21) | ścŔš, ÉĄ¤, źşTę, |JGş. XtBSżĚ@\đžđÚwľ˝ťwâ`wIđÍ.FGLm}CVŢĚćžĆťĚ\ť^. yęâ`wtH[ć50ń¤ńď. , 9, 2017. |
| 20) | źşTę, żqŤl, |JGş, źiÎ÷, ĺ÷łq, śŁ`v, Carvalho, S., Cortes, J., Ribas, J. Xe[đWIɡéR^Űť¨ZIl~hÉćé×EÇŮí. yęâ`wtH[ć50ń¤ńď. , 9, 2017. |
| 19) | şşsl, öčžY, R´î, źşTę, ó r˝, |JGş, öGN. Ą|{ÉćÁÄśYłęéegqhLmť¨ĚđÍ. ć32ńú{úüŰwďĺď, ˇě, 9, 2017. |
| 18) | |JGş. ŠRÉwÔTCGXuŔF÷ś¨ÔťwR~ jP[VĚäÉé. sĺwI[vLpX. s, 8, 2017. |
| 17) | ŕäëj, ŹŕV ľ, Ąň ú, ´Lž, |JGş. [NVbvuAJf~ARŞńňJĚiWvFvhbO^NN~đp˘˝VKRŞńňĚJ. ć15ńú{Ő°îáwďwpWď. şÉ, 7, 2017. |
| 16) | ŹěÍéŠ, @áX, @ž, ăĄeq, XéęÍă, ˝ŞáÁ°, ´c@_, |JGş. ŞqWIRŞńÜJđwüľ˝ErL`ťyfUCHL1jQÜĚTő¤. ć28ńVňnŹkbďužłĆnňĚCmx[Vv. ĂŞ, 7, 2017. |
| 15) | ścŔš, ÉĄ¤, Ącq˝, źşTę, |JGş. ×EżđWIơ靨ĚXN[jOyѝ̍]ż. ć28ńVňnŹkbďužłĆnňĚCmx[Vv. ĂŞ, 7, 2017.(DG\Üi§ăÜjđóÜ) |
| 14) | Lu, S., Nishimura, S., Ito, M., Kato, T., Kakeya, H. Novel natural products, saccharothriolides, from rare actinomycete Saccharothrix sp. and precursor-directed in situ synthesis (PDSS) of thier analogs. The 10th Anniversary Symposium of Division of Bioinformatics and Chemical Genomics, Graduate School of Pharmaceutical Sciences, Kyoto University, Kyoto, July, 2017. |
| 13) | ŕqŤî, | d, ˇöěfÔ, Îěśm, g˝ěa÷, Ü\ëV, |JGş. P~JXy[Xg[đwüľ˝śŹHwI¤. sĺwĺw@ňw¤ČăňnŹîńČwęU10üNLOV|WE. s, 7, 2017. |
| 12) | Ş[ž, c´, ž, |JGş. ErL`ťyfUSP47Ě|rL`˝Áť@\ĚđžĆjQÜTőnĚ\z. sĺwĺw@ňw¤ČăňnŹîńČwęU10üNLOV|WE. s, 7, 2017. |
| 11) | ´Lž, Ń@Gž, Viktors Poznacks, |JGş. á_fUąöqiHIFsjjQÜJđwüľ˝verucopeptinĚSʤ. sĺwĺw@ňw¤ČăňnŹîńČwęU10üNLOV|WE. s, 7, 2017. |
| 10) | |JGş. ÷ś¨Ą|{@ĚpÉćénňP~JoCIW[. ć12ńťwśÔw¤ď. Ů, 6, 2017. iľŇuj |
| 9) | ĂJ@T, |JGş, Źę. V|WEuB^̤ĚVWJvFcccDNA}§ÜCDM/iCDMĆGeJrĆĚšpřĘĚđÍ. ć53ńú{Ěwďď. L, 6, 2017. |
| 8) | Lu, S., Nishimura, S., Ito, M., Kato, T., Kakeya, H. Generation of saccharothriolide analogs by precursor-directed in situ synthesis (PDSS) and their SAR study. The 12th Annual Meeting of Japanese Society for Chemical Biology, Sapporo, June, 2017. |
| 7) | źşTę, ÉĄ¤, ´Lž, |JGş. T|jĆXe[ĚŞqÔÝěpɨŻéYť f˝ĘĆ _îĚdvŤ. ú{P~JoCIW[wď ć12ńNď, Dy, 6, 2017. |
| 6) | |JGş. ŠRÉwŃA´đRđŤAˇčđné. ú{wpUťďiJSPSjuú{ɨŻéP~JoCIW[ĚVWJvÉÖˇéYwŚÍ¤ĎőďiJSPSć189ĎőďjEH29Nxć1ńčáď, , 5, 2017.iľŇuj |
| 5) | Li, X.B., Takahashi, S., Hattori, A., Goto, Y., Morinobu, A., Hiraoka, M., Harada, H., Kakeya, H. Chemical biology research on the UCHL1-HIFs axis toward development of molecular targeted anticancer drugs. SKO Symposium 2017 (Joint Symposium 2017 of Seoull Univ., Kyoto Univ., and Osaka Univ.), Osaka, May, 2017. |
| 4) | @áX, ž, ăĄeq, XéęÍă, , ˝ŞáÁ°, ´c@_, |JGş. ĺw@śV|WEuňwŞń¤ĚWƢđ湡éáčŞń¤Ņ̌ívFUCHL1-HIFŤťoHđWIĆľ˝ŞqWIRŞńÜJ¤. ú{ňwďć137Nď. ĺä, 3, 2017. iľŇuj |
| 3) | Ń@ą˝, ´Lž, ěYî, Ëű^q, ˛ĄTü, ĂJ@T, Źę, |JGş. VKB^ĚĄĂňnťÉüŻ˝CDMsĚ\˘ŤÖ¤. ú{ňwďć137Nď. ĺä, 3, 2017. |
| 2) | |JGş. uV|WEF_|ťwŠçMˇé˘ă^VR¨ťwv\AJf~AnňɨŻé\ť^XN[jOƢăVR¨ťw\. ú{_|ťwď2017Nxĺď. s, 3, 2017. iľŇuj |
| 1) | |JGş. nňP~JoCIW[¤űŞF\ť^XN[jOĆV[hŞqJ. rbOf[^ěŽ^nňVXe¤_Eć3ńV|WE. cä`mĺw. Ąl, 3, 2017. iľŇuj |
| 24) | @áX, ăĄeq, ž, ˝ŞáÁ°, ´c@_, |JGş. VKŞqWIRŞńÜJđwüľ˝UCHL1-HIFŤťoHjQÜXN[jOnĚ\z. ć75ńú{ŕwďwpď. Ąl, 10, 2016. |
|---|---|
| 23) | źşTę, R´î, JG, öčžY, ó r˝, öGN, |JGş. ÷ś¨ĚĄ|{Ĺžçęé5aTHQĆstreptoaminalĚ\˘Ć\˘. ć21ńVRň¨ĚJĆpV|WE. çt, 10, 2016.iľŇuj |
| 22) | Kojima, S., Furutani, Y., Kakeya, H. Screening of novel cccDNA modulator compounds, iCDMs.The 2016 International HBV Meeting: The Molecular Biology of Hepatitis B Viruses. Seuol, Korea, Sep. 2016. |
| 21) | Îěśm, Ąě@ăÄ, }äşž, éŘT, °O@ź, |JGş. ń{\[Ťyv`hŹyfĚIđIxťZpĚJĆvŹ@\đÍVXeĚ\z. ć58ńVRL@ť¨˘_ď. ĺä, 9, 2016. |
| 20) | ź{×M, úäěa_, ˘iëO, |JGş, ŃYńY. XvCVOjQÜRQN-18690A (18-deoxyherboxidiene)ĚSŹ. ć58ńVRL@ť¨˘_ď. ĺä, 9, 2016. |
| 19) | Ş[ž, ÂŘ@L, @ž, |JGş. ErL`ťyfUSP47Ě|rL`˝ÁťÉÖíéŞqŕĚćĚŻč. ć89ńú{śťwďĺď. ĺä, 9, 2016. |
| 18) | ăÉî, ŹŃSq, @ž, |JGş. ErL`ťyfjQÉćéHIF-1ťx̧ä. ć89ńú{śťwďĺď. ĺä, 9, 2016. |
| 17) | ÎěśmA}äşžAĄě@ăÄA|JGş. ń{\[Ťyv`hŹyfĚÔ I@\đÍZpĚJ. ć10ńoCIÖAťwV|WE. Îě, 9, 2016. |
| 16) | |JGş. uVľ˘R^ŰňV[hJĆKgĺíŞv\R^ŰňJĚ˝ßĚP~JoCIW[¤űŞFV[hŞqJĆJjYđÍ. ZpîńŚďZ~i[. , 8, 2016.iľŇuj |
| 15) | Kakeya, H. Development of new anticancer drugs targeting TGF-Ŕ and HIF signaling pathway. 2016 BIO International Convention. San Francisco, CA, USA, Jun. 2016. |
| 14) | |JGş. nňP~JoCIW[FśĚŕ÷ŹÂŤVOi̧ä. VKfŢTő¤ďEć15ńZ~i[. Ąl, 6, 2016. iľŇuj |
| 13) | JG, R´î, źşTę, |JGş. śĚĆÝěpˇé5aTHQŢĚ\˘ŤÖ¤Ćuőv[uJ. ú{P~JoCIW[wď ć11ńNď. s, 6, 2016. |
| 12) | Źę, |JGş, ĂJ T, čp÷, źYam. ˘ăś˝îŐZpđp˘˝B^̧łĚ˝ßĚnň¤. ć26ńREBXĂ@wďď. ¤m, 5, 2016. |
| 11) | Źę, ĂJ T, |JGş. V|WEEB^̤ĚUp-To-DateFC^[tFlŤđÂáŞqť¨CDMÉćécccDNA}§ěpĚđÍ. ć52ńú{Ěwďď. çt, 5, 2016. |
| 10) | |JGş. TGF-Ŕ¨ćŃá_fVOiđWIĆľ˝VKŞńĄĂňĚJ¤. ć15ńŰoCIeNmW[WŚďiBIOtech 2016j. , 5, 2016. |
| 9) | Kakeya, H. Microbial metabolites-prompted chemical biology: Phenotypic screening and a new platform for target identification. The Fifth Symposium of RIKEN-Max Planck Joint Research Center for System Chemical Biology. Berlin, Germany, Apr. 2016. iľŇuj |
| 8) | ´Lž, Ń@Gž, |JGş. á_fUąöqiHIFjjQŤđLˇéÂófvVyv`hverucopeptinĚSʤ. ú{ňwďć136Nď. Ąl, 3, 2016. |
| 7) | R´î, źşTę, öčžY, ó r˝, öGN, |JGş. ĺw@śV|WEFżŤVR¨Ěp\úüŰĄ|{tćčŠoľ˝VKAJChQÉÖˇé¤. ú{ňwďć136Nď. Ąl, 3, 2016. iľŇuj |
| 6) | Cornelio, K., Matsumori, N., Murata, M., Nishimura, S., Kakeya, H., Yoshida, M., Matsunaga, S. Examination of apossible mechanism for the membrane translocation of the marine sponge-derived bioactive metabolite TNM-A. ú{ťwď96tGNďi2016j, s, 3, 2016. |
| 5) | şşml, öčžY, R´î, źşTę, ó r˝, |JGş, öGN. Ą|{ÁŮIÉśYłęéegqhLmśŹâ`qĚđÍ. ú{_|ťwď2016Nxĺď. Dy, 3, 2016. |
| 4) | Nishimura, S., Ito, A., Kakeya, H. Strict recognition of membrane lipids by a sea cucumber saponin, holotoxin B. Gordon Research Conference-Marine Natural Products-, Ventra, CA, USA, Mar., 2016. |
| 3) | gş@Ę, źşTę, ĺËšD, @ž, |JGş. Eá_fUąöq(HIF)jQŤđLˇéverucopeptinĚ\˘đÍĆěp@đÍ, VwpĚć¤uVR¨P~JoCIW[FŞqWIĆŤ§ävnć~jV|WEisj, s, 2, 2016. |
| 2) | Kakeya, H. Academic drug discovery research: Phenotypic screening and target identification. University of Bordeaux-Kyoto University Mini-Symposium on Biomolecular Science. Kyoto, Jan. 2016. iľŇuj |
| 1) | Nishimura, S., Moriyama, A., Katagiri, N., Takahashi, N., Kakeya, H. In vivo linking of membrane lipids and membrane proteins using amphiphilic lipid probes. The 8th Takeda Science Foundation Symposium on PharmaSciences: Biomolecule-Based Medicinal Science: Featuring Mid-Size Drugs. Osaka, Jan. 2016. |
| 31) | Kakeya, H. Natural products-based academic drug discovery. International symposium on natural products chemistry and chemical biology 2015. Hawaii, USA, Dec., 2015. iľŇuj |
|---|---|
| 30) | Kakeya, H. Natural products-prompted chemical biology; Phenotypic screening and target identification. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. iľŇuj |
| 29) | Lu, S., Nishimura, S., Hirai, G., Ito, M., Kawahara, T., Izumikawa, M., Sodeoka, M., Shin-ya, K., Tsuchida, T., Kakeya, H. Saccharothliolides A-C, novel phenyl-substituted 10-membered macrolides from a rare actinomycete Saccharothrix sp., identified by HPLC-MS profiling of microbial metabolites. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
| 28) | Takahashi, N., Hayashi, H., Kakeya, H. Synthetic study on the antitumor cyclodepcipeptide metabolite, verucopeptin. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
| 27) | Sugiyama, R., Nishimura, S., Ozaki, T., Asamizu, S., Onaka, H., Kakeya, H. 5-Alkyl-1,2,3,4-tetrahydroquinolines (5aTHQs), new membrane-interacting lipophilic metabolites, produced by combined-culture of Streptomyces nigrescens and Tsukamurella pulmonis. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
| 26) | Nishimura, S., Sugiyama, R., Fujita, K., Ito, S., Sakanishi, K., Iwabuchi, Y., Kanoh, N., Matsumori, N., Kakeya, H. Structure and function of heronamides, polyene macrolactams from marine-derived actinomycetes . The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
| 25) | Ishikawa, F., Miyamoto, K., Konno, S., Kasai, S., Kakeya, H. Accurate detection and manipulation of adenylation domain functions in nonribosomal peptide synthetases by an enzyme-linked immunosorbent assay system using active site-directed probes for adenylation domains. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
| 24) | Konno, S., Ishikawa, F., Suzuki, T., Dohmae, N., Kakeya, H. Profiling of nonribosomal peptide synthetase activities using active site-directed proteomic probes for adenylation domains. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
| 23) | Nishimura, S., Kakeya, H. Sterol-targeting antibiotics and the balance of membrane trafficking. The International Chemical Congress of Pacific Basin Societies 2015 (PACIFICHEM 2015). Hawaii, USA, Dec., 2015. |
| 22) | Yoshimura, A., Nishimura, S., Otsuka, S., Hattori, A., Kakeya, H. Studies on the microbial metabolite verucopeptin, an inhibitor of HIF-signaling pathway. SKO Symposium 2015 (Joint Symposium 2015 of Seuol Univ., Kyoto Univ., and Osaka Univ.), Seoul, Nov., 2015. |
| 21) | }äşž, Îěśm, |JGş. ń{\[Ťyv`hŹyfĚ|óăCüđWIĆľ˝ťwv[uĚJ. ć65ńú{ňwďßExďEĺď. 10, ĺă, 2015. |
| 20) | Îěśm, ĄěăÄ, }äşž, éŘT, °Oź, |JGş. ŹŹŞqť¨QÉćéAfj[VhCĚIđIWŻť¨ćŃvt@COÖĚWJ. ć9ńoCIÖAťwV|WE. 9, F{, 2015.iuÜđóÜj |
| 19) | ź÷, ÉrĆ, Dž, âźq˝, âşDĄ, Ącq˝, R´î, źşTę, |JGş. Heronamides A-C ĚSŹĆ\˘üůA¨ćŃ\˘ŤÖ. ć57ńVRL@ť¨˘_ď. Ąl, 9, 2015. |
| 18) | Lu, S., Nishimura, S., Hirai, G., Ito, M., Kawahara, T., Izumikawa, M., Sodeoka, M., Shin-ya, K., Tsuchida, T., Kakeya, H. Studies on Saccharothriolides A-C, Novel Phenyl-substituted 10-Membered Macrolidesfrom a Rare Actinomycete Saccharothrix sp. 57th Symposium on the chemistry of natural products. Yokohama, Sep. 2015. |
| 17) | lűcIă, Ącq˝, űPËG˘, źşTę, ˝Ş^°, ´c_, |JGş. IDH3ż\HIF-1oHđ§äˇéś¨Ť¨żĚTő¤. ć26ńVňnťkbď. ĂŞ, 9, 2015. (DG\Üi§ăÜjđóÜ) |
| 16) | |JGş. żln˘^nňP~JoCIW[, ć7ńňw̢đlŚésV|WEuňEHEăAgÉćéżln˘^nň¤ĚteBAv, s, 8, 2015. |
| 15) | |JGş. sĺwI[vLpXEňwEÍ[öĆ. nňEçňÖ̧íFŠRÉwÔP~JoCIW[¤. s, 8, 2015. |
| 14) | |JGş. V|WEunňĚŤv. nňP~JoCIW[FV[hŞqJĆŞqvt@CO. ć63ńú{ťwĂ@wďď. , 6, 2015. iľŇuj |
| 13) | ĄěăÄ, Îěśm, éŘT, °O ź, |JGş. Afj[VhCÉΡéŤĘwü^v[uđp˘˝ń{\[Ťyv`hŹyfŤĚvt@CO. ć15ńú{`żČwďNď, ż, 6, 2015. |
| 12) | Nishimura, S., Sugiyama, R., Fujita, K., Kakeya, H. Abnormal cell wall deposition by heronamides, small molecules targeting phospholipids possessing saturated hydrocarbon chain. Pombe 2105 (8th International Fission Yeast Meeting), Kobe, Japan, June, 2015. |
| 11) | }äşž, Îěśm, |JGş. ń{\[Ťyv`hŹyfĚSĚ^pNżđWIĆľ˝áŞqv[uĚJ. ú{P~JoCIW[wďEć10ńNď, ĺä, 6, 2015. |
| 10) | ĄěăÄ, Îěśm, éŘT, °Oź, |JGş. Afj[VhCÉΡéŤĘwü^v[uđpľ˝ń{\[Ťyv`hŹyfŤĚvt@CO. ú{P~JoCIW[wďEć10ńNď, ĺä, 6, 2015.[DG|X^[ÜđóÜ] |
| 9) | |JGş. śĚŕ÷ŹÂŤVOiđWIĆľ˝nňP~JoCIW[. nňňtH[Eć58ńkbď. , 5, 2015. iľŇuj |
| 8) | |JGş. ˇúe[}V|WEiú{ťwďECujOZbVjuśŹ}Vi[ĆVR¨P~JoCIW[ĚZÉćéVWJv. ćąIVR¨P~JoCIW[F\ť^XN[jOĆWITőEŻč. ú{ťwďć95tGNď. çt, 3, 2015. iľŇuj |
| 7) | Kakeya, H. Technologies bridging metabolome and clock -Chemical biology for drug discovery; seed molecules development and target identification-. International Symposium on RNA and Clock: Epigenetic Landscape in Biological Rhythms. Hyogo, Mar. 2015. iľŇuj |
| 6) | Ącq˝, R´î, źşTę, |JGş. Heronamide A¨ćŃBĚśŹ@\ÉÖˇé¤. ú{ňwďć135Nďi_Ëj. _Ë, 3, 2015. |
| 5) | ĄěăÄAÎěśmAéŘTA°OźA|JGş. Afj[VhCÉΡéŤĘwü^v[uĚJ. ú{ňwďć135Nďi_Ëj. _Ë, 3, 2015. [DG\ÜđóÜ] |
| 4) | }äşž, Îěśm, |JGş, ń{\[Ťyv`hŹyfĚŘv`WSĚ^pNżđWIĆľ˝v[uĚJ¤. ú{ňwďć135Nďi_Ëj. _Ë, 3, 2015. |
| 3) | Îěśm, ĄěăÄ, |JGş. ŤĘwü^v[uÍAfj[VhCđIđIÉWݎé. ć17ńś˝ťw¤ď, m, 1, 2015. |
| 2) | Sugiyama, R., Nishimura, S., Ozaki, T., Onaka, H., Kakeya, H. 5-Alkyl-1,2,3,4-tetrahydroquinolines, membrane-interacting lipophilic metabolites, found in a unique combined culture of Streptomyces sp. and Tsukamurella pulmonis. Natural Products 2015; Natural product discovery & development in the post genomic era [Organized by Society for Industrial Microbiology and Biotechnology (SIMB)], San Diego, CA, USA, Jan. 2015. |
| 1) | Kakeya, H., Yoshimura, A., Sugiyama, R., Kishimoto, S., Nishimura, S., Hattori, A., Ishikawa, F., Yomoda, Y., Lu, S., Katagiri, N., Shimada, S., Seto, E., Hayashi, H., Takahashi, N., Harada, H. Chemical Biology for modulators targeting cancer microenvironment and cell membrane signaling. Natural Products 2015; Natural product discovery & development in the post genomic era [Organized by Society for Industrial Microbiology and Biotechnology (SIMB)] , San Diego, CA, USA, Jan. 2015. |
| 32) | |JGş. V|WEEmgĚVWJF nňV[YJđwüľ˝VR¨P~JoCIW[ -\ť^XN[jOĆWITőEŻč-. ć20ńVRň¨ĚJĆpV|WE. , 11, 2014.iľŇuj |
|---|---|
| 31) | Îěśm, ĄěăÄ, |JGş. Afj[VhCÉΡée[[ChP~JxO@ĚJ. ć20ńVRň¨ĚJĆpV|WE. , 11, 2014. |
| 30) | Nishimura, S., Sugiyama, R., Matsumori, N., Kakeya, H. Marine natural products targeting cell membrane. 3rd Annual Conference of the International Chemical Biology Society (ICBS2014), San Francisco, CA, USA, Nov. 2014. |
| 29) | Ý{^Ą, źşTę, ž, g˝ěa÷, Ü\ëV, |JGş. AVOAjW\˘đLˇéVKVftHAchlorocatechelinŢĚPŁE\˘čASŹA¨ćŃś¨Ť. ć56ńVRL@ť¨˘_ď. m, 10, 2014. |
| 28) | ĄěăÄ, Îěśm, |JGş. ŤĘwü^v[uđp˘˝Afj[VhCĚIđIWŻť. ć8ńoCIÖAťwV|WE. 9, ŞR, 2014. |
| 27) | Îě śm, {{ á, Ąě ăÄ, }ä şž, |J Gş. iťŞqHwđwüľ˝Afj[VhCÉΡéELISA@ĚJ. ć8ńoCIÖAťwV|WE. 9, ŞR, 2014. |
| 26) | żqŤl, źşTę, zqq, gcŤ, |JGş. AÉćé×EXe[b`hCĚÇݧä@\Ěđž. yęâ`wć47ń¤ńď. , 9, 2014. |
| 25) | Kakeya, H. Chemical biology for drug discovery and target identification. IUPAC2014 & 248th ACS (American Chemical Society) National Meeting, San Francisco, CA, USA, Aug. 2014. (ľŇu) |
| 24) | ÂŘL, pŃÔ, ŹŃSq, ž, |JGş.@ErL`ťyfUSP47ĚŤťÉ¨ŻéC[ĚćĚđ. ć19ńú{aÔveA[[wďwpWď. ĺă, 8, 2014. |
| 23) | |JGş. sĺwI[vLpXEňwEÍ[öĆ. nňEçňɧŢP~JoCIW[. s, 8, 2014. |
| 22) | XR˛, źşTę, |JGş. śĚđWIơéVR¨Ěěp@đÍđwüľ˝LiDEL@ĚJ. ú{P~JoCIW[wďEć9ńNď. ĺă, 6, 2014.[DG|X^[ÜđóÜ] |
| 21) | öčžY, R´î, źşTę, ó r˝, |JGş, öGN. Ą|{đpľ˝VKegqhLmŢĚPŁĆťĚśŹÉÖˇé¤. 2014Nxić29ńjú{úüŰwď. ďé, 6, 2014. |
| 20) | Konno, S., Ishikawa, S., Kakeya, H. Chemical labeling of adenylation domains in nonribosomal peptide synthetase. Gordon Research Conferences: Bioorganic Chemistry-Global Challenges in the 21st Century-. Andover, NH, USA, June, 2014. |
| 19) | Ishikawa, F., Konno, S., Kakeya, H Highly selective detection method for nonribosomal peptide synthetase using cocktails of active-site probes for adenylation domains. Gordon Research Conferences: Bioorganic Chemistry-Global Challenges in the 21st Century-. Andover, NH, USA, June, 2014. |
| 18) | |JGş. nňV[YJđwüľ˝VR¨P~JoCIW[. VR¨P~JoCIW[ -ŞqWIĆŤ§ä-Eć6ńöJV|WE. ¤m, 5, 2014.iľŇuj |
| 17) | Ý{^Ą, źşTę, ž, g˝ěa÷, Ü\ëV, |JGş. VKVftHAchlorocatechelinŢĚPŁE\˘čĆS\]ż. śČČuťwĂ@îŐxŽv ć3ńV|WEuAJf~AŠçĚRŞńÜnňÉüŻÄv. Ťę, 5, 2014 |
| 16) | c´, gşĘ, ŔcM, ´Lž, źşTę, ž, |JGş. ŞńŞqWInňđwüľ˝á_fUąöq(HIF)jQÜĚTőEJ¤. śČČuťwĂ@îŐxŽv ć3ńV|WEuAJf~AŠçĚRŞńÜnňÉüŻÄv. Ťę, 5, 2014. |
| 15) | |JGş. V|WEEVR¨P~JoCIW[(2)FPEoCIP~Xg[F÷ś¨@\đpľ˝nňP~JoCIW[¤. ú{ňwď134Nď. F{, 3, 2014.iľŇuj |
|---|
| 14) | Ý{^Ą, źşTę, ž, g˝ěa÷, Ü\ëV, |JGş. StreptomycesŽúüŰćčŠoľ˝f´qÜLVKVftHAĚPŁE\˘č. ú{ňwď134Nď. F{, 3, 2014. [DG\ÜđóÜ], [Nď\nCCgÉĚđ] |
|---|
| 13) | R´î, źşTę, öčžY, öGN, |JGş. egqhLmiđLˇéVKúüŰăÓ¨Ě\˘˝lŤĆś¨Ť. ú{ňwď134Nď. F{, 3, 2014. [DG\ÜđóÜ] |
|---|
| 12) | gşĘ, źşTę, ĺËŃD, ž, |JGş. á_fUąöq(HIF)ŤťoHđjQˇéverucopeptinĚěp@đÍ. ú{ňwď134Nď. F{, 3, 2014. |
|---|
| 11) | ŔcM, ęcLü, rěž, c´, ž, źşTę, ĺÎ^ç, ĄäMF, |JGş. VKá_fUąöqHIFjQÜĚTőĆ\˘ŤÖ¤. ú{ňwď134Nď. F{, 3, 2014. |
|---|
| 10) | ´Lž, |JGş. RîáŤÂófvVyv`hverucopeptinĚSʤ. ú{ňwď134Nď. F{, 3, 2014. |
|---|
| 9) | ĄěăÄ, Îěśm, |JGş. őeaŤv[uđpľ˝Afj[VhCÉΡéKhËśIWŻť. ú{ňwď134Nď. F{, 3, 2014 |
|---|
| 8) | ëěžF, źşTę, ÁĄ˝, |JGş. Chaetoglobosin DÍROSYśÉćč×EĚZťđjQˇé. ú{ňwď134Nď. F{, 3, 2014. |
|---|
| 7) | ŹŃSq, ž, ÂŘL, |JGş. EUrm1ťŤĚo¨ćŃŞqŻč. ú{ňwď134Nď. F{, 3, 2014. |
|---|
| 6) | ÂŘ@L, p@ŃÔ, ŹŃ@Sq, @ž, |J@Gş. ErL`ťyf(USP)47ĚŞqŕhCĚ@\đÍ. ú{ňwď134Nď. F{, 3, 2014. |
|---|
| 5) | ŞşMq, ťězę, â×j, ˝ěG, ŔŘër, nçłYę, yäC, ĄníL, ´i, źäl, ŕ_cFq, Ąňú, ´{ł, |JGş, ac[š, ĂÍ, ˇJě_ń, X{Bç. łě×tNXI[o[2dÓąÉćÁÄTheracurminÍźĚNN~ťÜćčŕDę˝zűřŚĚüăŞÝçę˝. ú{ňwď134Nď. F{, 3, 2014. |
|---|
| 4) | Sugiyama, R., Nishimura, S., Matsumori, N., Tsunematsu, Y., Hattori, A., Kakeya, H. Mode of action of heronamides, polyene macrolactams from a marine-derived Streptomyces sp. Gordon Research Conferences: Marine natural products- from discovery to human health-. Ventura, CA, USA, Mar. 2014. |
|---|
| 3) | |JGş. nňEçňɧŢP~JoCIW[FňwÖĚUi˘´Čj˘. kq|NeXäy, s{§kwZ. 3, 2014.iľŇuj |
|---|
| 2) | Yoshimura, A., Nishimura, S., Otsuka, S., Hattori, A. Kakeya, H. Mode of action of vercopeptin, an inhibitor of HIF-signaling pathway isolated from an actinomycete. The 12th International Student Seminar (12th ISS), Kyoto Univeristy. Kyoto, Feb. 2014. |
|---|
| 1) | |JGş. ˝Ź25NxsňČĺwć2ńnňČwteBAV|WE. nňP~JoCIW[F\ť^XN[jOĆWIŻč. s, 2, 2014.iľŇuj |
|---|
| 21) | ëěžF, źşTę, ÁĄ ˝, |JGş. ZăÓÍAN`jQÜÖĚ´óŤđ㸳šé. ć5ńHiňwV|WE. s, 11, 2013. |
|---|---|
| 20) | źşTę, żqŤl, zqq, gcŤ, |JGş. Xe[b`×EhCĚ`Ź@\ĚđÍ. ć5ńHiňwV|WE. s, 11, 2013. [DG\ÜđóÜ] |
| 19) | {{á, Îěśm, Ń@L, |JGş. óŰNeosartoryaŽRvjî]ÚyfÉÖˇé¤. ć5ńHiňwV|WE. 11, s, 2013. |
| 18) | }äşž, đäCX, PźYž, ž, źşTę, |JGş. TGF-ŔVOijQŤđLˇéVR¨gvgyv`AĚWIŞqTő¤. ć5ńHiňwV|WE. s, 11, 2013.@[DG\ÜđóÜ] |
| 17) | Kakeya, H. Natural Products-Initiated Chemical Biology; Screening, Discovery, and Target Identification. 13th International Conference on the Chemistry and other bioactive compounds (ICCA-13), Yamanashi, Sep. 2013. (Invited Lecture) |
| 16) | R´î, źşTę, źXMž, PźYž, ž, şcšY, |JGş. CmRúüŰŞśYˇéheronamideŢĚPŁĆś¨Ť. ć55ńVRL@ť¨˘_ď. s, 9, 2013. |
| 15) | ĄěăÄ, Îěśm, |JGş. Afj[VhCđWIĆľ˝őeaŤv[uĚJ. ć7ńoCIÖAťwV|WE. ¤m, 9, 2013. |
| 14) | {×N, Îěśm, {{á, Icëj, ĄěăÄ, |JGş. AndrimidĚśŹyfĚ@\đÍ. ć7ńoCIÖAťwV|WE. ¤m, 9, 2013. |
| 13) | Nishimura, S., Tokukura, M., Ochi, J., Yoshida, M., Kakeya, H. Sterol-rich membrane domains and the balance of membrane traffic. Pombe 2013 (7th International fission yeast meeting), June, London, UK, 2013. |
| 12) | {{á, Îěśm, Ń@L, |JGş. óŰNeosartorya sp. Rvjî]ÚyfĚ@\đÍ. ú{P~JoCIW[wďEć8ńNď. , 6, 2013. |
| 11) | Îěśm, |JGş. AdenylationhCđWIĆľ˝eaŤv[uĚJ. ú{P~JoCIW[wďEć8ńNď. , 6, 2013. |
| 10) | Îěśm, |JGş. LC-MS/MSđp˘˝áŞqv[uÉΡéWI^pNżĚŻč. ć13ńú{`żČwď. šć, 6, 2013. |
| 9) | ÉĄş, |JGş, gcŤ. ESUMOťyfSENP1jQÜĚTő. ć17ńú{ŞńŞqWIĄĂwďEwpWď. s, 6, 2013. |
| 8) | gş@Ę, źşTę, ž, |JGş. á_fUąöq(HIF)ŤťoHđjQˇéúüŰRverucopeptinĚâΧĚzuĚč. ć17ńú{ŞńŞqWIĄĂwďEwpWď. s, 6, 2013. |
| 7) | ëěžF, źşTę, |JGş. A~m_ăÓđϲˇéVRť¨ĚTő¤. ć17ńú{ŞńŞqWIĄĂwďEwpWď. s, 6, 2013. |
| 6) | {{á, Îěśm, Ń@L, |JGş. Şq@\ϡđwüľ˝ óŰNeosartorya sp. Rvjî]ÚyfĚ@\đÍ. ú{ňwďć133Nď. _Ţě, 3, 2013. |
| 5) | Îěśm, |JGş. LpśŹyfĚŻčE@\đÍđwüľ˝ťwc[ĚJ\AdenylationhCđWIĆľ˝eaŤv[uĚJ\. ú{ňwďć133Nď. _Ţě, 3, 2013. |
| 4) | R´î, źşTę, PźYž, ž, |JGş. VK|G}NN^ĚPŁE\˘čƝ̜¨Ť. ú{ňwďć133Nď. _Ţě, 3, 2013. |
| 3) | gş@Ę, źşTę, Ý{^Ą, ž, |JGş. 1,3-dimethyl˝ó\˘Ě§Ězuč@ĚŘFtumescenamide CĆverucopeptinđáÉ. ú{ňwďć133Nď. _Ţě, 3, 2013. |
| 2) | pŃÔ, ž, ÂŘL, ŹŃSq, Xgpq, |JGş. ErL`ťyf(USP)47ĚŤť@\ĚđÍ. ú{ňwďć133Nď. _Ţě, 3, 2013. |
| 1) | X{Bç, ťězę, â×j, ˝ěG, ŔŘër, nçłYę, yäC, éŘ´ü, RŕÝäŤ, ĄníL, ĺËěF, ŕ_cFq, Ąňú, ěSi, sjŞ, {MĽ, |JGş, ac[š, ˇJě_ń. 4ťÜłě×tNXI[o[2dÓąÉćčAZN~zůżĚ˘zűřŚŞŔŘłę˝. ú{ňwďć133Nď. _Ţě, 3, 2013. |
| 20) | pŃÔ, ž, ÂŘL, ŹŃSq, Xgpq, |JGş. ErL`ťyf(USP)47ĚŤťÉ¨ŻéŞqŕrL`lhCĚđ. ć85ńú{śťwď. 12, Ş, 2012. |
|---|---|
| 19) | ž, źě˘q, pŃÔ, ŹŃSq, Xgpq, |JGş. ErL`ťyfUCH-L3Í_ťXgXĚWI^pNżĹ é. ć85ńú{śťwď. 12, Ş, 2012. |
| 18) | |JGş. ľŇuFVR¨ťwđîŐĆľ˝nňP~JoCIW[. áč¤ŇĚ˝ßĚL@ťwDyZ~i[. 11, kCš, 2012. |
| 17) | đäCX, źşTę, ž, žcń¤, yëv, ŞşĎ, |JGş. 3Ŕ-Hydroxysteroid dehydrogenase (3Ŕ-HSD) jQÜĚJ¤. ć30ńfBViP~Xg[V|WE. 11, , 2012. |
| 16) | Kanou, A., Nishimura, S., Kakeya, H. Chemical genetics for dissecting the crosstalk between cell metabolism and cell morphology. The 1st International Symposium on Chemical Biology of Natural Products: Target ID and Regulation of Bioactivity. Kyoto, Oct., 2012. |
| 15) | gşĘ, ĺËŃD, źşTę, ž, |JGş. á_fUąöq(HIF)ŤťoHđjQˇéverucopeptinÉÖˇé¤. ć19ńVRň¨ĚJĆpV|WE. 10, ĺă, 2012. |
| 14) | Jű˘}, đäCX, źşTę, ž, |JGş. GBF1jQŤđLˇégolgicide A Ě\˘ŤÖ¤. ć62ńú{ňwďßExďEĺď, 10, şÉ, 2012.[DG|X^[\ÜđóÜ] |
| 13) | gşĘ, ĺËŃD, źşTę, ž, ˇcTV, |JGş. á_fUąöq(HIF)ŤťoHđjQˇéverucopeptinĚťwIđͤ. ć54ńVRL@ť¨˘_ď. 10, , 2012. |
| 12) | ÓĹ, ž, |JGş. á_fUąöq(HIF)jQÜTőĚ˝ßĚnCRecEXN[jOnĚ\z. ć16ńú{ŞńŞqWIĄĂwďEwpWď. Ş, 6, 2012. |
| 11) | R´î, źşTę, X[óq, öGN, |JGş. úüŰĚĄ|{ÉćÁÄžçęéVKegqhLmUąĚÉÖˇé¤. ú{P~JoCIW[wď ć7ńNď. 6, s, 2012. |
| 10) | ž, źě˘q, pŃÔ, ŹŃSq, Xgpq, |JGş. Activity-based ProfillingÉćé_ťXgX´óŤErL`ťyfĚŻč. ú{P~JoCIW[wď ć7ńNď. 6, s, 2012. |
| 9) | Hu, X.-T., Hattori, A., Tokiwa, R., Kakeya, H. A high content screening system to develop novel HIF-1 inhibitors disrupting its heterodimeric formation. Organization for Oncology and Translational Research (OOTR) 8th Annual Meeting, Kyoto, Japan, Apr. 2012.[DG|X^[\ÜđóÜ] |
| 8) | Piao, J.-H., Tashiro, A., Nishikawa, M., Moriyoshi, E., Hattori, A., Kakeya, H. Enzymatic properties of recombinant human ubiquitin specific protease 47. Organization for Oncology and Translational Research (OOTR) 8th Annual Meeting, Kyoto, Japan, Apr. 2012. |
| 7) | }äşž, đäCX, PźYž, ž, ĺÎ^ç, ĄäMF, źşTę, |JGş. VKTGF-ŔVOi`BjQÜtryptopeptin A¨ćŃŞqv[uĚŹ¤. ú{ňwďć132Nď. Dy, 3, 2012. |
| 6) | R´î, źşTę, X[óq, öGN, |JGş. úüŰŞśYˇéVKegqhLmUąĚĚPŁE\˘đÍ. ú{ňwďć132Nď. Dy, 3, 2012. |
| 5) | ÓĹ, ž, íŐç, |JGş. ńŞquőâVXeđpľ˝á_fUąöq(HIF)jQÜŤ]żnĚ\z. ú{ňwďć132Nď. Dy, 3, 2012. |
| 4) | źě˘q, ŹŃSq, pŃÔ, Xgpq, ž, |JGş. ErL`ťyfUCH-L3Í_ťXgXşĹsŤťłęé. ú{ňwďć132Nď. Dy, 3, 2012. |
| 3) | pŃÔ, căß, źě˘q, Xgpq, ž, |JGş. qgUSP47ĚErL`ťyfŤĚđÍ. ú{ňwďć132Nď. Dy, 3, 2012 |
| 2) | źşTę, |JGş. V|WEuVR¨ťwĚVľ˘ŞŹvFśĚđđ͡éťwâ`w. ú{ňwďć132Nď. Dy, 3, 2012. iľŇuj |
| 1) | |JGş. V|WEuHi@\wĆňwFÚ_Ćá_ŠçwÔĚAv[`FhŕĚĆčhEhŕĚĂčhđîŐĆľ˝P~JoCIW[¤. ú{_|ťwď2011Nxĺď. s, 3, 2012. iľŇuj |
| 15) | |JGş. nňP~JoCIW[FŠRÉwÔhňhĂč. ČwEZptFX^ in s. s, 12, 2011. |
|---|---|
| 14) | Morimoto, T., Wada, H., Sunagawa, Y., Fujita, M., Kakeya, H., Sasaki, H., Imaizumi, A., Hashimoto, T., Akao, M., Osakada, G., Kambara, H., Doi, O., Shiomi, H., Kimura, T., Shimatsu, A., Hasegawa, K., Effects of highly absorptive curcumin on systolic and diastolic function in hypertensive patients with left ventricular hypertrophy. Heart failure: Pharmacologic Therapy in Advanced Preclinical and Clinical Trials. American Association Scientific Sessions 2011. Orland, FL, USA, Nov. 2011. |
| 13) | Hattori, A., Tashiro, A., Piao, J.-H., Moriyoshi, E., Kakeya, H. Characterization of enzymatic properties of recombinant human specific protease 47. 7th General Meeting of the International Proteolysis Society. San Diedo, CA, USA, Oct. 2011. |
| 12) | Ý{^Ą, PźYž, źşTę, ž, |JGş. úüŰŞYśˇéVKÂó|fvVyv`hpentadepsin AÉÖˇé¤. ć53ńVRL@ť¨˘_ď. ĺă. 9, 2011. |
| 11) | Espiritu, R.A., Matsumori, N., Murata, M., Nishimura, S., Kakeya, H., Matsunaga, S., Yoshida, M. Interaction of the marine sponge cyclic peptide theonellamide A with lipid bilayers investigated by membrane-permeabilizing activities and solid state 2H NMR. 14th Asian Chemical Congress 2011. Bangkok, Thailand, Sep. 2011. |
| 10) | zqq, źşTę, |JGş. ŞôyęɨŻé×EXe[ĚÇݧäĚđÍ. yęâ`wtH[Eć44ń¤ńď. Ş, 9, 2011. |
| 9) | ĺěTi, ž, ăcłš, eRi, gMB°, |JGş. qgC7orf24Ěâ`qťÍA]ĘJn_ßTĚ3ĚCCAATzńɧäłęé. ć84ńú{śťwď. s, 9, 2011. |
| 8) | ž, pŃÔ, căß, Xgpq, |JGş. OUCBđ|[^[Ép˘˝ErL`ťyfŤŞč@Ě\z. ć84ńú{śťwď. s, 9, 2011. |
| 7) | i{C÷, ž, |JGş, |{Ŕi, {´˝, Ü đĹĚAą˝đpľ˝pHËśŤVKDNAALťÜĚÝv. ć9ń˘ăđS¤L@ťwV|WE. , 5, 2011. |
| 6) | Ý{^Ą, PźYž, źşTę, ž, |JGş. ÷ś¨^{[đÍÉćčŠoľ˝VKÂó|fvVyv`h. ú{ňwďć131Nď. ĂŞ, 3, 2011. |
| 5) | ˝, ž, PźYž, źşTę, Żi, ŃYńY, ˇcTV, |JGş. ÇVśjQÜazaspireneĚěp@đÍĆWI^pNżTő. ú{ňwďć131Nď. ĂŞ, 3, 2011. |
| 4) | ž, căß, Xgpq, pŃÔ, |JGş. ErL`ťyfŤĚVľ˘Şč@Ěm§. ú{ňwďć131Nď. ĂŞ, 3, 2011. |
| 3) | PźYž, ž, ĺÎ^ç, ĄäMF, źşTę, |JGş. úüŰĚśYˇéVKRŞńÜ[hť¨tryptopeptinĚťw\˘č. ú{ňwďć131Nď. ĂŞ, 3, 2011. |
| 2) | |JGş. ÁĘV|WEVR¨ťwĆP~JoCIW[uVKś¨ŤVRL@ŞqĚJńĆP~JoCIW[¤v. ú{ňwďć131Nď. ĂŞ, 3, 2011.iľŇuj |
| 1) | |JGş. á_fUąöq(HIF)Ě@\§ä¨żĚTőE]ż. ŞńxŽuťwĂ@îŐxŽv-AJf~AŠçĚRŞńÜnňÖüŻÄ-. s, 3, 2011. |
| 12) | Tsunematsu, Y., Oishi, S., Fujii, N., Nishimura, S., Hattori, A., Kakeya, H. Tryptopeptin A, a novel TGF-beta signaling inhibitor from Streptomyces sp. International Chemical Congress of Pacific Basin Societies 2010 (PACIFICHEM 2010). Hawaii, USA, Dec., 2010. |
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| 11) | Nishimura, S., Matsunaga, S., Kakeya, H., Yoshida, M. Mode of action of theonellamides, antifungal bicyclic peptides from a marine sponge. International Chemical Congress of Pacific Basin Societies 2010 (PACIFICHEM 2010). Hawaii, USA, Dec., 2010. |
| 10) | căß, ž, pŃÔ, Rc¤, ĺÎ^ç, ĄäMF, |JGş. qgErL`ťyfUSP47ĚyfwIŤóđÍ. 83ńú{śťwďĺďEć33ńú{Şqś¨wďNďŻĺď: Biochemistry and Molecular Biology 2010 (BMB2010). 12, _Ë, 2010. |
| 9) | ĺěTi, ž, ăcłš, eRi, gMB°, |JGş. C7orf24/GGCTĚ]ĘÍNF-YÉć荝łęé. ć83ńú{śťwďĺďEć33ńú{Şqś¨wďNďŻĺď: Biochemistry and Molecular Biology 2010 (BMB2010). 12, _Ë, 2010. |
| 8) | źşTę, zqq, LcSq, źRWv, źiÎ÷, gcŤ, |JGş. CYR^ۨżtheonellamideĚěp@đž. ć60ńú{ňwďßExďEĺď. 10, ĺă, 2010. |
| 7) | PźYž, ĺÎ^ç, ĄäMF, źşTę, ž, |JGş. úüŰŞśYˇéVKTGF-ŔVOi`BjQÜĚPŁE\˘đÍĆŹ. ćTQńVRL@ť¨˘_ď. 9, ĂŞ, 2010. [§ăÜđóÜ] |
| 6) | Ń@L, şńN, ĺuN, ł˝, ˇcTV, |JGş. VKÇVśjQ¨żĚśŹâ`qQĚN[jO. 2010Nxić25ńjú{úüŰwďĺď. 9, , 2010. |
| 5) | ĺγ, {Nž, ¨Đł}, ´ jY, ˇcTV, ž, |JGş. VKá_fUąöq(HIF)jQÜĚnť¤. ć1Sńú{ŞńŞqWIĄĂwďEwpWď. 7, , 2010. |
| 4) | {Nž, ¨Đł}, ž, |JGş. VKscaffoldđLˇéTGF-ŔVOi`BŐfňĚnť¤. ć1Sńú{ŞńŞqWIĄĂwďEwpWď. 7, , 2010. |
| 3) | źşTę, zqq, LcSq, źRWv, źiÎ÷, gcŤ, |JGş. Xe[đWIơétheonellamideĚěp@đÍ. ú{P~JoCIW[wď ć5ńNď. 5, _Ţě, 2010. |
| 2) | Ohno, Y., Hattori, A., Ueda, M., Kageyama, S., Yoshiki, T., Kakeya, H. Involvement of NF-Y in transcriptional regulation if the human C7orf24/GGCT gene. Organisation for Oncology and Translational Research (OOTR) 6th Annual Conference. Kyoto, Japan, Feb., 2010. [DG|X^[\ÜđóÜ] |
| 1) | {Nž, ž, |JGş.@VKĚžłĄĂňĚJ¤FhHit to ProbehĚíŞĆŔŘ. uTGF-ŔŤť˝đWIĆľ˝ĚžłĚVKff@, ĄĂE\h@ĚJv¤ÇV|WE. 2, ĺă, 2010. |
| 7) | ÁĄź÷, ŘC, |JGş, ˇcTV. Aspergillus fumigatusɨŻépseurotinśŹâ`qNX^[ĚđÍ. ć9ń óŰŞqś¨wRt@X. , 11, 2009. |
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| 6) | Nishimura, S., Matsuyama, A.., Yoshida, M., Matsunaga, S., Kakeya, H. Regulation of sterol localization revealed by chemical genetics using theonellamide. The 5th International Fission Meeting. Tokyo, Oct. 2009. |
| 5) | |JGş. V|WEuQmňwĆnňvFP~JoCIW[¤đîŐĆľ˝AJf~AɨŻénň¤. ć68ńú{ŕwďwpď. Ąl, 10, 2009iľŇuj. |
| 4) | źşTę, źRWv, źiÎ÷, |JGş, gcŤ. Xe[đWIơétheonellamideŢŞUąˇéŞôyęĚ`ÔŮí. yęâ`wtH[ć42ń¤ńď. }g, 7, 2009. |
| 3) | ĺěTi, ž, |JGş. VKŕÖAöqqgC7orf24Ě]ʧä@\ĚđÍ. ć13ńú{ŕŞqWIĄĂwď. ż, 6, 2009. |
| 2) | ž, PźYž, ĺËŃD, {Nž, źşTę, îqO, ĺÎ^ç, ĄäMF, ´ jY, ˇcTV, |JGş. HIF-1@\§äť¨Ě]żn\zĆTő¤. ú{ňwďć129Nď. s, 3, 2009. |
| 1) | Kakeya, H. Natural products-initiated chemical biology. Organic Chemistry Seminar in University of Louis Pasteur. Strasbourg, France, Apr. 2009 (Invited Lecture). |
| 5) | |JGş. ÷ś¨šđîŐĆľ˝P~JoCIW[¤. ć17ńVRň¨ĚJĆpV|WE. V|WE1\u÷ś¨öÝ\ÍĚÄFŻ-nňĆîb¤ÖĚpv. ˝, 11, 2008.iľŇuj |
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| 4) | îqOA|JGşAÉĄüçäA{˝`ş. žĚCŹŞśŹÉÖ^ˇéeyŹyfâ`qĚđͤ. ć55ńú{śňwďNď. ˇč, 9, 2008. |
| 3) | ŃYńYAŻiAÎěElARűęYAcşFTAĄä_MAźJmăAŤęA|JGşAˇcTV. AT}CVnRîáVR¨ATCggGjAĚSŹ. ć50ńVRL@ť¨˘_ď. ˝, 9, 2008. |
| 2) | |JGş. "ŕĚĆč"đîŐĆľ˝P~JoCIW[¤. ć128ńú{ňwďV|WE VR¨p[FwŕĚĆčCŹC@\đžx`ĺwVR¨ňw¤`. Ąl, 3, 2008.iľŇuj |
| 1) | |JGş. nňV[YJđwüľ˝VKVRL@ť¨ĚJńEnťĆP~JoCIW[¤. \SEÇaĄĂĚlbTX\Ő°SÇÄś¤ď. s, 1, 2008.iľŇuj |
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