{"id":219,"date":"2025-04-25T13:12:58","date_gmt":"2025-04-25T04:12:58","guid":{"rendered":"https:\/\/www.pharm.kyoto-u.ac.jp\/souyaku?page_id=219"},"modified":"2026-04-24T11:43:01","modified_gmt":"2026-04-24T02:43:01","slug":"publication","status":"publish","type":"page","link":"https:\/\/www.pharm.kyoto-u.ac.jp\/souyaku\/?page_id=219","title":{"rendered":"Publication"},"content":{"rendered":"

[2026][2025<\/a>][2024<\/a>][2023<\/a>][2022<\/a>][2021<\/a>][2020<\/a>][2019<\/a>][2018<\/a>][2017<\/a>][2016<\/a>][2015<\/a>] [2014<\/a>] [2013\u4ee5\u524d<\/a>] <\/span><\/p>\n

2026<\/span><\/h4>\n
    \n
  1. \n
    Fujii, T.; Araki, M.; Matsumoto, S.; Ma, B.; Otsuka, T.; Bekker, G.-J.; Kamiya, N.; Ohno, H.; Inuki, S.; Okuno, Y.<\/span><\/div>\n
    Elucidating Ligand Charge Effects in MR1 Cell Surface Translocation Using Molecular Simulations.<\/span><\/div>\n
    J. Chem. Inf. Model.<\/em>\u00a02026<\/strong>,\u00a066<\/em>, 2211\u20132219.<\/span><\/div>\n
    DOI: 10.1021\/acs.jcim.5c02141<\/span><\/a><\/div>\n
    \"Abstract<\/pre>\n<\/li>\n
  2. \n
    Yamamoto, Y.; Takenaka, S.; Arichi, N.; Inuki, S.; Ohno, H.
    \nGold-Catalyzed Cyclization of Pyrrole-Tethered Allenynes for the Synthesis of 4-Acylindoles and Its Application to the Ergot Alkaloid Scaffold.\u00a0<\/span><\/div>\n
    Org. Lett<\/em>. 2026<\/strong>, 28<\/em>, 1331\u20131336.
    \n    DOI: 10.1021\/acs.orglett.5c05144<\/a> <\/span><\/span><\/div>\n
    \"Abstract\r\n<\/span><\/span><\/pre>\n<\/li>\n
  3. \n
    Shimamoto, N.; Arichi, N.; Ohno, H.<\/span><\/div>\n
    Triplet Nitrene-Mediated Photocatalytic Azidation of Tertiary C(sp3<\/sup>)\u2013H Bonds.<\/span><\/div>\n
    Chem. Commun.<\/em> 2026<\/strong>, 62<\/em>, 164\u2013167.<\/span><\/span><\/div>\n
    DOI: 10.1039\/D5CC05587C<\/span><\/a><\/div>\n
    \"\"<\/pre>\n<\/li>\n<\/ol>\n
    <\/a>2025<\/span><\/h4>\n
      \n
    1. \n
      Hasegawa, D.; Arichi, N.; Ohno, H.<\/span><\/div>\n
      Stereoselective Synthesis of Spirocyclic Indolin-3-ones through a Gold(I)-Catalyzed Cascade Cyclization of Azido-alkynes.
      \nJ<\/em>. Org<\/em>. Chem<\/em>. 2025<\/strong>, 90<\/em>, 11737\u201311741.
      \n      DOI: 10.1021\/acs.joc.5c01284<\/a><\/span><\/span><\/div>\n
      \"Abstract<\/span><\/pre>\n<\/li>\n
    2. \n
    3. \n
      Iwamoto, N.; Ohno, S.; Nakamura, K.; Naito, T.; Miura, S.; Inuki, S.; Ohno, H.; Hayashi, G.; Murakami, H.; Oishi, S.
      \nDesign and Evaluation of Stable Cysteine-Modified Monobody Scaffolds for Mirror-Image Synthesis.
      \nBioconjug. Chem.<\/em>\u00a02025<\/strong>,\u00a036<\/em>, 1504\u20131515.
      \n      DOI: 10.1021\/acs.bioconjchem.5c00181<\/a><\/span><\/span><\/div>\n
      \"Abstract\r\n<\/span><\/pre>\n<\/li>\n
    4. \n
      Ohno, H.; Tsuji, A.; Hasegawa, D.; Inuki, S.; Arichi, N.<\/span>
      \nSynthetic Study of Caulerpin: Construction of the Core Structure through Gold-Catalyzed Cascade Cyclization of Azido-Alkynes.
      \n<\/b>Chem<\/em>. Pharm<\/em>. Bull<\/em>. 2025<\/strong>, 73<\/em>, 645\u2013649.
      \n      DOI: 10.1248\/cpb.c25-00268<\/a><\/span>
      \n<\/span><\/span><\/span><\/p>\n
      \"\"\r\n<\/span><\/pre>\n<\/div>\n<\/li>\n
    5. \n
      Takahara, A.; Nakatsu, T.; Hirata, K.; Hayashi, H.; Kawaji, K.; Aoki, K.; Inuki, S.; Ohno, H.; Kato, H.; Kodama, E.; Oishi, S.
      \nElucidation of Postfusion Structures of the Measles Virus F Protein for the Structure-Based Design of Fusion Inhibitors.
      \nJ. Med. Chem.<\/em> 2025<\/strong>,\u00a068<\/em>, 3123\u20133133.
      \n      DOI: 10.1021\/acs.jmedchem.4c02337<\/span><\/a><\/span>
      \n<\/span><\/span><\/div>\n
      \"\"<\/span><\/pre>\n<\/li>\n
    6. \n
    7. \n
    8. \n
    9. \n
    10. \n
    11. \n
      Hasegawa, D.; Tsuji, A.; Greiner, L. C.; Arichi, N.; Inuki, S.; Ohno, H.
      \n<\/span><\/div>\n
      Synthesis of Azocine-Fused Indoles via Gold(I)-Catalyzed Cyclization of Azido-alkynes.
      \n<\/span><\/div>\n
      J. Org. Chem.<\/em> 2025<\/strong>, 90<\/em>, 925\u2013930.
      \n      DOI: 10.1021\/acs.joc.4c02704<\/a><\/span><\/span><\/div>\n
      \"\"<\/span><\/pre>\n<\/li>\n
    12. \n
      Matsuoka, T.; Takasaki, R.; Akiba, H.; Ogata, K.; Hattori, A.; Arichi, N.; Kakeya, H.; Yamasaki, S.; Ishihama, Y.; Ohno, H.; Inuki, S.
      \n<\/span><\/div>\n
      Visible light-mediated photocatalytic coupling between tetrazoles and carboxylic acids for biomolecule labelling.<\/span><\/div>\n
      Chem. Commun.<\/em> 2025<\/strong>, 61<\/em>, 6320\u20136323.
      \n<\/span>      DOI: 10.1039\/D4CC04452E<\/a> <\/span><\/span><\/div>\n
      \"\"<\/pre>\n<\/li>\n<\/ol>\n
      <\/a>2024<\/span><\/h4>\n
        \n
      1. \n
        Takasaki, R.; Ito, E.; Nagae, M.; Takahashi, Y.; Matsuoka, T.; Yasue, W.; Arichi, N.; Ohno, H.; Yamasaki, S.; Inuki, S.<\/span><\/div>\n
        Development of Ribityllumazine Analog as Mucosal-associated Invariant T Cell Ligand.<\/span><\/div>\n
        J. Am. Chem. Soc. <\/i>2024<\/strong>, 146<\/em>, 29964\u201329976.
        \n        DOI: 10.1021\/jacs.4c12997<\/a><\/span><\/span><\/div>\n
        \"\"<\/span><\/pre>\n<\/li>\n
      2. \n
        Nakamura, S.; Nishiwaki, K.; Tsuyuguchi, M.; Kinoshita, T.; Oishi, S.; Ohni. H.; Nakanishi, I.
        \n<\/span><\/div>\n
        Compounds Designs of CK2\u03b1 Inhibitors Derived from Virtual Screening Hit Compounds by Computational Chemistry with Crystallography.
        \n<\/span><\/div>\n
        Chem. Pharm. Bull.<\/em> 2024<\/strong>, 72<\/em>, 776\u2013780.
        \n<\/span><\/div>\n
        DOI: 10.1248\/cpb.c23-00824<\/a><\/span><\/div>\n
        \"\"\r\n<\/span><\/pre>\n<\/li>\n
      3. \n
        Aoki, K.; Maeda, K.; Inuki, S.; Ohno, H.; Nonaka, M.; Oishi, S.
        \nChemical Synthesis of Interleukin-6 for Mirror-Image Screening.
        \nBioconjug. Chem.<\/em>\u00a02024<\/strong>,\u00a035<\/em>, 1190\u20131199.
        \n        DOI: doi\/10.1021\/acs.bioconjchem.4c00204<\/span><\/a><\/span><\/span><\/div>\n
        \"\"<\/span><\/pre>\n<\/li>\n
      4. \n
        Hashimoto, N.; Taguchi, J.; Kasagi, T.; Arichi, N.; Inuki, S.; Ohno, H.
        \nConstruction of the Akuammiline Alkaloid Core Structure via Stereoselective E-ring Formation.
        \nJ. Org. Chem. <\/i>2024<\/strong>, 89<\/em>, 10388\u201310392.<\/span><\/div>\n
        DOI: 10.1021\/acs.joc.4c01105<\/a><\/span><\/div>\n
        \"\"\r\n<\/span><\/pre>\n<\/li>\n
      5. \n
        Arichi, N.; Amano, T.; Wu, S.; Inuki, S.; Ohno, H.
        \nSynthesis of Sulfilimines via Visible-Light-Mediated Triplet Energy Transfer to Sulfonyl Azides.
        \nChem. Eur. J. <\/i>2024<\/strong>, 30<\/em>, e202401842.
        \n        DOI: 10.1002\/chem.202401842<\/a> <\/span><\/span><\/div>\n
        \"\"<\/span><\/pre>\n<\/li>\n
      6. \n
        Iwamoto, N.; Kai, T.; Inuki, S.; Ohno, H.; Maeda, H.; Watanabe, H.; Maruyama, T.; Oishi, S.
        \nMirror-Image Human Serum Albumin Domain III as a Tool for Analyzing Site II-Dependent Molecular Recognition.
        \nBioconjug. Chem<\/em>.\u00a02024<\/strong>,\u00a035<\/em>, 816\u2013825. 
        \n        DOI: 10.1021\/acs.bioconjchem.4c00150<\/span><\/a>
        \n<\/span><\/span><\/div>\n
         \"\"<\/span><\/pre>\n<\/li>\n
      7. \n
      8. \n
      9. \n
        Inuki, S.; Miyamoto, J.; Hashimoto, N.; Shimizu, H.; Tabuchi, H.; Kawai, A.; Greiner, L. C.; Kimura, I.; Ohno, H.
        \n<\/span><\/div>\n
        Structure-Activity Relationship Studies of Tetrahydroquinolone Derivatives as GPR41 Modulators.
        \nBioorg. Med. Chem. Lett. <\/em>2024<\/strong>, 107<\/em>, 129758.
        \n        DOI: 10.1016\/j.bmcl.2024.129758<\/a><\/span>
        \n<\/span><\/span><\/div>\n
        \"\"<\/span><\/pre>\n<\/li>\n
      10. \n
        Aoki, K.; Tsuda, S.; Ogata, N.; Kataoka, M.; Sasaki, J.; Inuki, S.; Ohno, H.; Watashi, K.; Yoshiya, T.; Oishi, S.
        \nSynthetic Study of Full-length Hepatitis B Virus Core Protein and Its Capsid Formation.
        \nOrg. Biomol. Chem. <\/i>2024<\/strong>, 22<\/em>, 2218\u20132225.
        \n        DOI: doi.org\/10.1039\/D3OB02099A<\/a> <\/span><\/span><\/div>\n
        \"\"<\/span><\/pre>\n<\/li>\n
      11. \n
        Yamaguchi, A.; Obiya, N.; Arichi, N.; Oishi, S.; Ohno, H.; Inuki, S.
        \nSynthesis of Labionin and Avionin Precursors via Nitrogen-centred-radical-triggered 1,5-HAT Reaction of Tris Derivatives.
        \nOrg. Biomol. Chem. <\/i>2024<\/strong>, 22<\/em>, 2049\u20132055.
        \n        DOI: 10.1039\/D3OB02037A<\/a><\/span>
        \n<\/span><\/span><\/div>\n
        \"\"<\/span><\/pre>\n<\/li>\n
      12. \n
        Iwamoto, N.; Sakaki, J.; Ohno, S.; Aoki, K.; Usui, Y.; Inuki, S.; Ohno, H.; Oishi, S.
        \nSynthetic Studies on the Extracellular Domain of the T Cell Immunoreceptor with Immunoglobulin and Immunoreceptor Tyrosine-Based Inhibitory Motif Domain (TIGIT) Using Trt-K10 Solubilizing Tags.
        \nBioorg. Med. Chem. <\/i>2024<\/strong>, 99<\/em>, 117585.
        \n        DOI: 10.1016\/j.bmc.2023.117585<\/a><\/span><\/span><\/div>\n
        \"\"<\/span><\/pre>\n<\/li>\n
      13. \n
      14. \n
        Ohno, H.;\u00a0Arichi, N.; Inuki, S.<\/span><\/div>\n
        Nonbiomimetic Total Synthesis of Polycyclic Alkaloids.<\/span><\/div>\n
        Modern Natural Product Synthesis: Overcoming Difficulties<\/i>, 1st ed; Springer, 2024<\/strong>.<\/span><\/div>\n<\/li>\n<\/ol>\n
        <\/a>2023<\/span><\/h4>\n
          \n
        1. \n
        2. \n
          Hashimoto, N.; Taguchi, J.; Arichi, N.; Inuki, S.; Ohno, H.
          \nGold(I)-Catalyzed Cascade Cyclization of Alkynyl Indoles for the Stereoselective Construction of the Quaternary Carbon Center of Akuammiline Alkaloids.
          \nJ. Org. Chem. <\/i>2023<\/strong>, 88<\/em>, 17306\u201317321.
          \n          DOI: 10.1021\/acs.joc.3c02142<\/span><\/span><\/a>
          \n<\/span><\/div>\n
          \"\"<\/pre>\n<\/li>\n
        3. \n
          Aoki, K.; Manabe, A.; Kimura, H.; Katoh, Y.; Inuki, S.; Ohno, H.; Nonaka, M.; Oishi, S.
          \n<\/span><\/div>\n
          Mirror-Image Single-Domain Antibody for a Novel Nonimmunogenic Drug Scaffold.
          \nBioconjug.<\/i> Chem<\/em>. 2023<\/strong>, 34<\/em>, 2055\u20132065.
          \n          DOI: <\/a>10.1021\/acs.bioconjchem.3c00372<\/a> <\/span><\/span><\/div>\n
          \"\"\r\n<\/span><\/pre>\n<\/li>\n
        4. \n
          Iwamoto, N.; Sato, Y.; Manabe, A.; Inuki, S.; Ohno, H.; Nonaka, M.; Oishi, S.
          \nDesign and Synthesis of Monobody Variants with Low Immunogenicity.
          \nACS Med. Chem. Lett.<\/i> 2023<\/strong>, 14<\/em>, 1596\u20131601.
          \n          DOI: 10.1021\/acsmedchemlett.3c00342<\/a><\/span><\/span><\/div>\n
          \"\"<\/pre>\n<\/li>\n
        5. \n
          Matsuoka, T.; Hattori, A.; Oishi, S.; Araki, M.; Ma, B.; Fujii, T.; Arichi, N.; Okuno, Y.; Kakeya, H.; Yamasaki, S.; Ohno, H.; Inuki, S.
          \nEstablishment of an MR1-Presentation Reporter Screening System and Identification of Phenylpropanoid Derivatives as MR1 Ligands.
          \nJ. Med. Chem. <\/i>2023<\/strong>, 66<\/em>, 12520\u201312535.
          \n          DOI: 10.1021\/acs.jmedchem.3c01122 <\/a><\/span><\/span><\/div>\n
          \"\"<\/span><\/pre>\n<\/li>\n
        6. \n
          Oka, S.; Watanabe, M.; Ito, E.; Takeyama, A.; Matsuoka, T.; Takahashi, M.; Izumi, Y.; Arichi, N.; Ohno, H.; Yamasaki, S.; Inuki, S.
          \nArchaeal Glycerolipids Are Recognized by C-type Lectin Receptor Mincle.
          \nJ. Am. Chem. Soc.<\/i>\u00a02023<\/strong>, 145<\/em>, 18538\u201318548.
          \n          DOI: 10.1021\/jacs.3c05473<\/a><\/span><\/span><\/div>\n
          \"\"\r\n<\/span><\/pre>\n<\/li>\n
        7. \n
          Suzuki, R.; Mattos, D. R.; Kitamura, T.; Tsujioka, R.; Kobayashi, K.; Inuki, S.; Ohno, H.; Ishmael, J. E.; McPhail, K. L.; Oishi, S.
          \nDesign of Synthetic Surrogates for the Macrolactone Linker Motif in Coibamide A.
          \n<\/span><\/div>\n
          ACS Med. Chem. Lett.<\/i> 2023<\/strong>, 14<\/em>, 1344\u20131350.
          \n<\/span><\/div>\n
          DOI: 10.1021\/acsmedchemlett.3c00232<\/a> <\/span><\/div>\n
          \"\"<\/span><\/pre>\n<\/li>\n
        8. \n
          Tsuno, H.; Shen, J.; Komatsu, H.; Arichi, N.; Inuki, S.; Ohno, H.
          \n<\/span><\/div>\n
          Gold(I)\u2010Catalyzed Bis\u2010Cyclization of Allenynes for the Synthesis of Strained and Planar Polycyclic Compounds.
          \n<\/span><\/div>\n
          Angew. Chem. Int. Ed.<\/i> 2023<\/strong>, 62<\/em>, e202307532.
          \n          DOI: 10.1002\/anie.202307532<\/a><\/span>
          \n<\/span><\/div>\n
          \"\"<\/span><\/pre>\n<\/li>\n
        9. \n
          Yoshida, Y.; Takeuchi, H.; Nakagawa, K.; Fujii, T.; Arichi, N.; Oishi, S.; Ohno, H.; Inuki, S.
          \nConstruction of a Bicyclo[2.2.2]octene Skeleton via a Visible-Light-Mediated Radical Cascade Reaction of Amino Acid Derivatives with N-(2-Phenyl)benzoyl Groups.<\/span><\/div>\n
          Org. Lett.<\/i>\u00a02023<\/strong>, 25<\/em>, 4846\u20134851.
          \n          DOI: 10.1021\/acs.orglett.3c01586<\/a><\/span><\/span><\/div>\n
          \"\"<\/span><\/pre>\n<\/li>\n
        10. \n
          Nishiyama, K.; Akiba, H.; Nagata, S.; Tsumoto, K.; Kamada, H.; Ohno, H.
          \nA Proximity-Induced Fluorogenic Reaction Triggered by Antibody\u2013Antigen Interactions with Adjacent Epitopes.<\/span><\/div>\n
          Angew. Chem. Int. Ed.<\/i> 2023<\/strong>, 62<\/em>, e202306431.
          \n          DOI: 10.1002\/anie.202306431<\/a><\/span><\/span><\/div>\n
          \"\"\r\n<\/span><\/pre>\n<\/li>\n
        11. \n
        12. \n
          Tsuji, A.; Masuya, T.; Arichi, N.; Inuki, S.; Murai, M.; Miyoshi, H.; Ohno, H.
          \n<\/span><\/div>\n
          Discovery of Bis-sulfonamides as Novel Inhibitors of Mitochondrial NADH-Quinone Oxidoreductase (Complex I).
          \n<\/span><\/div>\n
          ACS Med. Chem. Lett.<\/i> 2023<\/strong>, 14<\/em>, 211\u2013216.
          \n          DOI: 10.1021\/acsmedchemlett.2c00504<\/a><\/span><\/span><\/div>\n
          \"\"<\/span><\/pre>\n<\/li>\n
        13. \n
          Greiner, L. C.; Arichi, N.; Inuki, S.; Ohno, H.
          \nGold(I)-Catalyzed Benzylic C(sp3)-H Functionalizations: Divergent Synthesis of Indole[a]- and [b]-Fused Polycycles.<\/span><\/div>\n
          Angew. Chem. Int. Ed.<\/i> 2023<\/strong>, 62<\/em>, e202213653.
          \n          DOI: 10.1002\/anie.202213653<\/a><\/span><\/span><\/div>\n
          \"\"\r\n<\/span><\/span><\/pre>\n<\/li>\n
        14. \n
          Miyamoto, J; Shimizu, H.; Hisa, K.; Matsuzaki, C.; Inuki, S.; Ando, Y.; Nishida, A.; Izumi, A.; Yamano, M.; Ushiroda, C.; Irie, J.; Katayama, T.; Ohno, H.; Itoh, H.; Yamamoto, K.; Kimura, I.
          \nHost metabolic benefits of prebiotic exopolysaccharides produced by Leuconostoc mesenteroides<\/em>.
          \nGut Microbes\u00a0<\/i>2023<\/strong>, 15<\/em>, 2161271.
          \n          DOI: <\/span>10.1080\/19490976.2022.2161271<\/span><\/span><\/a><\/span><\/div>\n<\/li>\n<\/ol>\n
          <\/a>2022<\/span><\/h4>\n
            \n
          1. \n
          2. \n
          3. \n
          4. \n
            Kitamura, T.; Suzuki, R.; Inuki, S.; Ohno, H.; McPhail, K. L.; Oishi, S.
            \nDesign of coibamide A mimetics with improved cellular bioactivity.
            \n<\/span><\/div>\n
            ACS Med. Chem. Lett.\u00a0<\/em>2022<\/strong>, 13<\/em>, 105\u2013110.
            \n            DOI: 10.1021\/acsmedchemlett.1c00591<\/span><\/a><\/span><\/span><\/div>\n
            \"\"<\/span><\/pre>\n<\/li>\n<\/ol>\n
            <\/a>2021<\/span><\/h4>\n
              \n
            1. \n
              Komatsu, H.; Ikeuchi, T.; Tsuno, H.; Arichi, N.; Yasui, K.; Oishi, S.; Inuki, S.; Fukazawa, A.; Ohno, H.
              \nConstruction of Tricyclic Nitrogen Heterocycles by Gold(I)-Catalyzed Cascade Cyclization of Allenynes and Its Application to Polycyclic \u03c0-Electron Systems.
              \nAngew. Chem. Int. Ed.\u00a0<\/em>2021<\/strong>, 60<\/em>, 27019\u201327025.
              \n<\/span><\/div>\n
              DOI: 10.1002\/anie.202111267<\/a><\/span><\/div>\n
              \"\"  <\/i><\/i><\/span><\/pre>\n<\/li>\n
            2. \n
              Greiner, L. C.; Inuki, S.; Arichi, N.; Oishi, S.; Suzuki, R.; Iwai, T.; Sawamura, M.; Hashmi, A. S. K.; Ohno, H.
              \nAccess to Indole-Fused Benzannulated Medium-Sized Rings through Gold(I)-Catalyzed Cascade Cyclization of Azido-Alkynes.
              \nChem. Eur. J.<\/em> 2021<\/strong>, 27<\/em>, 12992\u201312997.
              \n              DOI: 10.1002\/chem.202101824<\/a><\/span><\/span><\/div>\n
              \"\"<\/span><\/pre>\n<\/li>\n
            3. \n
              Matsuoka, T.; Motozono, C.; Hattori, A.; Hideaki, K.; Yamasaki, S.; Oishi, S.; Ohno H.; Inuki, S.
              \nThe Effects of 5\u2010OP\u2010RU Stereochemistry on Its Stability and MAIT\u2010MR1 Axis.
              \nChemBioChem.\u00a0<\/em>2021<\/strong>, 22<\/em>, 672\u2013678.
              \n              DOI: 10.1002\/cbic.202000466<\/a><\/span><\/span><\/div>\n
              \"\"<\/span><\/pre>\n<\/li>\n
            4. \n
              Yamaguchi, A.; Inuki, S.; Ohta, K.; Oishi, S.; Asai, A.; Ohno, H.
              \nIdentification of a Novel Indoleamine 2,3-Dioxygenase Inhibitor Bearing an Eight-Membered Ring Fused Indole Scaffold and Its Structure-Activity Relationship.
              \nHeterocycles<\/em> 2021<\/strong>, 103<\/em>, 331\u2013347.
              \n<\/span><\/div>\n<\/li>\n
            5. \n
            6. \n
              Ohno, H.; Inuki, S.<\/span><\/div>\n
              Nonbiomimetic total synthesis of indole alkaloids using alkyne-based strategies.<\/span><\/div>\n
              Org. Biomol.<\/i> Chem<\/em>. 2021<\/strong>, 19<\/em>, 3551\u20133568.
              \n              DOI: 10.1039\/D0OB02577A<\/a><\/span><\/span><\/div>\n
              \"\"<\/pre>\n<\/li>\n
            7. \n
            8. \n
              Arichi, N.; Ohno, H.<\/span><\/div>\n
              Natural Product Synthesis via Palladium-Catalyzed C\u2013H Bond Activation.<\/span><\/div>\n
              In Handbook of CH-Functionalization, Ed. by D. Maiti, Wiley-VCH,<\/i> Weinheim, 2021<\/strong>.<\/i><\/span><\/div>\n<\/li>\n<\/ol>\n
              <\/a>2020<\/span><\/h4>\n
                \n
              1. \n
                Takeuchi, H.; Inuki, S.; Nakagawa, K.; Kawabe, T.; Ichimura, A.; Oishi, S.; Ohno H.
                \nTotal Synthesis of Zephycarinatines via Photocatalytic Reductive Radical ipso-Cyclization.
                \nAngew. Chem. Int. Ed.\u00a0<\/em>2020<\/strong>, 59<\/em>, 21210\u201321215.
                \n                DOI: 10.1002\/anie.202009399<\/span><\/span><\/a><\/span><\/div>\n
                \"\"<\/span><\/pre>\n<\/li>\n
              2. \n
                Matsuoka, J.; Inuki, S.; Matsuda, Y.; Miyamoto, Y.; Otani, M.; Oka, M.; Oishi, S.; Ohno, H.
                \nTotal Synthesis of Dictyodendrins A\u2013F by the Gold-Catalyzed Cascade Cyclization of Conjugated Diyne with Pyrrole.
                \nChem. Eur. J.<\/em>\u00a02020<\/strong>, 26<\/em>, 11150\u201311157.
                \n                DOI: 10.1002\/chem.202001950<\/span><\/a><\/span><\/span><\/div>\n
                \"\"<\/span><\/pre>\n<\/li>\n
              3. \n
                Matsuoka, T.; Inuki, S.; Miyagawa, T.; Oishi, S.; Ohno, H.
                \nTotal Synthesis of (+)-Polyoxamic Acid via Visible-Light-Mediated Photocatalytic \u03b2-Scission and 1,5-Hydrogen Atom Transfer of Glucose Derivative.
                \nJ. Org. Chem<\/em>. 2020<\/strong>, 85<\/em>, 8271\u20138278.
                \n                DOI: 10.1021\/acs.joc.0c00910<\/a><\/span><\/span><\/div>\n
                \"\"<\/span><\/pre>\n<\/li>\n
              4. \n
                Kimura, I.; Miyamoto, J.; Ohue-Kitano, R.; Watanabe, K.; Yamada, T.; Onuki, M.; Aoki, R.; Isobe, Y.; Kashihara, D.; Inoue, D.; Inaba, A.; Takamura, Y.; Taira, S.; Kumaki, S.; Watanabe, M.; Ito, M.; Nakagawa, F.; Irie, J.; Kakuta, H.; Shinohara, M.; Iwatsuki, K.; Tsujimoto, G.; Ohno, H.; Arita, M.; Itoh, H.; Hase, K.
                \n<\/span><\/div>\n
                Maternal gut microbiota in pregnancy influences offspring metabolic phenotype in mice.
                \nScience<\/em> 2020<\/strong>,\u00a0367<\/em>, eaaw8429.
                \n                DOI: 10.1126\/science.aaw8429<\/a><\/span>
                \n<\/span><\/div>\n
                \r\n\"\"<\/span><\/pre>\n<\/li>\n
              5. \n
              6. \n
                Miller, S.; Son, Y. L.; Aikawa, Y.; Makino, E.; Nagai, Y.; Srivastava, A.; Oshima, T.; Sugiyama, A.; Hara, A.; Abe, K.; Hirata, K.; Oishi, S.; Hagihara, S.; Sato, A.; Tama, F.; Itami, K.; Kay, S. A.; Hatori, M.; Hirota, T.
                \nIsoform-selective regulation of mammalian cryptochromes.
                \nNat. Chem. Biol.<\/em> 2020<\/strong>,\u00a016<\/em>, 676\u2013685.
                \n                DOI: 10.1038\/s41589-020-0505-1<\/span><\/a><\/span>
                \n<\/span><\/div>\n
                \"\"<\/span><\/pre>\n<\/li>\n
              7. \n
                Yamaguchi, A.; Inuki, S.; Tokimizu, Y.; Oishi, S.; Ohno, H.
                \nGold(I)-Catalyzed Cascade Cyclization of Anilines with Diynes: Controllable Formation of Eight-Membered Ring-Fused Indoles and Propellane-Type Indolines.<\/span><\/div>\n
                J. Org. Chem.<\/em> 2020<\/strong>, 85<\/em>, 2543\u20132559.
                \n                DOI: 10.1021\/acs.joc.9b03256<\/span><\/a><\/span><\/span><\/div>\n
                \"\"<\/span><\/span><\/pre>\n<\/li>\n<\/ol>\n
                <\/a>2019<\/span><\/h4>\n
                  \n
                1. \n
                2. \n
                3. \n
                  Miyagawa, T.; Inuki, S.; Oishi, S.; Ohno, H.
                  \nConstruction of Quaternary Carbon Stereocenter of \u03b1-Tertiary Amine through Remote C\u2013H Functionalization of Tris Derivatives: Enantioselective Total Synthesis of Myriocin.
                  \nOrg. Lett.<\/em> 2019<\/strong>, 21<\/em>, 5458\u20135490.
                  \n                  DOI: 10.1021\/acs.orglett.9b01778<\/span><\/a><\/span><\/span><\/div>\n
                  \"\"<\/span><\/pre>\n<\/li>\n
                4. \n
                  Matsuoka, J.; Kumagai, H.; Inuki, S.; Oishi, S.; Ohno, H.
                  \nConstruction of the pyrrolo[2,3-d]carbazole core of spiroindoline alkaloids by gold-catalyzed cascade cyclization of ynamide.
                  \nJ. Org. Chem.<\/em> 2019<\/strong>,\u00a084<\/em>, 9358\u20139363.
                  \n                  DOI: 10.1021\/acs.joc.9b01149<\/a><\/span><\/span><\/div>\n
                  \"\"\r\n<\/span><\/span><\/pre>\n<\/li>\n
                5. \n
                  Ikeuchi, T.; Inuki, S.; Oishi, S.; Ohno, H.<\/span>
                  \nGold(I)-catalyzed cascade cyclization reactions of allenynes for the synthesis of fused cyclopropanes and acenaphthenes.
                  \nAngew. Chem. Int. Ed.<\/em> 2019<\/strong>, 58<\/em>, 7792\u20137796.
                  \n                  DOI: 10.1002\/anie.201903384<\/a><\/span><\/span><\/div>\n
                  \"\"<\/span><\/span><\/pre>\n<\/li>\n
                6. \n
                  Yamamoto, K.; Inuki, S.; Ohno, H.; Oishi, S.
                  \nScaffold hopping of fused piperidine-type NK3 receptor antagonists to reduce environmental impact.
                  \nBioorg. Med. Chem.<\/em> 2019<\/strong>, 27<\/em>, 2019\u20132026.
                  \n                  DOI: 10.1016\/j.bmc.2019.03.059<\/a><\/span><\/span><\/div>\n
                  \"\"<\/span><\/pre>\n<\/li>\n
                7. \n
                  Shu, K.; Iwamoto, N.; Honda, K.; Kondoh, Y.; Hirano, H.; Osada, H.; Ohno, H.; Fujii, N.; Oishi, S.
                  \nDevelopment of mirror-image screening systems for XIAP BIR3 domain inhibitors.
                  \nBioconjug. Chem.<\/em> 2019<\/strong>, 30, 1395\u20131404.
                  \n                  DOI: 10.1021\/acs.bioconjchem.9b00154<\/a><\/span><\/span><\/div>\n
                  \"\"<\/span><\/pre>\n<\/li>\n
                8. \n
                9. \n
                  Yamamoto, K.; Yoshikawa, Y.; Ohue, M.; Inuki, S.; Ohno, H.; Oishi, S.
                  \n<\/span><\/div>\n
                  Synthesis of triazolo- and oxadiazolo-piperazines by gold(I)-catalyzed domino cyclization: application to the design of a MAP kinase inhibitor.
                  \nOrg. Lett.<\/em> 2019<\/strong>, 21<\/em>, 373\u2013377.
                  \n                  DOI: 10.1021\/acs.orglett.8b03500<\/span><\/a>
                  \n<\/span><\/span><\/div>\n
                  \"\"<\/span><\/pre>\n<\/li>\n<\/ol>\n
                  <\/a>2018<\/span><\/h4>\n
                    \n
                  1. \n
                    Kawada, Y.; Ohmura, S.; Kobayashi, M.; Nojo, W.; Kondo, M.; Matsuda, Y.; Matsuoka, J.; Inuki, S.; Oishi, S.; Wang, C.; Saito, T.; Uchiyama, M.; Suzuki, T.; Ohno, H.
                    \nDirect synthesis of aryl-annulated [c]carbazoles by gold(I)-catalysed cascade reaction of azide-diynes and arenes.
                    \nChem. Sci.<\/em> 2018<\/strong>, 44<\/em>, 8416\u20138425.
                    \n                    DOI: <\/span>10.1039\/C8SC03525C<\/span><\/span><\/a><\/span><\/div>\n
                    \"\"<\/pre>\n<\/li>\n
                  2. \n
                    Hamada, N.; Yamaguchi, A.; Inuki, S.; Oishi, S.; Ohno, H.
                    \nGold(I)-Catalyzed Oxidative Cascade Cyclization of 1,4-Diyn-3-ones for the Construction of Tropone-Fused Furan Scaffolds.
                    \nOrg. Lett.<\/em>\u00a02018<\/strong>, 20<\/em>, 4401\u20134405.<\/span><\/div>\n
                    DOI: 10.1021\/acs.orglett.8b01524<\/a><\/span><\/div>\n
                    \"Abstract<\/pre>\n<\/li>\n
                  3. \n
                    Inuki, S.; Miyagawa, T.; Oishi, S.; Ohno, H.
                    \nIntroduction of a Polar Functional Group to the Lipid Tail of 4-epi<\/em>-Jaspine B Affects Sphingosine Kinase Isoform Selectivity.
                    \nChem. Pharm. Bull.<\/em> 2018<\/strong>, 66<\/em>, 866\u2013872.<\/span><\/div>\n
                    DOI: 10.1248\/cpb.c18-00366<\/span><\/a>
                    \n<\/span><\/div>\n
                    \"\"<\/pre>\n<\/li>\n
                  4. \n
                    Kaneda, M.; Kawaguchi, S.; Fujii, N.; Ohno, H.; Oishi, S.
                    \n<\/span>Structure\u2013Activity Relationship Study on Odoamide: Insights into the Bioactivities of Aurilide-Family Hybrid Peptide-Polyketides.
                    \n<\/span>ACS Med. Chem. Lett.<\/em> 2018<\/strong>, <\/span>9<\/em>, 365\u2013369.<\/span>
                    \n                    DOI: 10.1021\/acsmedchemlett.8b00028<\/a><\/span><\/div>\n
                    \"Abstract<\/span><\/span><\/pre>\n<\/li>\n
                  5. \n
                  6. \n
                  7. \n
                  8. \n
                  9. \n
                  10. \n
                  11. \n
                    Kaneda, M.; Inuki, S.; Ohno, H.; Oishi, S.
                    \nTotal Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide\u2013Polyketide Macrocycle.
                    \nJ. Org. Chem.<\/em> 2018<\/strong>, 83<\/em>, 3047\u20133060.
                    \n                    DOI: 10.1021\/acs.joc.8b00118<\/span><\/a><\/span><\/div>\n<\/li>\n<\/ol>\n
                    <\/a>2017<\/span><\/h4>\n
                      \n
                    1. \n
                    2. \n
                    3. \n
                    4. \n
                    5. \n
                    6. \n
                    7. \n
                    8. \n
                    9. \n
                    10. \n
                    11. \n
                      Yano, Y.; Kondo, K.; Watanabe, Y.; Zhang, T. O.; Ho, J. J.; Oishi, S.; Fujii, N.; Zanni, M. T.; Matsuzaki, K.
                      \nGXXXG-mediated parallel and antiparallel dimerization of transmembrane helices and its inhibition by cholesterol: single-pair FRET and 2D IR studies.
                      \nAngew. Chem. Int. Ed.<\/em> 2017<\/strong>, 56<\/em>, 1756\u20131759.
                      \n                      DOI: 10.1002\/anie.201609708<\/a><\/span><\/span><\/div>\n<\/li>\n<\/ol>\n
                      <\/a>2016<\/span><\/h4>\n
                        \n
                      1. Alam, M.; Kuwata, T.; Shimura, K.; Yokoyama, M.; Ramirez Valdez, K. P.; Tanaka, K.; Maruta, Y.; Oishi, S.; Fujii, N.; Sato, H.; Matsuoka, M.; Matsushita, S.
                        \nEnhanced antibody-mediated neutralization of HIV-1 variants that are resistant to fusion inhibitors.
                        \nRetrovirology.\u00a013<\/b>(1), 70, (2016)<\/span><\/li>\n
                      2. Sawada, J.; Osawa, A.; Takeuchi, T.; Kaneda, M.; Oishi, S.; Fujii, N.; Asai, A.; Tanino, K.; Namba, K.
                        \nFunctional 1,3a,6a-triazapentalene scaffold: Design of fluorescent probes for kinesin spindle protein (KSP).
                        \nBioorg. Med. Chem. Lett.\u00a026<\/b>(23) 5765-5769. (2016)\u00a0<\/span><\/li>\n
                      3. Watanabe, M.; Hashimoto, K.; Abe, Y.; Kodama, E.N.; Nabika, R.; Oishi, S.; Ohara, S.; Sato, M.; Kawasaki, Y.; Fujii, N.; Hosoya, M.
                        \nA novel peptide derived from the fusion protein heptad repeat inhibits replication of subacute sclerosing panencephalitis virus in vitro and in vivo.
                        \nPLoS One.\u00a011<\/b>(9) e0162823.\u00a0<\/span><\/li>\n
                      4. Hattori, Y.; Machida,Y.;Honda, M.;Ohno, H.;Fujii, N.;Onishi, H.
                        \nSmall interfering RNA delivery into the liver by cationic cholesterol derivative-based liposomes.
                        \nJ. Liposome Res. (2016)\u00a0<\/span><\/li>\n
                      5. Suzuki, T.; Nojo, W.; Sakano, Y.; Katoono, R.; Ishigaki, Y.; Ohno, H.; Fujiwara, K.
                        \nRedox-induced conformational changes in 1,3-propylene- and m-xylylenebis[5-(10-butyl-5,10-dihydrobenzo[a]indolo[2,3-c]carbazole)]: twin-BIC donors that form sandwich-like dimeric cations exhibiting NIR absorption.
                        \nChem. Lett.\u00a045<\/b>(7) 720-722. (2016)<\/span><\/li>\n
                      6. Kaneda, M.; Sueyoshi, K.; Teruya, T.; Ohno, H.; Fujii, N.; Oishi, S.
                        \nTotal synthesis of odoamide, a novel cyclic depsipeptide from an Okinawan marine cyanobacterium.
                        \nOrg. Biomol. Chem.\u00a014<\/b>(38) 9093-9104. (2016)\u00a0<\/span><\/li>\n
                      7. Abdelouahab, H.; Zhang, Y.; Wittner, M.; Oishi, S.; Fujii, N.; Besancenot, R.; Plo, I.; Ribrag, V.; Solary, E.; Vainchenker, W.; Barosi, G.; Louache, F.
                        \nCXCL12\/CXCR4 pathway is activated by oncogenic JAK2 in a PI3K-dependent manner.
                        \nOncotarget, DOI: 10.18632\/oncotarget.10789.\u00a0<\/span><\/li>\n
                      8. Sueyoshi, K.; Kaneda, M.; Sumimoto, S.; Oishi, S.; Fujii, N.; Suenaga, K.; Teruya, T.
                        \nOdoamide, a cytotoxic cyclodepsipeptide from the marine cyanobacterium Okeania sp.
                        \nTetrahedron,\u00a072<\/b>(35) 5472-5478. (2016)<\/span><\/li>\n
                      9. Naoe, S.; Yoshida, Y.; Oishi, S.; Fujii, N.; Ohno, H.<\/span>
                        \nTotal synthesis of (+)-conolidine by the gold(I)-catalyzed cascade cyclization of a conjugated enyne.<\/span>
                        \nJ. Org. Chem.\u00a081<\/b>(13) 5690-5698. (2016)\u00a0<\/span><\/span><\/li>\n
                      10. Yamamoto, K.; Okazaki, S.; Ohno, H.; Matsuda, F.; Ohkura, S.; Maeda, K.; Fujii, N.; Oishi, S.
                        \nDevelopment of novel NK3 receptor antagonists with reduced environmental impact.
                        \nBioorg. Med. Chem.\u00a024<\/b>(16) 3494-3500. (2016)\u00a0<\/span><\/li>\n
                      11. Noguchi, T.; Oishi, S.; Honda, K.; Kondoh, Y.; Saito, T.; Ohno, H.; Osada, H.; Fujii, N.
                        \nScreening of a virtual mirror-image library of natural products.
                        \nChem. Commun.\u00a052<\/b>(49) 7653-7656. (2016)\u00a0<\/span><\/li>\n
                      12. Kato, F.; Ishida, Y.; Oishi, S.; Fujii, N.; Watanabe, S.; Vasudevan, S. G.; Tajima, S.; Takasaki, T.; Suzuki, Y.; Ichiyama, K.; Yamamoto, N.; Yoshii, K.; Takashima, I.; Kobayashi, T.; Miura, T.; Igarashi, T.; Hishiki, T.
                        \nNovel antiviral activity of bromocriptine against dengue virus replication.
                        \nAntiviral Res.\u00a0<\/i><\/i>131<\/b> 141-147. (2016)\u00a0<\/span><\/li>\n
                      13. Nishiyama, D.; Sakai, Y.; Sekiguchi, H.; Chiba, H.; Misu, R.; Oishi, S.; Fujii, N.; Ohno, H.
                        \nNovel 3,4,7-substituted benzofuran derivatives having binding affinity to \u03ba-opioid receptor.
                        \nChem. Pharm. Bull.\u00a064<\/b>(7) 996-1003. (2016)\u00a0<\/span><\/li>\n
                      14. Nishiyama, D.; Ohara, A.; Chiba, H.; Kumagai, H.; Oishi, S.; Fujii, N.; Ohno, H.
                        \nFormal total synthesis of (\u00b1)-strictamine based on a gold-catalyzed cyclization.
                        \nOrg. Lett.\u00a018<\/b>(7) 1670-1673. (2016)\u00a0<\/span><\/li>\n
                      15. Ohno, H.; Minamiguchi, D.; Nakamura, S.; Shu, K.; Okazaki, S.; Honda, M.; Misu, R.; Moriwaki, H.; Nakanishi, S.; Oishi, S.; Kinoshita, T.; Nakanishi, I.; Fujii, N.
                        \nStructure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitors.
                        \nBioorg. Med. Chem.\u00a024<\/b>(5) 1136-1141. (2016)\u00a0<\/span><\/li>\n
                      16. Wagner, B.; Hiller, W.; Ohno, H.; Krause, N.
                        \nGold-catalyzed three-component spirocyclization: a one-pot approach to functionalized pyrazolidines.
                        \nOrg. Biomol. Chem.\u00a014<\/b>(5) 1579-1583. (2016)\u00a0<\/span><\/li>\n<\/ol>\n
                        <\/a>2015<\/span><\/h4>\n
                          \n
                        1. \n
                          Shi, J.; Liu, N.; Xiao, Y.; Takei, Y.; Yasue, M.; Suzuki, Y.; Hou, Z.; Ohno, H.; Tsujimoto, G.; Hirasawa, A.
                          \n<\/i><\/i>The effects of a selective CK2 inhibitor on anti-glomerular basement membrane glomerulonephritis in rats.
                          \nBiol. Pharm. Bull<\/em>.\u00a038<\/b>(9) 1345\u20131351. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        2. \n
                          Miyamoto, F.; Kawaji, K.; Oishi, S.; Fujii, N.; Kaku, M.; Kodama, E. N.
                          \nAnti-HIV-1 activity determined by \u03b2-galactosidase activity in the multinuclear activation of an indicator assay is comparable with that by a conventional focus counting method.
                          \nAntivir. Chem. Chemother<\/em>.\u00a024<\/b> 77\u201382. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        3. \n
                          Taguchi, M.; Tokimizu, Y.; Oishi, S.; Fujii, N.; Ohno, H.
                          \nSynthesis of fused carbazoles by gold-catalyzed tricyclization of conjugated diynes via rearrangement of an \u039d-propargyl group.
                          \nOrg. Lett.\u00a017<\/b>(24) 6250\u20136253. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        4. \n
                          Umatani, C.; Misu, R.; Oishi, S.; Yamaguchi, K.; Abe, H.; Oka, Y.
                          \nGnRH suppresses excitability of visual-processing neurons in the optic tectum.
                          \nJ<\/em>. Neurophysiol.<\/em>\u00a0114<\/b>(5) 2775\u20132784. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        5. \n
                          Shimura, K.; Miyazato, P.; Oishi, S.; Fujii, N.; Matsuoka, M.
                          \n<\/i><\/i>Impact of HIV-1 infection pathways on susceptibility to antiviral drugs and on virus spread.
                          \nVirology<\/em>\u00a0484<\/b> 364\u2013376. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        6. \n
                          Oishi, S.; Kuroyanagi, T.; Kubo, T.; Montpas, N.; Yoshikawa, Y.; Misu, R.; Kobayashi, Y.; Ohno, H.; Heveker, N.; Furuya, T.; Fujii, N.
                          \nDevelopment of novel CXC chemokine receptor 7 (CXCR7) ligands: selectivity switch from CXCR4 antagonists with a cyclic pentapeptide scaffold.
                          \nJ<\/em>. Med<\/em>. Chem<\/em>.\u00a058<\/b>(13) 5218\u20135225. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        7. \n
                          Iwata, A.; Inuki, S.; Oishi, S.; Fujii, N.; Ohno, H.
                          \n<\/span><\/span><\/div>\n
                          C<\/span>onvenient synthesis of spiroindole derivatives via palladium-catalyzed cyclization of propargyl chlorides.
                          \n<\/span>Tetrahedron<\/em> 71<\/b>(37) 6580\u20136585. (2015)<\/span>
                          \n<\/b><\/span><\/div>\n<\/li>\n
                        8. \n
                          Takenaga, M.; Yamamoto, Y.; Takeuchi, T.; Ohta, T; Tokura, Y.; Hamaguchi, A.; Asai, D.; Nakashima, H.; Oishi, S.; Fujii, N.
                          \nPotential new chemotherapy strategy for human ovarian carcinoma with a novel KSP inhibitor.
                          \nBiochem. Biophys. Res. Commun.\u00a0463<\/b>(3) 222\u2013228. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        9. \n
                          Tokimizu, Y.; Oishi, S.; Fujii, N.; Ohno, H.
                          \nGold-catalyzed cascade cyclization of 2-alkynyl-N-propargylanilines via the rearrangement of a propargyl group.
                          \nAngew. Chem. Int. Ed.\u00a054<\/b>(27) 7862\u20137866. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        10. \n
                          Naoe, S.; Saito, T.; Uchiyama, M.; Oishi, S.; Fujii, N.; Ohno, H.
                          \nDirect construction of fused indoles by gold-catalyzed cascade cyclization of conjugated diynes.
                          \nOrg. Lett.\u00a017<\/b>(7) 1774\u20131777. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        11. \n
                          Yasuda, Y.; Arakawa, T.; Nawata, Y.; Shimada, S.; Oishi, S.; Fujii, N.; Nishimura, S.; Hattori, A.; Kakeya, H.
                          \nDesign, synthesis, and structure-activity relationships of 1-ethylpyrazole-3-carboxamide compounds as novel hypoxia-inducible factor (HIF)-1 inhibitors.
                          \nBioorg. Med. <\/i><\/i>Chem.\u00a023<\/b>(8) 1776\u20131787. (2015)<\/span><\/div>\n<\/li>\n
                        12. \n
                          Montpas, N.; Cabana, J.; St-Onge, G.; Gravel, S.; Morin, G.; Kuroyanagi, T.; Lavigne, P.; Fujii, N.; Oishi, S.; Heveker, N.
                          \nThe binding mode of the cyclic agonist peptide TC14012 to CXCR7 - Identification of receptor and compound determinants.
                          \nBiochemistry\u00a054<\/b>(7) 1505\u20131515. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        13. \n
                          Okazaki, S.; Oishi, S.; Mizuhara, T.; Shimura, K.; Murayama, H.; Ohno, H.; Matsuoka, M.; Fujii, N.
                          \nInvestigations of possible prodrug structures for 2-(2-mercaptophenyl)tetrahydropyrimidines: reductive conversion from anti-HIV agents with pyrimidobenzothiazine and isothiazolopyrimidine scaffolds.
                          \nOrg. Biomol. Chem.\u00a013<\/b>(16) 4706\u20134713. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        14. \n
                          Hattori, Y.; Hara, E.; Shingu, Y.; Minamiguchi, D.; Nakamura, A.; Arai, S.; Ohno, H.; Kawano, K.; Fujii, N.; Yonemochi, E.<\/span>
                          \nsiRNA delivery into tumor cells by cationic cholesterol derivative-based nanoparticles and liposomes.<\/span>
                          \nBiol. Pharm. Bull.\u00a038<\/b>(1) 30\u201338. (2015)<\/span><\/span><\/div>\n<\/li>\n
                        15. \n
                          Okazaki, S.; Mizuhara, T.; Shimura, K.; Murayama, H.; Ohno, H.; Oishi, S.; Matsuoka, M.; Fujii, N.
                          \nIdentification of anti-HIV agents with a novel benzo[4,5]isothiazolo[2,3-a]pyrimidine scaffold.
                          \nBioorg. Med. Chem.\u00a023<\/b>(7) 1447\u20131452. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        16. \n
                          Kawabata, H.; Uchiyama, T.; Sakamoto, S.; Kanda, J.; Oishi, S.; Fujii, F.; Tomosugi, N.; Kadowaki, N.; Takaori-Kondo, A.
                          \nA HAMP promoter bioassay system for identifying chemical compounds that modulate hepcidin expression.
                          \nExp. Hematol.\u00a043<\/b>(5) 404\u2013413. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        17. \n
                          Tokimizu, Y.; Wieteck, M.; Rudolph, M.; Oishi, S.; Fujii, N.; Hashmi, A. S. K.; Ohno, H.
                          \n<\/i><\/i>Dual gold catalysis: a novel synthesis of bicyclic and tricyclic pyrroles from N-propargyl ynamides.
                          \nOrg. Lett.\u00a017<\/b>(3) 604\u2013607. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        18. \n
                          Misu, R.; Yamamoto, K.; Yamada, A.; Noguchi, T.; Ohno, H.; Yamamura, T.; Okamura, H.; Matsuda, F.; Ohkura, S.; Oishi, S.; Fujii, N.
                          \nStructure-activity relationship study on senktide for development of novel potent neurokinin-3 receptor selective agonists.
                          \nMedChemCommun.\u00a06<\/b>(3) 469\u2013476. (2015)<\/b><\/span><\/div>\n<\/li>\n
                        19. \n
                          Tsunematsu, Y.; Nishimura, S.; Hattori, A.; Oishi, S.; Fujii, N.; Kakeya, H.
                          \nIsolation, structure elucidation and total synthesis of tryptopeptins A and B, new TGF-beta signaling modulators from Streptomyces sp.
                          \nOrg. Lett.\u00a017<\/b>(2) 258\u2013261. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        20. \n
                          Nabika, R.; Suyama, T. L.; Hau, A. M.; Misu, R.; Ohno, H.; Ishmael, J. E.; McPhail, K. L.; Oishi, S.; Fujii, N.
                          \nSynthesis and biological evaluation of the [D-MeAla11]-epimer of coibamide A.
                          \nBioorg. Med. Chem. Lett.\u00a025<\/b>(2) 302\u2013306. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        21. \n
                          Matsuda, Y.; Naoe, S.; Oishi, S.; Fujii, N.; Ohno, H.
                          \nFormal [4+2] reaction between 1,3-diynes and pyrroles: gold(I)-catalyzed indole synthesis by double hydroarylation.
                          \nChem. Eur. J.<\/em>\u00a021<\/b>(4) 1463\u20131467. (2015)\u00a0<\/span><\/div>\n<\/li>\n
                        22. \n
                          Zenda, M.; Yasui, H.; Oishi, S.; Masuda, R.; Fujii, N.; Koide, T.
                          \n<\/span><\/span>A cisplatin derivative that inhibits collagen fibril-formation in vitro.
                          \n<\/span>Chem. Biol. Drug Des<\/em>.\u00a085<\/b>(5) 519\u2013526. (2015)<\/span><\/div>\n<\/li>\n<\/ol>\n
                          <\/a><\/i>2014<\/span><\/h4>\n
                            \n
                          1. \n
                            Wieteck, M.; Tokimizu, Y.; Rudolph, M.; Rominger, F.; Ohno, H.; Fujii, N.; Hashmi, A. S.
                            \nDual gold catalysis: synthesis of polycyclic compounds via C-H insertion of gold vinylidenes.
                            \nChem. Eur. J.\u00a020<\/b>(49) 16331-16336. (2014)\u00a0<\/span><\/div>\n<\/li>\n
                          2. \n
                            Misu, R.; Oishi, S.; Yamada, A.; Yamamura, T.; Matsuda, F.; Yamamoto, K.; Noguchi, T.; Ohno, H.; Okamura, H.; Ohkura, S.; Fujii, N.
                            \n<\/i><\/i>Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation.
                            \nJ. Med. Chem.\u00a057<\/b>(20) 8646-8651. (2014)\u00a0<\/span><\/div>\n<\/li>\n
                          3. \n
                            Nabika, R.; Oishi, S.; Misu, R.; Ohno, H.; Fujii, N.
                            \nSynthesis of IB-01212 by multiple N-methylations of peptide bonds.
                            \nBioorg. Med. Chem.\u00a022<\/b>(21) 6156-6162. (2014)\u00a0<\/span><\/div>\n<\/li>\n
                          4. \n
                            Tokimizu, Y.; Oishi, S.; Fujii, N.; Ohno, H.
                            \nGold-catalyzed cascade cyclization of (azido)ynamides: an efficient strategy for the construction oflndoloquinolines.
                            \nOrg. Lett.\u00a016<\/b>(11) 3138-3141. (2014)\u00a0<\/span><\/div>\n<\/li>\n
                          5. \n
                            Tsutsui, A.; Imamaki, R.; Kitazume, S.; Hanashima, S.; Yamaguchi, Y.; Kaneda, M.; Oishi, S.; Fujii, N.; Taniguchi, N.; Tanaka, K.
                            \nPolyamine modification by acrolein exclusively produces 1,5-diazacyclooctanes: a previously unrecognized mechanism for acrolein-mediated oxidative stress.
                            \n<\/i><\/i>Org. Biomol. Chem.\u00a012<\/b>(28) 5151-5157. (2014)\u00a0<\/span><\/div>\n<\/li>\n
                          6. \n
                            Suzuki, T.; Sakano, Y.; Tokimizu, Y.; Miura, Y.; Katoono, R.; Fujiwara, K.; Yoshioka, N.; Fujii, N.; Ohno, H.
                            \nWurster's blue-type cation radicals framed in a 5,10-dihydrobenzo[a]indolo[2,3-c]carbazole (BIC) skeleton: dual electrochromism with drastic changes in UV-Vis-NIR and fluorescence.
                            \nChem. Ajian J.\u00a09<\/b>(7) 1841-1846. (2014)\u00a0<\/span><\/div>\n<\/li>\n
                          7. \n
                            Graf, K.; Hindenberg, P.D.; Tokimizu,Y.; Naoe, S.; Rudolph, M.; Rominger, F.; Ohno, H.; Hashmi, A.S.K.
                            \nThe role of acetylides in dual gold catalysis: a mechanistic investigation of the selectivity difference in the naphthalene synthesis from diynes.
                            \nChemCatChem\u00a06<\/b>(1), 199-204. (2014)<\/span><\/div>\n<\/li>\n
                          8. \n
                            Kaneda, M.; Misu, R.; Ohno, H.; Hirasawa, A.; Ieda, N.; Uenoyama, Y.; Tsukamura, H.; Maeda, K.; Oishi, S.; Fujii, N.
                            \nDesign and synthesis of fluorescent probes for GPR54.
                            \nBioorg. Med. Chem.\u00a022<\/b>(13) 3325-3330. (2014)\u00a0<\/span><\/div>\n<\/li>\n
                          9. \n
                            Takeuchi, T.; Oishi, S.; Kaneda, M.; Misu, R.; Ohno, H.; Sawada, J.; Asai, A.; Nakamura, S.; Nakanishi, I.; Fujii, N.
                            \nOptimization of diaryl amine derivatives as kinesin spindle protein inhibitors.
                            \nBioorg. Med. Chem.\u00a022<\/b>(12) 3171-3179. (2014)\u00a0<\/span><\/div>\n<\/li>\n
                          10. \n
                            Takeuchi, T.; Oishi, S.; Kaneda, M.; Ohno, H.; Nakamura, S.; Nakanishi, I.; Yamane, M.; Sawada, J.; Asai, A.; Fujii, N.
                            \nKinesin spindle protein inhibitors with diaryl amine scaffolds: crystal packing analysis for improved aqueous solubility.
                            \nACS Med. Chem. Lett.\u00a05<\/b>(5) 566-571. (2014)\u00a0<\/span><\/div>\n<\/li>\n
                          11. \n
                            Sano, K.; Masuda, R.; Hisada,H.; Oishi, S.; Shimokawa, K.; Ono, M.; Fujii, N.; Saji, H.; Mukai, T.
                            \nA radiogallium-DOTA-based bivalent peptidic ligand targeting a chemokine receptor, CXCR4, for tumor imaging.
                            \nBioorg. Med. Chem. Lett.\u00a024<\/b>(5) 1386-1388. (2014)\u00a0<\/span><\/div>\n<\/li>\n
                          12. \n
                            Iwata, A.; Inuki, S.; Oishi, S.; Fujii, N.; Ohno, H.
                            \nSynthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation.
                            \nChem. Commun.<\/i><\/i> 2014<\/strong>, 50<\/em>, 298\u2013300.<\/span><\/div>\n<\/li>\n<\/ol>\n","protected":false},"excerpt":{"rendered":"
                            [2026][2025][2024][2023][2022][2021][2020][2019][2018][2017][2016][2015] [2014] [2013\u4ee5\u524d] 2026 Fujii, T.; Araki […]<\/p>\n","protected":false},"author":47,"featured_media":0,"parent":0,"menu_order":18,"comment_status":"closed","ping_status":"closed","template":"","meta":{"_acf_changed":false,"footnotes":""},"class_list":["post-219","page","type-page","status-publish","hentry"],"acf":[],"_links":{"self":[{"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/souyaku\/index.php?rest_route=\/wp\/v2\/pages\/219","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/souyaku\/index.php?rest_route=\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/souyaku\/index.php?rest_route=\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/souyaku\/index.php?rest_route=\/wp\/v2\/users\/47"}],"replies":[{"embeddable":true,"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/souyaku\/index.php?rest_route=%2Fwp%2Fv2%2Fcomments&post=219"}],"version-history":[{"count":6,"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/souyaku\/index.php?rest_route=\/wp\/v2\/pages\/219\/revisions"}],"predecessor-version":[{"id":2736,"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/souyaku\/index.php?rest_route=\/wp\/v2\/pages\/219\/revisions\/2736"}],"wp:attachment":[{"href":"https:\/\/www.pharm.kyoto-u.ac.jp\/souyaku\/index.php?rest_route=%2Fwp%2Fv2%2Fmedia&parent=219"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}